KEGG   DRUG: Puxitatug
Entry
D12926                      Drug                                   
Name
Puxitatug (USAN/INN)
Formula
C6436H9968N1732O2006S40
Exact mass
144896.0057
Mol weight
144985.09
Sequence
(Heavy chain)
QVQLQQWGAG LLKPSETLSL ACTVYGGSFS GYYWNWIRQP PGKGLEWIGE INHSGSTSYN
PSLKSRVTIS VDTSKNQFSL KLSSVTAADT AVYYCARVLY NWNVDSWGQG TLVTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDKRVEPKSC DKTHTCPPCP APELLGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK PREEQYNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKALPA PIEKTISKAK GQPREPQVYT LPPSREEMTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRASQDIR NDVGWYQQKP GKAPKRLIYA ASRLQSGVPS
RFSGSGSGTE FTLTISSLQP EDFATYYCLQ HNSYPRTFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H95, H144-H200, H220-L214, H226-H'226, H229-H'229, H261-H321, H367-H425, H'22-H'95, H'144-H'200, H'220-L'214, H'261-H'321, H'367-H'425, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic, Immune checkpoint inhibitor
  Type
Monoclonal antibody
Target
B7H4 (VTCN1) [HSA:79679] [KO:K06747]
  Pathway
hsa04514  Cell adhesion molecules
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   Immune checkpoints
    B7H4 (VTCN1)
     D12926  Puxitatug (USAN/INN)
Other DBs
CAS: 2760250-47-1
PubChem: 497621339
LinkDB

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