KEGG   DRUG: Rocatinlimab
Entry
D12543                      Drug                                   
Name
Rocatinlimab (USAN/INN)
Formula
C6426H10000N1712O2000S42
Exact mass
144496.1692
Mol weight
144585.24
Sequence
(Heavy chain)
QITLKESGPT LVKPKQTLTL TCTFSGFSLS TSGMGVGWIR QPPGKALEWL AVIYWDDHQL
YSPSLKSRLT ITKDTSKNQV VLTMTNMDPV DTATYYCAHR RGAFQHWGQG TLVTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDKKVEPKSC DKTHTCPPCP APELLGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK PREEQYNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKALPA PIEKTISKAK GQPREPQVYT LPPSRDELTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCRASQSVS SSYLAWYQQK PGQAPRLLIY GASSRATGIP
DRFSGSGSGT DFTLTISRLE PEDFAVYYCQ QYDSSLTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H97, H144-H200, H220-L214, H226-H'226, H229-H'229, H261-H321, H367-H425, H'22-H'97, H'144-H'200, H'220-L'214, H'261-H'321, H'367-H'425, L23-L89, L134-L194, L'23-L'89, L'134-L'194)
  Type
Peptide
Efficacy
Immunomodulator, Anti-CD134 antibody
  Type
Monoclonal antibody
Comment
Treatment of atopic dermatitis and other immune mediated diseases
Target
TNFRSF4 (CD134, OX40) [HSA:7293] [KO:K05142]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF4 (CD134, OX40)
     D12543  Rocatinlimab (USAN/INN)
Other DBs
CAS: 2431972-52-8
PubChem: 497620956
LinkDB

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