KEGG   DRUG: Ozekibart
Entry
D12458                      Drug                                   
Name
Ozekibart (USAN)
Formula
C4730H7216N1268O1428S32
Exact mass
105652.2076
Mol weight
105717.68
Sequence
EVQLLESGGG EVQPGGSLRL SCAASGLTFP NYGMGWFRQA PGKEREFVSA IYWSGGTVYY
AESVKGRFTI SRDNAKNTLY LQMSSLRAED TAVYYCAVTI RGAATQTWKY DYWGQGTLVT
VKPGGSGGSE VQLLESGGGE VQPGGSLRLS CAASGLTFPN YGMGWFRQAP GKEREFVSAI
YWSGGTVYYA ESVKGRFTIS RDNAKNTLYL QMSSLRAEDT AVYYCAVTIR GAATQTWKYD
YWGQGTLVTV KPGGGGDKTH TCPPCPAPGG PSVFLFPPKP KDTLMISRTP EVTCVVVDVS
HEDPEVKFNW YVDGVEVHNA KTKPREEQYN STYRVVSVLT VLHQDWLNGK EYKCKVSNKA
LPAPIEKTIS KAKGQPREPQ VYTLPPSRDE LTKNQVSLTC LVKGFYPSDI AVEWESNGQP
ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW QQGNVFSCSV MHEALHNHYT QKSLSLSPGK
(Disulfide bridge: 22-96, 151-225, 262-262', 265-265', 294-354, 400-458, 22'-96', 151'-225', 294'-354', 400'-458')
  Type
Peptide
Efficacy
Antineoplastic, Death receptor 5 agonit
  Type
Monoclonal antibody
Target
TNFRSF10B (TRAILR2, CD262) [HSA:8795] [KO:K04722]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04115  p53 signaling pathway
hsa04210  Apoptosis
hsa04217  Necroptosis
hsa04650  Natural killer cell mediated cytotoxicity
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF10B (TRAILR2, CD262)
     D12458  Ozekibart (USAN)
Other DBs
CAS: 2539847-03-3
PubChem: 497620871
LinkDB

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