KEGG   DRUG: Etentamig
Entry
D12990                      Drug                                   
Name
Etentamig (USAN/INN)
Formula
C5461H8419N1489O1726S39
Exact mass
123721.5895
Mol weight
123797.83
Sequence
(Heavy chain)
EVQLLESGGG LVQPGGSLRL SCAASGFTVS SYGMSWVRQA PGKGPEWVSG IRGSDGSTYY
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCAKQG ENDGPFDHRG QGTLVTVSSG
GGGSEVQLLE SGGGLVQPGG SLRLSCAASG FTVSSYGMSW VRQAPGKGPE WVSGIRGSDG
STYYADSVKG RFTISRDNSK NTLYLQMNSL RAEDTAVYYC AKQGENDGPF DHRGQGTLVT
VSSESKYGPP CPPCPAPEAA GGPSVFLFPP KPKDTLMISR TPEVTCVVVD VSQEDPEVQF
NWYVDGVEVH NAKTKPREEQ FNSTYRVVSV LTVLHQDWLN GKEYKCKVSN KGLPSSIEKT
ISKAKGQPRE PQVYTLPPSQ EEMTKNQVSL SCAVKGFYPS DIAVEWESNG QPENNYKTTP
PVLDSDGSFF LVSRLTVDKS RWQEGNVFSC SVMHEALHNH YTQKSLSLSL G
(heavy chain)
EVQLVESGGG LVQPGRSLRL SCAASGFTFD DYAMHWVRQA PGKGLEWVSG ISWNSGSIGY
ADSVKGRFTI SRDNAKNSLY LQMNSLRAED TALYYCAKDS RGYGDYRLGG AYWGQGTLVT
VSSASTKGPS VFPLAPCSRS TSESTAALGC LVKDYFPEPV TVSWNSGALT SGVHTFPAVL
QSSGLYSLSS VVTVPSSSLG TKTYTCNVDH KPSNTKVDKR VESKYGPPCP PCPAPEAAGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS QEDPEVQFNW YVDGVEVHNA KTKPREEQFN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKG LPSSIEKTIS KAKGQPREPQ VYTLPPSQEE
MTKNQVSLWC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SRLTVDKSRW
QEGNVFSCSV MHEALHNHYT QKSLSLSLG
(Light chain)
EIVMTQSPAT LSVSPGERAT LSCRASQSVS SNLAWYQQKP GQAPRLLIYG ASTRATGIPA
RFSGSGSGTE FTLTISSLQS EDFAVYYCQQ YNNWPWTFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H146-H220, H251-h229, H254-h232, H286-H346, H392-H450, h22-h96, h137-h206, h150-L214, h264-h324, h370-h428, L23-L88, L134-L194)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody, bispecific antibody
Target
CD3E [HSA:916] [KO:K06451]
TNFRSF17 (BCMA, CD269) [HSA:608] [KO:K05153]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04640  Hematopoietic cell lineage
hsa04660  T cell receptor signaling pathway
hsa04672  Intestinal immune network for IgA production
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF17 (BCMA, CD269)
     D12990  Etentamig (USAN/INN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3E
     D12990  Etentamig (USAN/INN)
Other DBs
CAS: 2490552-52-6
PubChem: 504099506
LinkDB

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