KEGG   DRUG: Verzistobart
Entry
D12798                      Drug                                   
Name
Verzistobart (USAN/INN)
Formula
C6392H9874N1714O2006S40
Exact mass
144021.2148
Mol weight
144109.75
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFR QNAWSWVRRA PGKGLEWVSA ISGSGGSTYY
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCAKGG DYGGNYFDYW GQGTLVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKRVEP KSCDKTHTCP PCPAPELLGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS HEDPEVKFNW YVDGVEVHNA KTKPREEQYA
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSREE
MTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPG
(Light chain)
EIVLTQSPAT LSLSPGERAT LSCRASQSVS SYLAWYQQKP GQAPRLLIYD ASNRATGIPA
SFSGSGSGTD FTLTISRLEP EDFAVYYCQQ YGSSPLTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H147-H203, H223-L214, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'96, H'147-H'203, H'223-L'214, H'264-H'324, H'370-H'428, L23-L88, L134-L194, L'23-L'88, L'134-'194)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
HAVCR2 (CD366) [HSA:84868] [KO:K20414]
  Pathway
hsa04148  Efferocytosis
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    HAVCR2 (CD366)
     D12798  Verzistobart (USAN/INN)
Other DBs
CAS: 2649466-18-0
PubChem: 497621211
LinkDB

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