KEGG   DRUG: Pacibekitug
Entry
D13049                      Drug                                   
Name
Pacibekitug (USAN/INN)
Formula
C6414H9878N1698O2008S48
Exact mass
144352.9633
Mol weight
144442.44
Sequence
(Heavy chain)
QVQLQQWGAG LLKPSETLSL TCAIYGGSFR EYYWSWIRQP PGKGLEWIGE IFHSGSTNYN
PSLKSRVTIS VDTSKNQFSL KLSSVTAADT AVYYCAREEL DDFDIWGQGT MVTVSSASTK
GPSVFPLAPC SRSTSESTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS NFGTQTYTCN VDHKPSNTKV DKTVERKCCV ECPPCPAPPV AGPSVFLFPP
KPKDTLMISR TPEVTCVVVD VSHEDPEVQF NWYVDGVEVH NAKTKPREEQ FNSTFRVVSV
LTVVHQDWLN GKEYKCKVSN KGLPAPIEKT ISKTKGQPRE PQVYTLPPSR EEMTKNQVSL
TCLVKGFYPS DIAVEWESNG QPENNYKTTP PMLDSDGSFF LYSKLTVDKS RWQQGNVFSC
SVMHEALHNH YTQKSLSLSP GK
(Lightc chain)
DIQMTQSPSS LSASVGDRVT ITCRASQGIS SWLAWYQQKP EKAPKSLIYA ASSLQSGVPS
RFSGSGSGTD FTLTISSLQP EDFATYYCQQ YKSYPRTFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H95, H130-L214, H143-H199, H218-H'218, H219-H'219, H222-H'222, H225-H'225, H256-H316, H362-H420, H'22-H'95, H'130-L'214, H'143-H'199, H'256-H'316, H'362-H'420, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Class
Immunological agent
 DG02019  Interleukin inhibitor
Efficacy
Anti-inflammatory, Anti-IL-6 antibody
  Type
Monoclonal antibody
Comment
Treatment of inflammatory conditions mediated by interleukin 6
Target
IL6 [HSA:3569] [KO:K05405]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04620  Toll-like receptor signaling pathway
hsa04630  JAK-STAT signaling pathway
Brite
Drug groups [BR:br08330]
 Immunological agent
  DG02019  Interleukin inhibitor
   D13049  Pacibekitug
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Interleukins
    IL6
     D13049  Pacibekitug (USAN/INN)
Other DBs
CAS: 2948444-06-0
PubChem: 505917322
LinkDB

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