KEGG   DRUG: Sotigalimab
Entry
D12178                      Drug                                   
Name
Sotigalimab (USAN)
Formula
C6412H9970N1708O1993S46
Exact mass
144257.8461
Mol weight
144347.10
Sequence
(Heavy chain)
XVQLVESGGG VVQPGRSLRL SCAASGFSFS STYVCWVRQA PGKGLEWIAC IYTGDGTNYS
ASWAKGRFTI SKDSSKNTVY LQMNSLRAED TAVYFCARPD ITYGFAINFW GPGTLVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKKVEP KSCDKTHTCP PCPAPELLGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVE HEDPEVKFNW YVDGVEVHNA KTKPREEQYN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSRDE
LTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPG
(Light chain)
DIQMTQSPSS LSASVGDRVT IKCQASQSIS SRLAWYQQKP GKPPKLLIYR ASTLASGVPS
RFSGSGSGTD FTLTISSLQP EDVATYYCQC TGYGISWPIG GGTKVEIKRT VAAPSVFIFP
PSDEQLKSGT ASVVCLLNNF YPREAKVQWK VDNALQSGNS QESVTEQDSK DSTYSLSSTL
TLSKADYEKH KVYACEVTHQ GLSSPVTKSF NRGEC
(Disulfide bridge: H22-H96, H35-H50, H147-H203, H223-L215, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'96, H'35-H'50, H'147-H'203, H'223-L'215, H'264-H'324, H'370-H'428, L23-L88, L135-L195, L'23-L'88, L'135-L'195)
  Type
Peptide
Efficacy
Antineoplastic, Anti-CD40 antibody
  Type
Monoclonal antibody
Comment
Treatment of cancer
Target
TNFRSF5 (CD40) [HSA:958] [KO:K03160]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04514  Cell adhesion molecules
hsa04620  Toll-like receptor signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF5 (CD40)
     D12178  Sotigalimab (USAN)
Other DBs
CAS: 2305607-45-6
PubChem: 497620591
LinkDB

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