KEGG   DRUG: Barzolvolimab
Entry
D12409                      Drug                                   
Name
Barzolvolimab (USAN/INN)
Formula
C6436H9922N1708O2011S38
Exact mass
144529.6024
Mol weight
144618.3529
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKL SCKASGYTFT DYYINWVRQA PGKGLEWIAR IYPGSGNTYY
NEKFKGRATL TADKSTSTAY MQLSSLRSED TAVYFCARGV YYFDYWGQGT TVTVSSASTK
GPSVFPLAPS SKSTSGGTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTQTYICN VNHKPSNTKV DKKVEPKSCD KTHTCPPCPA PEAQGGPSVF
LFPPKPKDTL YITREPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP REEQYNSTYR
VVSVLTVLHQ DWLNGKEYKC QVSNKALPAP IEKTISKAKG QPREPQVYTL PPSRDELTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPG
(Light chain)
DIVMTQSPSS LSASVGDRVT ITCKASQNVR TNVAWYQQKP GKAPKALIYS ASYRYSGVPD
RFTGSGSGTD FTLTISSLQP EDFADYFCQQ YNSYPRTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H143-H199, H219-L214, H225-H'225, H228-H'228, H260-H320, H366-H424, H'22-H'96, H'143-H'199, H'219-L'214, H'260-H'320, H'366-H'424, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Immunomodulator, Anti-KIT antibody
  Type
Monoclonal antibody
Comment
Treatment of chronic urticaria
Target
KIT (CD117) [HSA:3815] [KO:K05091]
  Pathway
hsa04010  MAPK signaling pathway
hsa04072  Phospholipase D signaling pathway
hsa04151  PI3K-Akt signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Protein kinases
  Receptor tyrosine kinases (RTK)
   PDGFR family
    KIT (CD117)
     D12409  Barzolvolimab (USAN/INN)
Other DBs
CAS: 2438203-51-9
LinkDB

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