KEGG   DRUG: Vibecotamab
Entry
D11841                      Drug                                   
Name
Vibecotamab (USAN/INN)
Formula
C5629H8669N1503O1738S38
Exact mass
126345.5557
Mol weight
126423.63
Sequence
(A chain)
QVQLQQSGAE VKKPGASVKV SCKASGYTFT DYYMKWVKQS HGKSLEWMGD IIPSNGATFY
NQKFKGKATL TVDRSTSTAY MELSSLRSED TAVYYCARSH LLRASWFAYW GQGTLVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS DTKVDKKVEP KSCDKTHTCP PCPAPPVAGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVKH EDPEVKFNWY VDGVEVHNAK TKPREEEYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSREEM
TKNQVSLTCD VSGFYPSDIA VEWESDGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWE
QGDVFSCSVM HEALHNHYTQ KSLSLSPGK
(B chain)
DFVMTQSPDS LAVSLGERAT INCKSSQSLL NTGNQKNYLT WYQQKPGQPP KLLIYWASTR
ESGVPDRFTG SGSGTDFTLT ISSLQAEDVA VYYCQNDYSY PYTFGGGTKL EIKRTVAAPS
VFIFPPSDEQ LKSGTASVVC LLNNFYPREA KVQWKVDNAL QSGNSQESVT EQDSKDSTYS
LSSTLTLSKA DYEKHKVYAC EVTHQGLSSP VTKSFNRGEC
(C chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFS TYAMNWVRQA PGKGLEWVGR IRSKYNNYAT
YYADSVKGRF TISRDDSKNT LYLQMNSLRA EDTAVYYCVR HGNFGDSYVS WFAYWGQGTL
VTVSSGKPGS GKPGSGKPGS GKPGSQAVVT QEPSLTVSPG GTVTLTCGSS TGAVTTSNYA
NWVQQKPGKS PRGLIGGTNK RAPGVPARFS GSLLGGKAAL TISGAQPEDE ADYYCALWYS
NHWVFGGGTK LTVLEPKSSD KTHTCPPCPA PPVAGPSVFL FPPKPKDTLM ISRTPEVTCV
VVDVKHEDPE VKFNWYVDGV EVHNAKTKPR EEQYNSTYRV VSVLTVLHQD WLNGKEYKCK
VSNKALPAPI EKTISKAKGQ PREPQVYTLP PSREQMTKNQ VKLTCLVKGF YPSDIAVEWE
SNGQPENNYK TTPPVLDSDG SFFLYSKLTV DKSRWQQGNV FSCSVMHEAL HNHYTQKSLS
LSPGK
(Disulfide bridge: A22-A96, A147-A203, A223-B220, A229-C265, A232-C268, A263-A323, A369-A427, B23-B94, B140-B200, C22-C98, C167-C235, C299-C359, C405-C463)
  Type
Peptide
Efficacy
Antineoplastic, Immunomodulator
  Type
Bispecific antibody
Target
IL3RA (CD123) [HSA:3563] [KO:K04737]
CD3E [HSA:916] [KO:K06451]
  Pathway
hsa04640  Hematopoietic cell lineage
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    IL3RA (CD123)
     D11841  Vibecotamab (USAN/INN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3E
     D11841  Vibecotamab (USAN/INN)
Other DBs
CAS: 2138442-13-2
PubChem: 433774516
LinkDB

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