KEGG   DRUG: Tidutamab
Entry
D11845                      Drug                                   
Name
Tidutamab (USAN/INN)
Formula
C5633H8660N1504O1740S38
Exact mass
126430.4782
Mol weight
126508.60
Sequence
(A chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFS DYGMAWFRQA PGKGLEWVSF ISNLGYSIYY
ADSVKGRFTI SRDNAKNSLY LQMNSLRAED TAVYYCARAP YDYDSFDPMD YWGQGTLVTV
SSASTKGPSV FPLAPSSKST SGGTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ
SSGLYSLSSV VTVPSSSLGT QTYICNVNHK PSDTKVDKKV EPKSCDKTHT CPPCPAPPVA
GPSVFLFPPK PKDTLMISRT PEVTCVVVDV KHEDPEVKFN WYVDGVEVHN AKTKPREEEY
NSTYRVVSVL TVLHQDWLNG KEYKCKVSNK ALPAPIEKTI SKAKGQPREP QVYTLPPSRE
EMTKNQVSLT CDVSGFYPSD IAVEWESDGQ PENNYKTTPP VLDSDGSFFL YSKLTVDKSR
WEQGDVFSCS VMHEALHNHY TQKSLSLSPG K
(B chain)
DIVMTQSPDS LAVSLGERAT INCKSSQSLL NSRNRKNYLA WYQQKPDQSP KLLIYWASTR
ESGVPDRFSG SGSGTDFTLT ISSLQAEDVA VYYCKQSYYL WTFGGGTKVE IKRTVAAPSV
FIFPPSDEQL KSGTASVVCL LNNFYPREAK VQWKVDNALQ SGNSQESVTE QDSKDSTYSL
SSTLTLSKAD YEKHKVYACE VTHQGLSSPV TKSFNRGEC
(C chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFS TYAMNWVRQA PGKGLEWVGR IRSKYNNYAT
YYADSVKGRF TISRDDSKNT LYLQMNSLRA EDTAVYYCVR HGNFGDSYVS WFAYWGQGTL
VTVSSGKPGS GKPGSGKPGS GKPGSQAVVT QEPSLTVSPG GTVTLTCGSS TGAVTTSNYA
NWVQQKPGKS PRGLIGGTNK RAPGVPARFS GSLLGGKAAL TISGAQPEDE ADYYCALWYS
NHWVFGGGTK LTVLEPKSSD KTHTCPPCPA PPVAGPSVFL FPPKPKDTLM ISRTPEVTCV
VVDVKHEDPE VKFNWYVDGV EVHNAKTKPR EEQYNSTYRV VSVLTVLHQD WLNGKEYKCK
VSNKALPAPI EKTISKAKGQ PREPQVYTLP PSREQMTKNQ VKLTCLVKGF YPSDIAVEWE
SNGQPENNYK TTPPVLDSDG SFFLYSKLTV DKSRWQQGNV FSCSVMHEAL HNHYTQKSLS
LSPGK
(Disulfide bridge: A22-A96, A149-A205, A225-B219, A231-C265, A234-C268, A265-A325, A371-A429, B23-B94, B139-B199, C22-C98, C167-C235, C299-C359, C405-C463)
  Type
Peptide
Efficacy
Antineoplastic, Immunomodulator, Anti-somatostatin receptor 2 antibody
  Type
Bispecific antibody
Target
SSTR2 [HSA:6752] [KO:K04218]
CD3E [HSA:916] [KO:K06451]
  Pathway
hsa04024  cAMP signaling pathway
hsa04080  Neuroactive ligand-receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 G Protein-coupled receptors
  Rhodopsin family
   Somatostatin
    SSTR2
     D11845  Tidutamab (USAN/INN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3E
     D11845  Tidutamab (USAN/INN)
Other DBs
CAS: 2148354-90-7
PubChem: 433774520
LinkDB

» Japanese version   » Back

DBGET integrated database retrieval system