KEGG   DGROUP: Regorafenib
Entry
DG00720                     DGroup                                 
Name
Regorafenib
Type
Chemical
Member
D10138  
Regorafenib (USAN/INN)
D10137  
Regorafenib hydrate (JAN)  <JP/US>
Class
Antineoplastic
 DG01918  Tyrosine kinase inhibitor
  DG01917  Receptor tyrosine kinase inhibitor
Metabolizing enzyme substrate
 DG01633  CYP3A/CYP3A4 substrate
  DG02913  CYP3A4 substrate
 DG02924  UGT substrate
  DG03188  UGT1A9 substrate
Transporter substrate
 DG01665  ABCB1 substrate
 DG01913  ABCG2 substrate
Remark
ATC code: L01EX05
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