KEGG   DRUG: Linavonkibart
Entry
D12801                      Drug                                   
Name
Linavonkibart (USAN/INN)
Formula
C6410H9876N1692O2032S48
Exact mass
144602.8072
Mol weight
144692.33
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCTASGFTFS SFSMDWVRQA PGKGLEWVSY ISPSADTIYY
ADSVKGRFTI SRDNAKNTLY LQMNSLRAED TAVYYCARGV LDYGDMLMPW GQGTLVTVSS
ASTKGPSVFP LAPCSRSTSE STAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTKT YTCNVDHKPS NTKVDKRVES KYGPPCPPCP APEFLGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSQED PEVQFNWYVD GVEVHNAKTK PREEQFNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKGLPS SIEKTISKAK GQPREPQVYT LPPSQEEMTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSRL TVDKSRWQEG
NVFSCSVMHE ALHNHYTQKS LSLSLG
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCQASQDIT NYLNWYQQKP GKAPKLLIYD ASNLETGVPS
RFSGSGSGTD FTFTISSLQP EDIATYYCQQ ADNHPPWTFG GGTKVEIKRT VAAPSVFIFP
PSDEQLKSGT ASVVCLLNNF YPREAKVQWK VDNALQSGNS QESVTEQDSK DSTYSLSSTL
TLSKADYEKH KVYACEVTHQ GLSSPVTKSF NRGEC
(Disulfide bridge: H22-H96, H134-L215, H147-H203, H226-H'226, H229-H'229, H261-H321, H367-H425, H'22-H'96, H'134-L'215, H'147-H'203, H'261-H'321, H'367-H'425, L23-L88, L135-L195, L'23-L'88, L'135-L'195)
  Type
Peptide
Efficacy
Antineoplastic, Transforming growth factor beta 1 inhibitor
  Type
Monoclonal antibody
Target
TGFB1 [HSA:7040] [KO:K13375]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04350  TGF-beta signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Transforming growth factors (RSTK-binding)
    TGFB1
     D12801  Linavonkibart (USAN/INN)
Other DBs
CAS: 2640981-30-0
PubChem: 497621214
LinkDB

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