KEGG   DRUG: Abiprubart
Entry
D13033                      Drug                                   
Name
Abiprubart (USAN/INN)
Formula
C6400H9830N1698O2002S44
Exact mass
143912.7299
Mol weight
144001.64
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT NYWMHWVRQA PGQRLEWIGY INPSNDYTKY
NQKFKDRATL TADKSANTAY MELSSLRSED TAVYYCARQG FPYWGQGTLV TVSSASTKGP
SVFPLAPCSR STSESTAALG CLVKDYFPEP VTVSWNSGAL TSGVHTFPAV LQSSGLYSLS
SVVTVPSSSL GTKTYTCNVD HKPSNTKVDK RVESKYGPPC PPCPAPEFLG GPSVFLFPPK
PKDTLMISRT PEVTCVVVDV SQEDPEVQFN WYVDGVEVHN AKTKPREEQF NSTYRVVSVL
TVLHQDWLNG KEYKCKVSNK GLPSSIEKTI SKAKGQPREP QVYTLPPSQE EMTKNQVSLT
CLVKGFYPSD IAVEWESNGQ PENNYKTTPP VLDSDGSFFL YSRLTVDKSR WQEGNVFSCS
VMHEALHNHY TQKSLSLSPG K
(Light chain)
EIVLTQSPAT LSLSPGERAT LSCSASSSVS YMHWYQQKPG QAPRRWIYDT SKLASGVPAR
FSGSGSGTDY TLTISSLEPE DFAVYYCHQL SSDPFTFGGG TKVEIKRTVA APSVFIFPPS
DEQLKSGTAS VVCLLNNFYP REAKVQWKVD NALQSGNSQE SVTEQDSKDS TYSLSSTLTL
SKADYEKHKV YACEVTHQGL SSPVTKSFNR GEC
(Disulfide bridge: H22-H96, H128-L213, H141-H197, H220-H'220, H223-H'223, H255-H315, H361-H419, H'22-H'96, H'218-L'213, H'141-H'197, H'255-H'315, H'361-H'419, L23-L87, L133-L193, L'23-L'87, L'133-L'193)
  Type
Peptide
Efficacy
Immunosuppressant, Anti-CD40 antibody
  Type
Monoclonal antibody
Comment
Treatment of autoimmune diseases
Target
TNFRSF5 (CD40) [HSA:958] [KO:K03160]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04064  NF-kappa B signaling pathway
hsa04514  Cell adhesion molecule (CAM) interaction
hsa04620  Toll-like receptor signaling pathway
hsa04672  Intestinal immune network for IgA production
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF5 (CD40)
     D13033  Abiprubart (USAN/INN)
Other DBs
CAS: 2765071-95-0
PubChem: 505120122
LinkDB

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