KEGG   DGROUP: CYP3A/CYP3A4 substrate
Entry
DG01633                     DGroup                                 
Name
CYP3A/CYP3A4 substrate
Type
Metabolism
Member
CYP3A4 substrate
 DG00011  
Dexamethasone
  D00292  
Dexamethasone (JP18/USP/INN)  <JP/US>
  D00975  
Dexamethasone sodium phosphate (JAN/USP)  <JP/US>
  D01510  
Dexamethasone metasulfobenzoate sodium (JAN)  <JP>
  D01615  
Dexamethasone palmitate (JAN)  <JP>
  D01632  
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN)  <JP>
  D01948  
Dexamethasone valerate (JAN)  <JP>
  D02174  
Dexamethasone acetate (JAN/USP)
  D02591  
Dexamethasone acefurate (USAN/INN)
  D02592  
Dexamethasone beloxil (USAN)
  D07073  
Dexamethasone cipecilate (JAN/INN)  <JP>
  D07796  
Dexamethasone 21-acetate
  D07797  
Dexamethasone isonicotinate
  D07798  
Dexamethasone sodium hemisulfate
  D07799  
Dexamethasone 21-tebutate
  D07800  
Dexamethasone 21-valerate
  D07801  
Dexamethasone phenylpropionate
  D07802  
Dexamethasone phosphate
 D01131  
Lafutidine (JP18/INN)  <JP>
 DG00020  
Omeprazole
  D00455  
Omeprazole (JP18/USP/INN)  <JP/US>
  D01207  
Omeprazole sodium (USAN)
  D05261  
Omeprazole sodium injection (JAN)  <JP>
  D05259  
Omeprazole magnesium (USP)  <US>
 DG00021  
Pantoprazole
  D05353  
Pantoprazole (USAN/INN)
  D02593  
Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN)  <US>
 D00355  
Lansoprazole (JP18/USP/INN)  <JP/US>
 DG00022  
Rabeprazole
  D08463  
Rabeprazole (INN)
  D00724  
Rabeprazole sodium (JP18/USP)  <JP/US>
 DG00023  
Esomeprazole
  D07917  
Esomeprazole (INN)
  D01984  
Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN)  <JP/US>
  D04056  
Esomeprazole sodium (USAN)  <US>
  D09339  
Esomeprazole potassium (USAN)
  D10120  
Esomeprazole strontium (USAN)  <US>
  D11114  
Esomeprazole magnesium dihydrate  <US>
 DG03298  
Dexlansoprazole
  D08903  
Dexlansoprazole (INN/USAN)  <US>
  D12816  
Dexlansoprazole sesquihydrate  <US>
 DG03104  
Vonoprazan
  D11784  
Vonoprazan (USAN/INN)
  D10466  
Vonoprazan fumarate (JAN/USAN)  <JP/US>
 D09742  
Lansoprazole, amoxicillin hydrate and metronidazole
 D10246  
Omeprazole, clarithromycin and amoxicillin  <US>
 D08774  
Amoxicillin hydrate, clarithromycin and lansoprazole  <US>
 D10519  
Rabeprazole, amoxicillin and clarithromycin  <JP>
 D10520  
Rabeprazole, amoxicillin and metronidazole  <JP>
 D10775  
Vonoprazan, amoxicillin and clarithromycin  <JP>
 D10774  
Vonoprazan, amoxicillin and metronidazole  <JP>
 D01121  
Rebamipide (JP18/INN)  <JP>
 DG00046  
Alosetron
  D07129  
Alosetron (INN)
  D02829  
Alosetron hydrochloride (USAN)  <US>
 DG00057  
Domperidone
  D01745  
Domperidone (JP18/USAN/INN)  <JP>
  D07868  
Domperidone maleate
 DG01285  
Mosapride
  D01994  
Mosapride citrate hydrate (JP18)  <JP>
  D08236  
Mosapride (INN)
 DG00060  
Ondansetron
  D00456  
Ondansetron (JAN/USP/INN)  <US>
  D00678  
Ondansetron hydrochloride hydrate (JAN/USP)  <JP/US>
 DG00061  
Granisetron
  D04370  
Granisetron (JAN/USAN/INN)  <US>
  D00677  
Granisetron hydrochloride (JAN/USP)  <JP/US>
 DG00064  
Palonosetron
  D07175  
Palonosetron (INN)
  D05343  
Palonosetron hydrochloride (JAN/USP)  <JP/US>
 D10572  
Fosnetupitant and palonosetron hydrochloride  <US>
 DG00066  
Aprepitant
  D02968  
Aprepitant (JAN/USP/INN)  <JP/US>
  D10895  
Fosaprepitant (INN)
  D06597  
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN)  <JP/US>
 DG01868  
Rolapitant
  D10742  
Rolapitant (USAN/INN)
  D08988  
Rolapitant hydrochloride (USAN)  <US>
 DG01342  
Naldemedine
  D10188  
Naldemedine (USAN/INN)
  D10478  
Naldemedine tosylate (JAN/USAN)  <JP/US>
 DG03072  
Tenapanor
  D11652  
Tenapanor (USAN/INN)
  D11653  
Tenapanor hydrochloride (JAN/USAN)  <JP/US>
 D02554  
Rifaximin (JAN/USAN/INN)  <JP/US>
 DG00092  
Loperamide
  D08144  
Loperamide (INN)
  D00729  
Loperamide hydrochloride (JAN/USP)  <JP/US>
  D07113  
Loperamide oxide (INN)
 D00246  
Budesonide (JP18/USP/INN)  <JP/US>
 D00689  
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18)  <JP/US>
 D11572  
Beclomethasone dipropionate monohydrate  <US>
 DG00103  
Fenfluramine
  D07945  
Fenfluramine (INN)
  D04148  
Fenfluramine hydrochloride (JAN/USAN)  <JP/US>
 D11710  
Phentermine and topiramate  <US>
 D00336  
Glyburide (USP); Glibenclamide (JP18/INN)  <JP/US>
 D10263  
Metformin hydrochloride and saxagliptin hydrochloride  <US>
 DG00119  
Saxagliptin
  D08996  
Saxagliptin (USAN/INN)
  D09753  
Saxagliptin hydrate (JAN)  <JP>
  D10262  
Saxagliptin hydrochloride  <US>
 DG01283  
Teneligliptin
  D08616  
Teneligliptin (INN)
  D09756  
Teneligliptin hydrobromide hydrate (JAN)  <JP>
  D11968  
Teneligliptin hydrobromide (JAN)
 D10669  
Sotagliflozin (USAN/INN)  <US>
 D00594  
Repaglinide (JAN/USP/INN)  <JP/US>
 DG00148  
Eliglustat
  D09893  
Eliglustat (USAN/INN)
  D09894  
Eliglustat tartrate (JAN/USAN)  <JP/US>
 DG00155  
Clopidogrel
  D07729  
Clopidogrel (USP/INN)
  D00769  
Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18)  <JP/US>
  D10823  
Clopidogrel hydrochloride
  D10824  
Clopidogrel besilate
 D01896  
Cilostazol (JP18/USP/INN)  <JP/US>
 DG01349  
Vorapaxar
  D09765  
Vorapaxar (USAN/INN)
  D09766  
Vorapaxar sulfate (JAN/USAN)
 D09994  
Selexipag (JAN/USAN/INN)  <JP/US>
 D10513  
Clopidogrel sulfate and aspirin  <JP>
 D10527  
Acetylsalicylic acid and lansoprazole  <JP>
 DG00163  
Argatroban
  C04931  
Argatroban
  D00181  
Argatroban (USP); Argatroban hydrate (JP18)  <JP/US>
 D07086  
Rivaroxaban (JAN/USAN/INN)  <JP/US>
 D03213  
Apixaban (JAN/USAN/INN)  <JP/US>
 DG01976  
Avatrombopag
  D10306  
Avatrombopag (USAN/INN)
  D10307  
Avatrombopag maleate (JAN/USAN)  <JP/US>
 DG01419  
Fostamatinib
  D09347  
Fostamatinib (USAN)
  D09348  
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN)  <JP/US>
 D11330  
Voxelotor (USAN)  <US>
 DG00194  
Disopyramide
  D00303  
Disopyramide (JP18/USAN/INN)  <JP>
  D00637  
Disopyramide phosphate (JAN/USP)  <JP/US>
 DG00196  
Lidocaine
  D00358  
Lidocaine (JP18/USP/INN)  <JP/US>
  D02086  
Lidocaine hydrochloride (JAN/USP)  <JP/US>
  D08127  
Lidocaine hydrochloride monohydrate  <JP/US>
 DG00200  
Propafenone
  D08435  
Propafenone (INN)
  D00640  
Propafenone hydrochloride (JP18/USP)  <JP/US>
 DG00204  
Amiodarone
  D02910  
Amiodarone (USAN/INN)
  D00636  
Amiodarone hydrochloride (JP18/USP)  <JP/US>
 DG00209  
Cibenzoline
  D03492  
Cifenline (USAN); Cibenzoline (INN)
  D01455  
Cifenline succinate (USAN); Cibenzoline succinate (JP18)  <JP>
 DG00246  
Ivabradine
  D07165  
Ivabradine (USAN/INN)
  D08095  
Ivabradine hydrochloride (JAN/USAN)  <JP/US>
 D12265  
Mavacamten (JAN/USAN/INN)  <US>
 DG00250  
Guanfacine
  D08031  
Guanfacine (INN)
  D00606  
Guanfacine hydrochloride (JAN/USP)  <JP/US>
 DG00266  
Bosentan
  D07538  
Bosentan (INN)
  D01227  
Bosentan (USAN); Bosentan hydrate (JAN)  <JP/US>
 D10135  
Macitentan (JAN/USAN)  <JP/US>
 D01115  
Eplerenone (JP18/USAN/INN)  <JP/US>
 D10633  
Finerenone (JAN/USAN/INN)  <JP/US>
 D01213  
Tolvaptan (JAN/USAN/INN)  <JP/US>
 DG01977  
Dihydroergotoxine
  D07839  
Dihydroergotoxine
  D02268  
Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18)
 DG00331  
Diltiazem
  D07845  
Diltiazem (INN)
  D00616  
Diltiazem hydrochloride (JP18/USP)  <JP/US>
  D03830  
Diltiazem malate (USAN)
 DG00321  
Carvedilol
  D00255  
Carvedilol (JP18/USP/INN)  <JP/US>
  D03415  
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN)  <US>
 DG00322  
Amlodipine
  D07450  
Amlodipine (USP/INN)
  D00615  
Amlodipine besylate (USP); Amlodipine besilate (JP18)  <JP/US>
  D02914  
Amlodipine maleate (USAN)
  D11881  
Amlodipine benzoate  <US>
 D00319  
Felodipine (JP18/USP/INN)  <JP/US>
 DG00323  
Nicardipine
  D08270  
Nicardipine (INN)
  D00617  
Nicardipine hydrochloride (JP18/USAN)  <JP/US>
 D00437  
Nifedipine (JP18/USP/INN)  <JP/US>
 D00438  
Nimodipine (USP/INN)  <US>
 D00618  
Nisoldipine (JAN/USAN/INN)  <US>
 D00629  
Nitrendipine (JP18/USAN/INN)  <JP>
 D01908  
Nilvadipine (JP18/USAN/INN)  <JP>
 DG00324  
Manidipine
  D08155  
Manidipine (INN)
  D01553  
Manidipine hydrochloride (JP18)  <JP>
 DG00325  
Barnidipine
  D07494  
Barnidipine (INN)
  D01104  
Barnidipine hydrochloride (JAN)  <JP>
 D01173  
Cilnidipine (JP18/INN)  <JP>
 DG00327  
Benidipine
  D07509  
Benidipine (INN)
  D02045  
Benidipine hydrochloride (JP18)  <JP>
 DG00329  
Verapamil
  D02356  
Verapamil (USAN/INN)
  D00619  
Verapamil hydrochloride (JP18/USP)  <JP/US>
 DG00333  
Bepridil
  D07520  
Bepridil (INN)
  D00631  
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN)  <JP>
 D09745  
Valsartan and amlodipine besilate  <JP/US>
 D09743  
Telmisartan and amlodipine besilate (JP18)  <JP/US>
 D10243  
Irbesartan and amlodipine besilate (JP18)  <JP>
 D07569  
Candesartan cilexetil and anmlodipine besylate (JP18)  <JP>
 D10805  
Telmisartan, amlodipine and hydrochlorothiazide  <JP>
 DG00352  
Aliskiren
  D03208  
Aliskiren (USAN/INN)
  D06412  
Aliskiren fumarate (JAN/USAN)  <JP/US>
 D00434  
Simvastatin (JP18/USP/INN)  <JP/US>
 D00359  
Lovastatin (USP/INN)  <US>
 DG00354  
Fluvastatin
  D07983  
Fluvastatin (INN)
  D00892  
Fluvastatin sodium (JAN/USP)  <JP/US>
 DG00355  
Atorvastatin
  D07474  
Atorvastatin (INN)  <US>
  D00887  
Atorvastatin calcium anhydorous
  D02258  
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18)  <JP/US>
  D11095  
Atorvastatin calcium propylene glycol solvate  <US>
 DG00356  
Cerivastatin
  D07661  
Cerivastatin (INN)
  D00889  
Cerivastatin sodium (JAN/USAN)
 DG00362  
Lomitapide
  D09637  
Lomitapide (USAN/INN)
  D09638  
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN)  <JP/US>
 D10385  
Ezetimibe and atorvastatin  <JP/US>
 D08488  
Amlodipine besilate and atorvastatin calcium  <JP/US>
 D00351  
Ketoconazole (JP18/USP)  <JP/US>
 DG00375  
Terbinafine
  D02375  
Terbinafine (USAN/INN)
  D02219  
Terbinafine hydrochloride (JP18/USP)  <JP/US>
 D05744  
Roflumilast (JAN/USAN/INN)  <US>
 D09544  
Ozenoxacin (JAN/USAN/INN)  <JP/US>
 DG00410  
Methylprednisolone
  D00407  
Methylprednisolone (JP18/USP/INN)  <JP/US>
  D00751  
Methylprednisolone sodium succinate (JAN/USP)  <JP/US>
  D00979  
Methylprednisolone acetate (JAN/USP)  <JP/US>
  D05000  
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18)
  D05001  
Methylprednisolone sodium phosphate (USAN)
  D05002  
Methylprednisolone suleptanate (USAN/INN)
  D07203  
Methylprednisolone aceponate (INN)
 DG00419  
Mometasone
  D08227  
Mometasone (INN)
  D00690  
Mometasone furoate (JAN/USP)  <JP/US>
  D03325  
Mometasone furoate hydrate (JAN)  <JP/US>
 DG00420  
Fluticasone
  D07981  
Fluticasone (INN)
  D01708  
Fluticasone propionate (JAN/USP)  <JP/US>
  D06315  
Fluticasone furoate (JAN/USAN/INN)  <JP/US>
 D00592  
Dapsone (USP); Diaphenylsulfone (JAN)  <JP/US>
 DG00439  
Tacrolimus
  D08556  
Tacrolimus (INN)
  D00107  
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18)  <JP/US>
 DG00719  
Ruxolitinib
  D09959  
Ruxolitinib (USAN/INN)
  D09960  
Ruxolitinib phosphate (JAN/USAN)  <JP/US>
 D00321  
Finasteride (JAN/USP/INN)  <JP/US>
 D00804  
Ivermectin (JAN/USP/INN)  <JP/US>
 DG00974  
Caffeine
  D00528  
Caffeine (USP); Anhydrous caffeine (JP18)  <JP>
  D01453  
Caffeine hydrate (JP18)  <JP>
  D07603  
Caffeine citrate (USP)  <US>
 DG00445  
Methylergometrine
  D08207  
Methylergometrine (INN)
  D00680  
Methylergonovine maleate (USP); Methylergometrine maleate (JP18)  <JP/US>
 DG00834  
Ergotamine
  D07906  
Ergotamine (INN)
  D00679  
Ergotamine tartrate (JP18/USP)  <US>
 DG00446  
Ergometrine
  D07905  
Ergometrine (INN)
  D01163  
Ergonovine maleate (USP); Ergometrine maleate (JP18)
 DG00452  
Bromocriptine
  D03165  
Bromocriptine (USAN/INN)
  D00780  
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18)  <JP/US>
 D00987  
Cabergoline (JP18/USP/INN)  <JP/US>
 D02577  
Flibanserin (USAN/INN)  <US>
 D04463  
Norgestrel and ethinylestradiol tablets (JP18)  <JP/US>
 D09741  
Drospirenone and ethinylestradiol  <JP/US>
 D03917  
Drospirenone (JAN/USP/INN)  <US>
 DG00461  
Ethinylestradiol
  D00554  
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN)  <JP>
  D07928  
Ethinylestradiol propanesulfonate
 DG00462  
Estradiol
  D00105  
Estradiol (JAN/USP/INN)  <JP/US>
  D01413  
Estradiol valerate (JAN/USP/INN)  <JP/US>
  D01617  
Estradiol dipropionate (JAN)
  D01953  
Estradiol benzoate (JP18/USP)
  D04061  
Estradiol acetate (USAN)  <US>
  D04063  
Estradiol cypionate (USP)  <US>
  D04064  
Estradiol enanthate (USAN)
  D04065  
Estradiol undecylate (USAN/INN)
  D07918  
Estradiol hemihydrate  <US>
  D07919  
Estradiol 17 beta-hemisuccinate
 DG00464  
Estrone
  D00067  
Estrone (JAN/USP/INN)
  D00312  
Estrone sodium sulfate
  D00948  
Estropipate (USP)
 DG00465  
Conjugated estrogen
  D04070  
Estrogens, conjugated (JAN/USP)  <JP/US>
  D05987  
Synthetic conjugated estrogens, B (USAN)
 D00066  
Progesterone (JP18/USP/INN)  <JP/US>
 D01217  
Dydrogesterone (JP18/USP/INN)  <JP>
 D03799  
Dienogest (JAN/USAN/INN)  <JP>
 D09188  
Estradiol and norethindrone  <JP/US>
 D09187  
Estradiol and levonorgestrel  <JP/US>
 D00585  
Mifepristone (JAN/USAN/INN)  <US>
 DG00478  
Oxybutynin
  D00465  
Oxybutynin (USAN/INN)  <US>
  D00722  
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18)  <JP/US>
 DG00479  
Propiverine
  D08441  
Propiverine (INN)
  D01007  
Propiverine hydrochloride (JP18)  <JP>
 DG00480  
Tolterodine
  D00646  
Tolterodine (USAN/INN)
  D01148  
Tolterodine tartrate (JAN/USP)  <JP/US>
 DG00481  
Solifenacin
  D08522  
Solifenacin (INN)
  D01269  
Solifenacin succinate (JAN/USAN/INN)  <JP/US>
 DG00482  
Darifenacin
  D03654  
Darifenacin (USAN/INN)
  D01699  
Darifenacin hydrobromide (JAN/USAN)  <US>
 DG00483  
Fesoterodine
  D07226  
Fesoterodine (INN)
  D08923  
Fesoterodine fumarate (JAN/USAN)  <JP/US>
 D09535  
Mirabegron (JAN/USAN/INN)  <JP/US>
 D06273  
Imidafenacin (JAN/INN)  <JP>
 D10433  
Vibegron (JAN/USAN/INN)  <JP/US>
 DG00484  
Sildenafil
  D08514  
Sildenafil (INN)
  D02229  
Sildenafil citrate (JAN/USP)  <JP/US>
 D02008  
Tadalafil (JAN/USP/INN)  <JP/US>
 DG00487  
Vardenafil
  D08668  
Vardenafil (USAN/INN)
  D02731  
Vardenafil dihydrochoride (USAN)
  D03260  
Vardenafil hydrochloride hydrate (JAN)  <JP/US>
  D09989  
Vardenafil hydrochloride (USP)
 D03217  
Avanafil (USAN/INN)  <US>
 DG00489  
Alfuzosin
  D07124  
Alfuzosin (INN)
  D01692  
Alfuzosin hydrochloride (JAN/USAN)  <US>
 D01965  
Silodosin (JP18/INN)  <JP/US>
 D11389  
Dutasteride and tamsulosin  <US>
 D03820  
Dutasteride (JAN/USP/INN)  <JP/US>
 D12486  
Finasteride and tadalafil  <US>
 D03671  
Deflazacort (USAN/INN)  <US>
 D11000  
Vamorolone (USAN/INN)  <US>
 DG02839  
Osilodrostat
  D11061  
Osilodrostat (USAN/INN)
  D11062  
Osilodrostat phosphate (JAN/USAN)  <JP/US>
 DG00513  
Cinacalcet
  D03504  
Cinacalcet (USAN)
  D03505  
Cinacalcet hydrochloride (JAN/USAN)  <JP/US>
 D01322  
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN)
 DG00605  
Clarithromycin
  D00276  
Clarithromycin (JP18/USP/INN)  <JP/US>
  D07710  
Clarithromycin lactobionate
 DG00616  
Ofloxacin
  D00453  
Ofloxacin (JP18/USP/INN)  <JP/US>
  D08291  
Ofloxacin hydrochloride
 DG03066  
Lefamulin
  D11631  
Lefamulin (USAN/INN)
  D11632  
Lefamulin acetate (USAN)  <US>
 D00350  
Itraconazole (JP18/USP)  <JP/US>
 D00424  
Rifabutin (JAN/USP/INN)  <JP/US>
 DG00644  
Bedaquiline
  D09872  
Bedaquiline (USAN/INN)
  D09873  
Bedaquiline fumarate (JAN/USAN)  <JP/US>
 D09785  
Delamanid (JAN/USAN)  <JP>
 DG00653  
Saquinavir
  D00429  
Saquinavir (JAN/USP/INN)
  D01160  
Saquinavir mesylate (USP); Saquinavir mesilate (JAN)  <US>
 DG00654  
Indinavir
  C07051  
Indinavir
  D03833  
Indinavir (USAN)
  D00897  
Indinavir sulfate (USP)
  D02861  
Indinavir sulfate ethanolate (JAN)
 DG00655  
Nelfinavir
  D08259  
Nelfinavir (INN)
  D00899  
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN)  <US>
 D00894  
Amprenavir (JAN/USAN/INN)
 DG00656  
Fosamprenavir
  D02497  
Fosamprenavir (INN)
  D02867  
Fosamprenavir calcium hydrate (JAN)
  D03835  
Fosamprenavir calcium (USAN)  <US>
  D03837  
Fosamprenavir sodium (USAN)
 DG00659  
Darunavir
  D03656  
Darunavir (USAN/INN)  <US>
  D06478  
Darunavir ethanolate (JAN)  <JP/US>
  D12637  
Darunavir hydrate  <US>
  D12752  
Darunavir propylene glycolate  <US>
 D12269  
Nirmatrelvir and ritonavir  <JP/US>
 D00435  
Nevirapine (JAN/USP/INN)  <JP/US>
 D00896  
Efavirenz (JAN/USP/INN)  <US>
 D04112  
Etravirine (JAN/USAN/INN)  <US>
 DG00667  
Dolutegravir
  D10066  
Dolutegravir (USAN)
  D10113  
Dolutegravir sodium (JAN/USAN)  <JP/US>
 D09012  
Telaprevir (JAN/USAN/INN)
 DG01669  
Daclatasvir
  D10065  
Daclatasvir (USAN)
  D10105  
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN)
 D10745  
Ombitasvir, paritaprevir and ritonavir
 D10827  
Sofosbuvir and velpatasvir  <JP/US>
 D10600  
Dolutegravir, abacavir and lamivudine  <JP/US>
 D10753  
Atazanavir and cobicistat  <US>
 D06670  
Maraviroc (JAN/INN)  <JP/US>
 D04859  
Maribavir (JAN/USAN/INN)  <US>
 DG00675  
Cyclophosphamide
  D07760  
Cyclophosphamide (INN)
  D00287  
Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18)  <JP/US>
 D00343  
Ifosfamide (JAN/USP/INN)  <JP/US>
 DG00689  
Vinblastine
  D08675  
Vinblastine (INN)
  D01068  
Vinblastine sulfate (JP18/USP)  <JP/US>
 DG00692  
Vinorelbine
  D08680  
Vinorelbine (INN)
  D01935  
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN)  <JP/US>
 DG01430  
Paclitaxel
  D00491  
Paclitaxel (JAN/USP/INN)  <JP/US>
  D05333  
Paclitaxel poliglumex (USAN/INN)
 DG00694  
Docetaxel
  D07866  
Docetaxel (JAN/INN)  <JP/US>
  D02165  
Docetaxel (USP); Docetaxel hydrate (JP18)  <JP/US>
 DG00726  
Irinotecan
  D08086  
Irinotecan (INN)
  D01061  
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18)  <JP/US>
  D10642  
Irinotecan sucrosofate (USAN)
 D06199  
Trabectedin (JAN/USAN/INN)  <JP/US>
 D04645  
Ixabepilone (JAN/USAN/INN)  <US>
 DG00710  
Imatinib
  D08066  
Imatinib (INN)
  D01441  
Imatinib mesylate (USAN); Imatinib mesilate (JAN)  <JP/US>
 DG00714  
Dasatinib
  D03658  
Dasatinib (JAN/INN)  <JP>
  D06414  
Dasatinib (USAN); Dasatinib hydrate (JAN)  <JP/US>
  D12609  
Dasatinib laurylsulfate (USAN)
 DG00716  
Nilotinib
  D08953  
Nilotinib (USAN/INN)
  D06413  
Nilotinib hydrochloride hydrate (JAN)  <JP/US>
  D12444  
Nilotinib hydrochloride dihydrate (JAN)
  D12854  
Nilotinib laurylsulfate (USAN)
 DG00718  
Bosutinib
  D03252  
Bosutinib (USAN)
  D09728  
Bosutinib hydrate (JAN)  <JP/US>
 DG03004  
Asciminib
  D11403  
Asciminib (USAN/INN)
  D11404  
Asciminib hydrochloride (JAN/USAN)  <JP/US>
 DG00711  
Erlotinib
  D07907  
Erlotinib (INN)
  D04023  
Erlotinib hydrochloride (JAN/USAN)  <JP/US>
 DG00721  
Dabrafenib
  D10064  
Dabrafenib (USAN)
  D10104  
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN)  <JP/US>
 D11053  
Encorafenib (JAN/USAN/INN)  <JP/US>
 D09731  
Crizotinib (JAN/USAN/INN)  <JP/US>
 DG01625  
Alectinib
  D10542  
Alectinib (USAN/INN)
  D10450  
Alectinib hydrochloride (JAN)  <JP/US>
 D10866  
Brigatinib (JAN/USAN)  <JP/US>
 DG01414  
Selumetinib
  D09666  
Selumetinib (USAN/INN)
  D10024  
Selumetinib sulfate (JAN/USAN)  <JP/US>
 DG02084  
Ribociclib
  D10883  
Ribociclib (USAN/INN)
  D10979  
Ribociclib succinate (USAN)  <US>
 D06068  
Temsirolimus (JAN/USAN/INN)  <JP/US>
 D02714  
Everolimus (JAN/USAN/INN)  <JP/US>
 D00753  
Sirolimus (JAN/USAN/INN)  <JP/US>
 DG00715  
Lapatinib
  D08108  
Lapatinib (INN)
  D04024  
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN)  <JP/US>
 DG02303  
Neratinib
  D08950  
Neratinib (USAN/INN)
  D10898  
Neratinib maleate  <US>
 DG02968  
Fedratinib
  D10630  
Fedratinib (USAN/INN)
  D11296  
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN)  <US>
 D11768  
Pacritinib (USAN/INN)  <US>
 DG01366  
Momelotinib
  D10315  
Momelotinib (USAN/INN)
  D10358  
Momelotinib dihydrochloride (USAN)
  D10889  
Momelotinib hydrochloride hydrate (JAN)  <US>
 D03218  
Axitinib (JAN/USAN)  <JP/US>
 DG01375  
Tivozanib
  D09683  
Tivozanib (USAN/INN)
  D10190  
Tivozanib hydrochloride (USAN)  <US>
 D10927  
Erdafitinib (JAN/USAN/INN)  <US>
 D11417  
Pemigatinib (JAN/USAN/INN)  <JP/US>
 DG00712  
Sunitinib
  D08552  
Sunitinib (INN)
  D06402  
Sunitinib malate (JAN/USAN)  <JP/US>
 D06407  
Vandetanib (JAN/USAN/INN)  <JP/US>
 DG00720  
Regorafenib
  D10138  
Regorafenib (USAN/INN)
  D10137  
Regorafenib hydrate (JAN)  <JP/US>
 D05029  
Midostaurin (JAN/USAN/INN)  <US>
 DG01948  
Gilteritinib
  D10709  
Gilteritinib (USAN/INN)
  D10800  
Gilteritinib fumarate (JAN/USAN)  <JP/US>
 D10926  
Entrectinib (JAN/USAN/INN)  <JP/US>
 DG02960  
Pexidartinib
  D11270  
Pexidartinib (USAN/INN)
  D11271  
Pexidartinib hydrochloride (JAN/USAN)  <US>
 DG02081  
Capmatinib
  D10696  
Capmatinib (USAN/INN)
  D10891  
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN)  <JP/US>
 DG03087  
Tepotinib
  D11717  
Tepotinib (USAN/INN)
  D11073  
Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN)  <JP/US>
 D11713  
Selpercatinib (JAN/USAN/INN)  <JP/US>
 D11371  
Capivasertib (JAN/USAN)  <JP/US>
 D03259  
Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN)  <JP/US>
 D10954  
Mirvetuximab soravtansine (USAN/INN)  <US>
 DG01403  
Panobinostat
  D10319  
Panobinostat (USAN/INN)
  D10019  
Panobinostat lactate (JAN)
 D08870  
Belinostat (USAN/INN)  <US>
 D08914  
Eribulin mesylate (USAN); Eribulin mesilate (JAN)  <JP/US>
 D11222  
Selinexor (USAN/INN)  <US>
 D11954  
Belzutifan (JAN/USAN/INN)  <US>
 D12301  
Adagrasib (USAN/INN)  <US>
 DG00734  
Tamoxifen
  D08559  
Tamoxifen (INN)
  D00966  
Tamoxifen citrate (JP18/USP)  <JP/US>
 DG00735  
Toremifene
  D08620  
Toremifene (INN)
  D00967  
Toremifene citrate (JAN/USAN)  <JP/US>
 D01161  
Fulvestrant (JAN/USP/INN)  <JP/US>
 DG03078  
Elacestrant
  D11671  
Elacestrant (USAN/INN)
  D11672  
Elacestrant hydrochloride (USAN)  <US>
 D10218  
Enzalutamide (JAN/USAN)  <JP/US>
 D11040  
Apalutamide (JAN/INN)  <JP/US>
 D00964  
Letrozole (JAN/USP/INN)  <JP/US>
 D00963  
Exemestane (JAN/USP/INN)  <JP/US>
 D09701  
Abiraterone acetate (JAN/USP)  <JP/US>
 DG02927  
Leniolisib
  D11158  
Leniolisib (USAN/INN)
  D11159  
Leniolisib phosphate (USAN)  <US>
 D00184  
Cyclosporine (USP); Ciclosporin (JP18)  <JP/US>
 D09033  
Voclosporin (JAN/USAN/INN)  <US>
 DG03018  
Siponimod
  D11460  
Siponimod (USAN/INN)
  D11072  
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN)  <JP/US>
 DG02444  
Etrasimod
  D10930  
Etrasimod (USAN)
  D10931  
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN)  <US>
 DG00742  
Tofacitinib
  D09970  
Tofacitinib (USAN)
  D09783  
Tofacitinib citrate (JAN/USAN)  <JP/US>
 DG02829  
Upadacitinib
  D10994  
Upadacitinib (USAN/INN)  <US>
  D10995  
Upadacitinib tartrate (USAN)
  D11048  
Upadacitinib hydrate (JAN)  <JP>
 D11093  
Avacopan (JAN/USAN/INN)  <JP/US>
 D00749  
Leflunomide (JAN/USP/INN)  <JP/US>
 D08976  
Pomalidomide (JAN/USAN/INN)  <JP/US>
 D00969  
Meloxicam (JAN/USP/INN)  <JP/US>
 D11576  
Naproxen and esomeprazole magnesium  <US>
 D00570  
Colchicine (JP18/USP)  <JP/US>
 D11406  
Risdiplam (JAN/USAN/INN)  <JP/US>
 D09365  
Palovarotene (JAN/USAN/INN)  <US>
 D00542  
Halothane (JP18/USP/INN)
 DG00791  
Fentanyl
  D00320  
Fentanyl (JAN/USP/INN)  <JP/US>
  D01399  
Fentanyl citrate (JP18/USP)  <JP/US>
  D10811  
Fentanyl hydrochloride (JAN)
 D03852  
Droperidol and fentanyl citrate
 DG01829  
Esketamine
  D07283  
Esketamine (USAN/INN)
  D10627  
Esketamine hydrochloride (JAN/USAN)  <US>
 DG00801  
Bupivacaine
  D07552  
Bupivacaine (USAN/INN)  <US>
  D01450  
Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18)  <JP/US>
 DG00806  
Ropivacaine
  D08490  
Ropivacaine (INN)
  D04048  
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN)  <JP/US>
 DG00807  
Levobupivacaine
  D08116  
Levobupivacaine (INN)
  D01287  
Levobupivacaine hydrochloride (JAN/USAN)  <JP>
 D02740  
Lidocaine and prilocaine  <JP/US>
 DG00813  
Oxycodone
  D05312  
Oxycodone (USAN/INN)  <US>
  D00847  
Oxycodone hydrochloride (USP)  <US>
  D02175  
Compound oxycodone (JP18)
  D03783  
Oxycodone terephthalate (USP)
  D05462  
Oxycodone hydrochloride hydrate (JP18)  <JP>
 DG00814  
Dihydrocodeine
  D07831  
Dihydrocodeine (INN)
  D01481  
Dihydrocodeine phosphate (JP18)  <JP>
  D03825  
Dihydrocodeine bitartrate (USP)
  D07832  
Dihydrocodeine thiocyanate
 D08695  
dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea  <JP>
 DG00820  
Buprenorphine
  D07132  
Buprenorphine (JAN/INN)  <JP/US>
  D00836  
Buprenorphine hydrochloride (JP18/USP)  <JP/US>
 D09999  
Tramadol hydrochloride and acetaminophen  <JP/US>
 D11573  
Oxycodone and ibuprofen
 DG00824  
Tramadol
  D08623  
Tramadol (INN)
  D01355  
Tramadol hydrochloride (JP18/USP)  <JP/US>
 D00544  
Methoxyflurane (USP/INN)
 DG00833  
Dihydroergotamine
  D07837  
Dihydroergotamine (INN)
  D02211  
Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18)  <US>
  D07838  
Dihydroergotamine tartrate
 D07585  
Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine  <JP>
 DG00837  
Naratriptan
  D08255  
Naratriptan (INN)
  D00674  
Naratriptan hydrochloride (JAN/USP)  <JP/US>
 DG00839  
Almotriptan
  D02824  
Almotriptan (USAN)
  D02825  
Almotriptan malate (USP)  <US>
 DG00840  
Eletriptan
  D07887  
Eletriptan (INN)
  D01973  
Eletriptan hydrobromide (JAN/USAN)  <JP/US>
  D11617  
Eletriptan hydrobromide monohydrate
 D10673  
Ubrogepant (USAN/INN)  <US>
 DG01845  
Rimegepant
  D10662  
Rimegepant (USAN/INN)
  D10663  
Rimegepant sulfate (USAN)  <US>
 D11313  
Atogepant (USAN)  <US>
 D00539  
Ethosuximide (JP18/USP/INN)  <JP/US>
 D00252  
Carbamazepine (JP18/USP/INN)  <JP/US>
 D00537  
Topiramate (JAN/USP/INN)  <JP/US>
 D05928  
Stiripentol (JAN/USAN/INN)  <JP>
 D07299  
Lacosamide (JAN/USAN/INN)  <JP/US>
 D10915  
Cannabidiol (USAN/INN)  <US>
 D11150  
Cenobamate (USAN/INN)  <US>
 D04300  
Ganaxolone (USAN/INN)  <US>
 DG00864  
Selegiline
  D03731  
Selegiline (USAN/INN)  <US>
  D00785  
Selegiline hydrochloride (JAN/USP)  <JP/US>
 DG01260  
Safinamide
  D10158  
Safinamide (USAN/INN)
  D10191  
Safinamide mesylate (USAN); Safinamide mesilate (JAN)  <JP/US>
 D04641  
Istradefylline (JAN/USAN/INN)  <JP/US>
 DG00885  
Haloperidol
  D00136  
Haloperidol (JP18/USP/INN)  <JP/US>
  D01898  
Haloperidol decanoate (JAN/USP)  <JP/US>
  D08035  
Haloperidol lactate  <US>
 DG00890  
Bromperidol
  D01101  
Bromperidol (JAN/USAN/INN)  <JP>
  D02626  
Bromperidol decanoate (USAN)
 D04820  
Lurasidone hydrochloride (JAN/USAN)  <JP/US>
 D00560  
Pimozide (JP18/USP/INN)  <US>
 DG00897  
Loxapine
  D02340  
Loxapine (USAN/INN)  <US>
  D00794  
Loxapine succinate (USP)  <US>
  D08148  
Loxapine hydrochloride
 D00283  
Clozapine (JAN/USP/INN)  <JP/US>
 DG00899  
Quetiapine
  D08456  
Quetiapine (INN)
  D00458  
Quetiapine fumarate (JP18/USP)  <JP/US>
 D00426  
Risperidone (JP18/USP/INN)  <JP/US>
 DG00906  
Aripiprazole
  D01164  
Aripiprazole (JAN/USP/INN)  <JP/US>
  D10355  
Aripiprazole cavoxil (USAN)
  D10364  
Aripiprazole lauroxil (USAN)  <US>
  D10516  
Aripiprazole hydrate (JAN)  <JP/US>
 D02666  
Iloperidone (USAN/INN)  <US>
 DG01305  
Cariprazine
  D09997  
Cariprazine (USAN/INN)
  D09876  
Cariprazine hydrochloride (JAN/USAN)  <US>
 D10309  
Brexpiprazole (JAN/USAN/INN)  <JP/US>
 D08969  
Pimavanserin tartrate (USAN)  <US>
 D00293  
Diazepam (JP18/USP/INN)  <JP/US>
 D01253  
Clobazam (JAN/USAN/INN)  <JP/US>
 D08283  
Nordazepam (INN)
 D01293  
Ethyl loflazepate (JP18/INN)  <JP>
 D01514  
Etizolam (JP18/INN)  <JP>
 D01316  
Mexazolam (JAN/INN)  <JP>
 D00387  
Triazolam (JP18/USP/INN)  <JP/US>
 DG00920  
Midazolam
  D00550  
Midazolam (JAN/USP/INN)  <JP/US>
  D00696  
Midazolam hydrochloride (USAN)  <US>
  D05028  
Midazolam maleate (USAN)
 D01744  
Brotizolam (JP18/USAN/INN)  <JP>
 D00457  
Quazepam (JAN/USP/INN)  <JP/US>
 D01372  
Zopiclone (JP18/INN)  <JP>
 DG00922  
Zolpidem
  D08690  
Zolpidem (INN)
  D00706  
Zolpidem tartrate (JP18/USP)  <JP/US>
 D00530  
Zaleplon (JAN/USP/INN)  <US>
 D02624  
Eszopiclone (JAN/USP/INN)  <JP/US>
 D09388  
Tasimelteon (USAN/INN)  <US>
 D11022  
Lemborexant (JAN/USAN/INN)  <JP/US>
 D11886  
Daridorexant (USAN/INN)
 DG00928  
Imipramine
  D08070  
Imipramine (INN)
  D00815  
Imipramine hydrochloride (JP18/USP)  <JP/US>
  D08071  
Imipramine pamoate (USP)  <US>
 DG00929  
Clomipramine
  D07727  
Clomipramine (INN)
  D00811  
Clomipramine hydrochloride (JP18/USP)  <JP/US>
 DG00934  
Amitriptyline
  D07448  
Amitriptyline (INN)
  D00809  
Amitriptyline hydrochloride (JP18/USP)  <JP/US>
 DG00943  
Citalopram
  D07704  
Citalopram (USP/INN)
  D00822  
Citalopram hydrobromide (USP)  <US>
  D07705  
Citalopram hydrochloride
 DG00945  
Sertraline
  D02360  
Sertraline (INN)
  D00825  
Sertraline hydrochloride (JAN/USP)  <JP/US>
 DG00947  
Escitalopram
  D07913  
Escitalopram (INN)
  D02567  
Escitalopram oxalate (JAN/USP)  <JP/US>
 DG00951  
Mianserin
  D08216  
Mianserin (INN)
  D01358  
Mianserin hydrochloride (JAN/USAN)  <JP>
 DG00952  
Trazodone
  D08626  
Trazodone (INN)
  D00820  
Trazodone hydrochloride (JAN/USP)  <JP/US>
 DG02838  
Mirtazapine
  D00563  
Mirtazapine (JAN/USP/INN)  <JP/US>
  D11056  
Mirtazapine hydrate (JAN)
 DG00959  
Venlafaxine
  D08670  
Venlafaxine (INN)
  D00821  
Venlafaxine hydrochloride (JAN/USP)  <JP/US>
  D12403  
Venlafaxine besylate monohydrate  <US>
 D04314  
Gepirone hydrochloride (USAN)  <US>
 DG00963  
Desvenlafaxine
  D07793  
Desvenlafaxine (INN)  <US>
  D02570  
Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN)  <US>
  D11619  
Desvenlafaxine succinate anhydrous  <US>
 DG00964  
Vilazodone
  D09698  
Vilazodone (USAN/INN)
  D09699  
Vilazodone hydrochloride (USAN)  <US>
 DG00965  
Vortioxetine
  D10184  
Vortioxetine (USAN)
  D10185  
Vortioxetine hydrobromide (JAN/USAN)  <JP/US>
  D12544  
Vortioxetine hemihydrobromide (USAN)
 D01832  
Modafinil (JAN/USP/INN)  <JP/US>
 D03215  
Armodafinil (USAN/INN)  <US>
 DG00983  
Donepezil
  D07869  
Donepezil (JAN/INN)  <JP>
  D00670  
Donepezil hydrochloride (JP18/USP)  <JP/US>
 DG00985  
Galantamine
  D04292  
Galantamine (USAN/INN)
  D02173  
Galantamine hydrobromide (JAN/USP)  <JP/US>
 DG00993  
Cevimeline
  D07667  
Cevimeline (INN)
  D00661  
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN)  <JP/US>
 DG00999  
Methadone
  D08195  
Methadone (BAN)
  D02102  
Methadone hydrochloride (JAN/USP)  <JP/US>
 DG01000  
Levacetylmethadol
  D04716  
Levomethadyl acetate (USAN); Levacetylmethadol (INN)
  D00840  
Levomethadyl acetate hydrochloride (USAN)
 D08575  
Tetrabenazine (JAN/INN)  <JP/US>
 DG03021  
Pitolisant
  D10749  
Pitolisant (USAN/INN)
  D11490  
Pitolisant hydrochloride (USAN)  <US>
 DG02115  
Valbenazine
  D10675  
Valbenazine (USAN/INN)
  D10999  
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN)  <JP/US>
 DG01015  
Hydroxychloroquine
  D08050  
Hydroxychloroquine (INN)
  D02114  
Hydroxychloroquine sulfate (JAN/USP)  <JP/US>
 DG01019  
Quinine
  D08460  
Quinine (BAN)
  D01663  
Quinine ethylcarbonate (JP18)
  D02261  
Quinine hydrochloride hydrate (JP18)
  D02262  
Quinine sulfate (USP); Quinine sulfate hydrate (JP18)  <US>
  D05681  
Quinine ascorbate (USAN)
  D08461  
Quinine dihydrochloride
 D11252  
Fexinidazole (USAN/INN)  <US>
 D00471  
Praziquantel (JAN/USP/INN)  <JP/US>
 DG01040  
Flunisolide
  C07005  
Flunisolide
  D00324  
Flunisolide (JAN/USP)  <US>
  D04214  
Flunisolide acetate (USAN)
 D01703  
Ciclesonide (JAN/USAN/INN)  <JP/US>
 D08699  
Salmeterol xinafoate and fluticasone propionate  <JP/US>
 DG01051  
Salmeterol
  D05792  
Salmeterol (USAN/INN)
  D00687  
Salmeterol xinafoate (JAN/USP)  <JP/US>
 DG01055  
Procaterol
  D08424  
Procaterol (INN)
  D02404  
Procaterol hydrochloride (USAN)
  D05366  
Procaterol hydrochloride hydrate (JP18)  <JP>
 DG01057  
Indacaterol
  D09318  
Indacaterol (USAN/INN)
  D09319  
Indacaterol maleate (JAN/USAN)  <JP>
  D11009  
Indacaterol acetate (JAN)
 D09595  
Budesonide and formoterol fumarate dihydrate  <JP/US>
 D10501  
Fluticasone furoate and vilanterol trifenatate  <JP/US>
 D10506  
Fluticasone propionate and formoterol fumarate hydrate  <JP>
 D10533  
Umeclidinium bromide and vilanterol  <JP/US>
 D10505  
Glycopyrronium bromide and indacaterol maleate  <JP>
 DG01065  
Pranlukast
  D08408  
Pranlukast (INN)
  D02732  
Pranlukast hydrate (JP18)  <JP>
 DG01066  
Montelukast
  D08229  
Montelukast (INN)
  D00529  
Montelukast sodium (JP18/USP)  <JP/US>
 DG01074  
Ethylmorphine
  D07929  
Ethylmorphine (BAN)
  D02205  
Ethylmorphine hydrochloride hydrate (JP18)
 DG01075  
Hydrocodone
  D08045  
Hydrocodone (INN)
  D03725  
Hydrocodone bitartrate (USP)  <US>
  D04461  
Hydrocodone polistirex (USAN)
  D08046  
Hydrocodone hydrochloride
 DG01076  
Codeine
  C06174  
Codeine
  D00195  
Codeine (USP)
  D02101  
Codeine phosphate (USP); Codeine phosphate hydrate (JP18)  <JP>
  D03579  
Codeine polistirex (USAN)
  D03580  
Codeine sulfate (USP)  <US>
  D07740  
Codeine hydrochloride
 D12312  
Codeine phosphate and chlorpheniramine maleate  <US>
 D04340  
Dextromethorphan hydrobromide and potassium cresolsulfonate  <JP>
 D04313  
Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate  <JP>
 D04447  
Betamethasone and d-chlorpheniramine maleate  <JP>
 D12313  
Chlorpheniramine polistirex and codeine polistirex
 DG01108  
Levocetirizine
  D07402  
Levocetirizine (USAN/INN)
  D08118  
Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN)  <JP/US>
 D00364  
Loratadine (JAN/USP/INN)  <JP>
 D01478  
Ebastine (JP18/USAN/INN)  <JP>
 DG01118  
Rupatadine
  D07407  
Rupatadine (INN)
  D08497  
Rupatadine fumarate (JAN)  <JP>
 DG01119  
Doxapram
  D07873  
Doxapram (INN)
  D01872  
Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18)  <JP/US>
 DG01135  
Dorzolamide
  D07871  
Dorzolamide (INN)
  D00653  
Dorzolamide hydrochloride (JP18/USP)  <JP/US>
 D10512  
Brinzolamide and timolol maleate  <JP>
 D08493  
Dorzolamide hydrochloride and timolol maleate (JP18)  <JP/US>
 D06405  
Nalfurafine hydrochloride (JAN/USAN)  <JP>
 DG01307  
Rilmazafone
  D08481  
Rilmazafone (INN)
  D01564  
Rilmazafone hydrochloride hydrate (JP18)  <JP>
 DG01333  
Sarpogrelate
  D08508  
Sarpogrelate (INN)
  D01624  
Sarpogrelate hydrochloride (JP18)  <JP>
 DG03016  
Nirogacestat
  D10960  
Nirogacestat (USAN/INN)
  D11453  
Nirogacestat hydrobromide (USAN)  <US>
 D01098  
Maxacalcitol (JAN/USAN/INN)  <JP>
 D01145  
Azelnidipine (JP18/INN)  <JP>
 D01176  
Blonanserin (JAN/INN)  <JP>
 D01418  
Tamibarotene (JAN/USAN/INN)  <JP>
 D01468  
Nemonapride (JAN/INN)  <JP>
 D04052  
Epinephrine and lidocaine hydrochloride  <JP/US>
 D04338  
Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride  <JP>
 D04446  
Betamethasone acetate and betamethasone sodium phosphate  <JP/US>
 D04813  
Lidocaine hydrochloride and epinephrine bitartrate  <JP/US>
 D08697  
Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate
 D08856  
Anamorelin hydrochloride (JAN/USAN)  <JP>
 D09594  
Olmesartan medoxomil and azelnidipine  <JP>
 D10524  
Azilsartan and amlodipine besilate  <JP>
 D10525  
Valsartan and cilnidipine  <JP>
 D10897  
Teneligliptin and canagliflozin  <JP>
 D11454  
Repotrectinib (JAN/USAN)  <US>
 D11553  
Lidocaine and tetracaine  <US>
 D11616  
Aspirin and omeprazole
 D11628  
Benzhydrocodone and acetaminophen
 D11656  
Azelastine hydrochloride and fluticasone propionate  <US>
 D11706  
Omeprazole and sodium bicarbonate  <US>
 D11793  
Zuranolone (JAN/USAN/INN)  <US>
 D11851  
Butalbital, acetaminophen, caffeine and codeine phosphate  <US>
 D11860  
Butalbital, aspirin, caffeine and codeine  <US>
 D12130  
Drospirenone, ethinyl estradiol and levomefolate calcium  <US>
 D12483  
Olutasidenib (USAN/INN)  <US>
 D12497  
Drospirenone and estradiol  <US>
 DG01850  
Benzhydrocodone
  D10612  
Benzhydrocodone (USAN/INN)
  D10692  
Benzhydrocodone hydrochloride (USAN)
 D01562  
Aranidipine (JAN/INN)
 D01855  
Mozavaptane hydrochloride (JAN)
 D12756  
Vonoprazan and amoxicillin  <US>
Hydrocortisone
 D00088  
Hydrocortisone (JP18/USP/INN)  <JP/US>
 D00165  
Hydrocortisone acetate (JP18/USP)  <US>
 D00976  
Hydrocortisone cypionate
 D00977  
Hydrocortisone sodium phosphate (JP18/USP)  <JP>
 D00978  
Hydrocortisone sodium succinate (JP18/USP)  <JP/US>
 D01442  
Hydrocortisone succinate (JP18)
 D01619  
Hydrocortisone butyrate (JP18/USP)  <JP/US>
 D01886  
Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN)  <JP/US>
 D02288  
Hydrocortisone valerate (USP)  <US>
 D04467  
Hydrocortisone hemisuccinate (USP)
 D06876  
Hydrocortisone aceponate (INN)
 D09796  
Hydrocortisone caproate (JAN)
D00472  
Prednisolone (JP18/USP/INN)  <JP/US>
D11858  
Omeprazole magnesium, amoxicillin and rifabutin  <US>
Cisapride
 D00274  
Cisapride (USP/INN)
 D02092  
Cisapride (JAN)
Dolasetron
 D07867  
Dolasetron (INN)
 D00725  
Dolasetron mesylate (USP)  <US>
Naloxegol
 D10479  
Naloxegol (USAN/INN)
 D10375  
Naloxegol oxalate (USAN)  <US>
D10865  
Bexagliflozin (USAN)  <US>
D09017  
Ticagrelor (JAN/USAN/INN)  <JP/US>
D00297  
Digitoxin (JAN/USP/INN)
Dronedarone
 D02537  
Dronedarone (INN)
 D03914  
Dronedarone hydrochloride (USP)  <US>
Ranolazine
 D05700  
Ranolazine (USAN/INN)  <US>
 D05701  
Ranolazine hydrochloride (USAN)
D09572  
Riociguat (JAN/USAN/INN)  <JP/US>
Conivaptan
 D07748  
Conivaptan (INN)
 D01236  
Conivaptan hydrochloride (JAN/USAN)
Lercanidipine
 D08111  
Lercanidipine (INN)
 D01849  
Lercanidipine hydrochloride (JAN/USAN)
D10711  
Pemafibrate (JAN)  <JP>
Erythromycin
 D00140  
Erythromycin (JP18/USP/INN)  <JP/US>
 D00851  
Erythromycin estolate (USP); Erythromycin estorate (JAN)
 D01361  
Erythromycin ethylsuccinate (JP18/USP)  <JP/US>
 D02009  
Erythromycin lactobionate (JP18/USP)  <JP/US>
 D02184  
Erythromycin stearate (JP18/USP)  <JP/US>
 D02523  
Erythromycin acistrate (USAN)
 D02524  
Erythromycin gluceptate (USP)
 D02525  
Erythromycin propionate (USAN)
 D03098  
Berythromycin (USAN/INN)
 D04054  
Erythromycin salnacedin (USAN)
 D07909  
Erythromycin thiocyanate
 D07910  
Erythromycin stinoprate (INN)
D10461  
Dienogest and estradiol valerate  <US>
D12586  
Mifepristone and misoprostol  <JP>
D12137  
Elagolix, estradiol and norethisterone  <US>
D01710  
Roxithromycin (JP18/USAN/INN)  <JP>
D01078  
Telithromycin (JAN/USAN/INN)
D00427  
Ritonavir (JAN/USP/INN)  <JP/US>
Ensitrelvir
 D12619  
Ensitrelvir (USAN/INN)
 D12353  
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN)  <JP>
Delavirdine
 D07782  
Delavirdine (INN)
 D00895  
Delavirdine mesylate (USAN); Delavirdine mesilate (JAN)
Rilpivirine
 D09720  
Rilpivirine (JAN/USAN/INN)  <JP>
 D09958  
Rilpivirine hydrochloride (JAN/USAN)  <JP/US>
D10624  
Doravirine (JAN/USAN/INN)  <JP/US>
Simeprevir
 D10081  
Simeprevir (JAN/USAN)
 D10469  
Simeprevir sodium (JAN)
D10093  
Asunaprevir (JAN/USAN)
D10625  
Elbasvir (JAN/USAN/INN)
Grazoprevir
 D11565  
Grazoprevir (USAN/INN)
 D10639  
Grazoprevir (USAN); Grazoprevir hydrate (JAN)
D10582  
Dasabuvir, ombitasvir, paritaprevir and ritonavir
D10882  
Daclatasvir, asunaprevir and beclabuvir
D11521  
Lamivudine, nevirapine and zidovudine
D10571  
Rilpivirine hydrochloride, tenofovir disoproxil fumarate and emtricitabine  <US>
D10756  
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil  <US>
D02498  
Lopinavir and ritonavir  <JP/US>
D10835  
Emtricitabine and tenofovir alafenamide  <JP/US>
D10836  
Emtricitabine, rilpivirine and tenofovir alafenamide  <JP/US>
D11282  
Dolutegravir sodium and rilpivirine hydrochloride  <JP/US>
D11396  
Doravirine, lamivudine and tenofovir disoproxil  <US>
D10564  
Amenamevir (JAN/INN)  <JP>
Temsavir
 D10734  
Temsavir (USAN/INN)
 D10707  
Fostemsavir (USAN)
 D10708  
Fostemsavir tromethamine (USAN)  <US>
Lenacapavir
 D12161  
Lenacapavir (USAN/INN)
 D12162  
Lenacapavir sodium (JAN/USAN)  <JP/US>
Vincristine
 D08679  
Vincristine (INN)
 D02197  
Vincristine sulfate (JP18/USP)  <JP/US>
Vindesine
 D06304  
Vindesine (USAN/INN)
 D01769  
Vindesine sulfate (JAN/USAN)  <JP>
Cabazitaxel
 D09755  
Cabazitaxel (USAN/INN)
 D10452  
Cabazitaxel acetonate (JAN)  <JP/US>
Ponatinib
 D09950  
Ponatinib (USAN/INN)
 D09951  
Ponatinib hydrochloride (JAN/USAN)  <JP/US>
D10766  
Osimertinib mesylate (USAN); Osimertinib mesilate (JAN)  <JP/US>
Mobocertinib
 D12001  
Mobocertinib (USAN/INN)
 D11969  
Mobocertinib succinate (JAN)  <US>
D10551  
Ceritinib (JAN/USAN/INN)  <JP/US>
D11012  
Lorlatinib (JAN/USAN/INN)  <JP/US>
D10688  
Abemaciclib (JAN/USAN/INN)  <JP/US>
Tucatinib
 D11141  
Tucatinib (USAN/INN)  <US>
 D12442  
Tucatinib ethanolate (JAN)
D11977  
Fruquintinib (JAN/USAN)  <US>
D10223  
Ibrutinib (JAN/USAN)  <JP/US>
Acalabrutinib
 D10893  
Acalabrutinib (JAN/USAN/INN)  <JP/US>
 D11720  
Acalabrutinib maleate (USAN)
 D12704  
Acalabrutinib maleate hydrate (JAN)
D11422  
Zanubrutinib (JAN/USAN/INN)  <US>
D10560  
Idelalisib (JAN/USAN/INN)  <US>
Copanlisib
 D10867  
Copanlisib (USAN/INN)
 D10797  
Copanlisib hydrochloride (USAN)
 D10798  
Copanlisib hydrochloride hydrate (JAN)  <US>
Lenvatinib
 D09919  
Lenvatinib (USAN/INN)
 D09920  
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN)  <JP/US>
Quizartinib
 D09955  
Quizartinib (USAN/INN)
 D09956  
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN)  <JP/US>
Larotrectinib
 D11137  
Larotrectinib (USAN/INN)
 D11138  
Larotrectinib sulfate (JAN/USAN)  <JP/US>
D10761  
Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN)  <JP/US>
D06637  
Romidepsin (JAN/USAN/INN)  <JP/US>
Sonidegib
 D10119  
Sonidegib (USAN/INN)
 D10729  
Sonidegib phosphate (USAN)  <US>
D09730  
Olaparib (JAN/USAN/INN)  <JP/US>
D12055  
Sotorasib (JAN/USAN)  <JP/US>
Dantrolene
 D02347  
Dantrolene (USAN/INN)
 D02274  
Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18)  <JP/US>
D03844  
Phenytoin, phenobarbital and caffeine and sodium benzoate
D00538  
Zonisamide (JP18/USP/INN)  <JP/US>
Perampanel
 D08964  
Perampanel (USAN)
 D10780  
Perampanel hydrate (JAN)  <JP/US>
D00225  
Alprazolam (JP18/USP/INN)  <JP/US>
D02615  
Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital
D00311  
Estazolam (JP18/USP/INN)  <JP/US>
D10082  
Suvorexant (JAN/USAN)  <JP/US>
Mefloquine
 D04895  
Mefloquine (USAN/INN)
 D00831  
Mefloquine hydrochloride (JP18/USP)  <JP/US>
D02484  
Artemether and lumefantrine  <JP/US>
Dexchlorpheniramine
 D07803  
Dexchlorpheniramine (INN)
 D00668  
Dexchlorpheniramine maleate (USP); d-Chlorpheniramine maleate (JP18)  <JP/US>
D00234  
Astemizole (JAN/USP/INN)
D00521  
Terfenadine (JAN/USAN/INN)
D11700  
Elexacaftor, ivacaftor and tezacaftor  <US>
D09881  
Cobicistat (JAN/USAN/INN)  <US>
Isavuconazonium
 D10644  
Isavuconazonium (USAN)
 D10643  
Isavuconazonium sulfate (JAN/USAN)  <JP/US>
Colforsin
 D03584  
Colforsin (USAN/INN)
 D01697  
Colforsin daropate hydrochloride (JAN)  <JP>
D10892  
Esaxerenone (JAN/INN)  <JP>
D10964  
Omaveloxolone (USAN/INN)  <US>
D11776  
Sparsentan (USAN/INN)  <US>
D11966  
Cabotegravir and rilpivirine  <US>
D01425  
Lopinavir (JAN/USP/INN)
D05152  
Netupitant (USAN/INN)
D09987  
Vaniprevir (JAN/USAN/INN)
 » expand
Class
Metabolizing enzyme substrate
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