KEGG   DRUG: Osemitamab
Entry
D12781                      Drug                                   
Name
Osemitamab (USAN/INN)
Formula
C6502H10052N1724O2036S48
Exact mass
146396.2624
Mol weight
146486.92
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT GYNMNWVRQA PGQGLEWMGN IDPYYGGTSY
NQKFKGRVTM TIDKSTSTVY MELSSLRSED TAVYYCARMY HGNAFDYWGQ GTTVTVSSAS
TKGPSVFPLA PSSKSTSGGT AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTQTYI CNVNHKPSNT KVDKKVEPKS CDKTHTCPPC PAPELLGGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSHE DPEVKFNWYV DGVEVHNAKT KPREEQYNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKALP APIEKTISKA KGQPREPQVY TLPPSRDELT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSK LTVDKSRWQQ
GNVFSCSVMH EALHNHYTQK SLSLSPGK
(Light chain)
DIVMTQSPDS LAVSLGERAT INCKSSQSLL NSGNLKNYLT WYQQKPGQPP KLLIYWASTR
KSGVPDRFSG SGSGTDFTLT ISSLQAEDVA VYYCQNDYSY PLTFGGGTKV EIKRTVAAPS
VFIFPPSDEQ LKSGTASVVC LLNNFYPREA KVQWKVDNAL QSGNSQESVT EQDSKDSTYS
LSSTLTLSKA DYEKHKVYAC EVTHQGLSSP VTKSFNRGEC
(Disulfide bridge: H22-H96, H221-L220, H145-H201, H227-H'227, H230-H'230, H262-H322, H368-H426, H'22-H'96, H'221-L'220, H'145-H'201, H'262-H'322, H'368-H'426, L23-L94, L140-L200, L'23-L'200)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Comment
Treatment of solid tumors
Target
CLDN18 [HSA:51208] [KO:K06087]
  Pathway
hsa04514  Cell adhesion molecules
hsa04530  Tight junction
hsa04670  Leukocyte transendothelial migration
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   Other
    CLDN18
     D12781  Osemitamab (USAN/INN)
Other DBs
CAS: 2460539-61-9
PubChem: 497621194
LinkDB

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