KEGG   DRUG: Dargistotug
Entry
D13000                      Drug                                   
Name
Dargistotug (USAN/INN)
Formula
C6444H9903N1693O2013S42
Exact mass
144556.2857
Mol weight
144645.52
Sequence
(Heavy chain)
QVQLVQSGSE LKKPGASVKV SCKASGYTFT SYPMNWVRQA PGQGLEWMGW INTNTGNPTY
AQGFTGRFVF SLDTSVSTAY LQISSLKAED TAVYYCARVG GYSVDEYAFD VWGQGTLVTV
SSASTKGPSV FPLAPSSKST SGGTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ
SSGLYSLSSV VTVPSSSLGT QTYICNVNHK PSNTKVDKRV EPKSCDKTHT CPPCPAPELL
GGPSVFLFPP KPKDTLMISR TPEVTCVVVD VSHEDPEVKF NWYVDGVEVH NAKTKPREEQ
YNSTYRVVSV LTVLHQDWLN GKEYKCKVSN KALPAPIEKT ISKAKGQPRE PQVYTLPPSR
EEMTKNQVSL TCLVKGFYPS DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSKLTVDKS
RWQQGNVFSC SVMHEALHNH YTQKSLSLSP G
(Light chain)
DIQLTQSPSF LSASVGDRVT ITCRASQGIS SYLAWYQQKP GKAPKLLIYA ASTLQSGVPS
RFSGSGSGTE FTLTISSLQP EDFATYYCQQ LSSYPTFGGG TKVEIKRTVA APSVFIFPPS
DEQLKSGTAS VVCLLNNFYP REAKVQWKVD NALQSGNSQE SVTEQDSKDS TYSLSSTLTL
SKADYEKHKV YACEVTHQGL SSPVTKSFNR GEC
(Disulfide bridge: H22-H96, H149-H205, H225-L213,H231-H'231, H234-H'234, H266-H326, H372-H430, H'22-H'96, H'149-H'205, H'225-L'213, H'266-H'326, H'372-H'430, L23-L88, L133-L193, L'23-L'88, L'133-L'193)
  Type
Peptide
Class
Antineoplastic
 DG02938  Immune checkpoint inhibitor
Efficacy
Antineoplastic, Immune checkpoint inhibitor, Anti-TIGIT receptor antibody
  Type
Monoclonal antibody
Target
TIGIT [HSA:201633] [KO:K16350]
  Pathway
hsa04514  Cell adhesion molecule (CAM) interaction
Brite
Drug groups [BR:br08330]
 Antineoplastic
  DG02938  Immune checkpoint inhibitor
   D13000  Dargistotug
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   Immune checkpoints
    TIGIT
     D13000  Dargistotug (USAN/INN)
Other DBs
CAS: 2649362-29-6
PubChem: 504099516
LinkDB

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