KEGG   DRUG: Uliledlimab
Entry
D12401                      Drug                                   
Name
Uliledlimab (USAN/INN)
Formula
C6430H9908N1704O2022S42
Exact mass
144691.3129
Mol weight
144780.48
Sequence
(Heavy chain)
EVQLQESGPG LVKPSETLSL TCAVSGYSIT SGYYWNWIRQ PPGKKLEWMG YINYGGSNGY
NPSLKSRITI SRDTSKNQFS LKLSSVTAAD TAVYYCARDY DAYYEALDDW GQGTTVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKKVEP KSCDKTHTCP PCPAPELLGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS HEDPEVKFNW YVDGVEVHNA KTKPREEQYA
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSREE
MTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPGK
(Light chain)
EIVLSQSPAT LSLSPGERAT LSCRASSRVN YMHWYQQKPG QSPRPWISAT SNLASGVPAR
FSGSGSGTSY TLTISSLEPE DFAVYYCQQW SSNPPTFGGG TKVEIKRTVA APSVFIFPPS
DEQLKSGTAS VVCLLNNFYP REAKVQWKVD NALQSGNSQE SVTEQDSKDS TYSLSSTLTL
SKADYEKHKV YACEVTHQGL SSPVTKSFNR GEC
(Disulfide bridge: H22-H96, H147-H203, H223-L213, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'96, H'147-H'203, H'223-L'213, H'264-H'324, H'370-H'428, L23-L87, L133-L193, L'23-L'87, L'133-L'193)
  Type
Peptide
Efficacy
Antineoplastic, Immunomodulator, Anti-CD73 antibody
  Type
Monoclonal antibody
Target
NT5E (CD73) [HSA:4907] [KO:K19970]
  Pathway
hsa00230  Purine metabolism
hsa00240  Pyrimidine metabolism
hsa00760  Nicotinate and nicotinamide metabolism
Brite
Target-based classification of drugs [BR:br08310]
 Enzymes
  Hydrolases (EC3)
   Phosphatases
    NT5E (CD73)
     D12401  Uliledlimab (USAN/INN)
Other DBs
CAS: 2378407-27-1
PubChem: 497620814
LinkDB

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