KEGG   DRUG: Surzebiclimab
Entry
D12429                      Drug                                   
Name
Surzebiclimab (USAN/INN)
Formula
C6428H9986N1716O2009S42
Exact mass
144706.0262
Mol weight
144795.17
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFS RYAMSWVRQA PGKGLEWVAA ISSGGSLYYP
DSVKGRFTIS RDNAKNTLYL QMNSLRAEDT AVYYCARGRE ADGGYFDYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP CPAPPAAGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSHE DPEVKFNWYV DGVEVHNAKT KPREEQYNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKALA APIEKTISKA KGQPREPQVY TLPPSRDELT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSK LTVDKSRWQQ
GNVFSCSVMH EALHNHYTQK SLSLSPGK
(Light chain)
EIVLTQSPAT LSVSPGERAT LSCRASESVE YYGTSLMQWY QQKPGQAPRL LIYAASNVES
GIPARFSGSG SGTEFTLTIS SLQSEDFAVY YCQQSLKVPL TFGGGTKVEI KRTVAAPSVF
IFPPSDEQLK SGTASVVCLL NNFYPREAKV QWKVDNALQS GNSQESVTEQ DSKDSTYSLS
STLTLSKADY EKHKVYACEV THQGLSSPVT KSFNRGEC
(Disulfide bridge: H22-H95, H146-H202, H222-L218, H231-H'231, H262-H322, H368-H426, H'22-H'95, H'146-H'202, H'222-L'218, H'262-H'322, H'368-H'426, L23-L92, L138-L198, L'23-L'92, L'138-L'198)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
HAVCR2 (CD366) [HSA:84868] [KO:K20414]
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    HAVCR2 (CD366)
     D12429  Surzebiclimab (USAN/INN)
Other DBs
CAS: 2342597-90-2
PubChem: 497620842
LinkDB

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