KEGG   DRUG: Izalontamab
Entry
D13052                      Drug                                   
Name
Izalontamab (USAN/INN)
Formula
C8704H13394N2362O2774S52
Exact mass
197054.5101
Mol weight
197175.12
Sequence
(Heavy chain)
QVQLKQSGPG LVQPSQSLSI TCTVSGFSLT NYGVHWVRQS PGKGLEWLGV IWSGGNTDYN
TPFTSRLSIN KDNSKSQVFF KMNSLQSNDT AIYYCARALT YYDYEFAYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKRVEPK SCDKTHTCPP CPAPELLGGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPREEQYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSRDEL
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPGGG GGSGGGGSQV QLQESGGGLV KPGGSLRLSC
AASGFTFSSY WMSWVRQAPG KGLEWVANIN RDGSASYYVD SVKGRFTISR DDAKNSLYLQ
MNSLRAEDTA VYYCARDRGV GYFDLWGRGT LVTVSSGGGG SGGGGSGGGG SQSALTQPAS
VSGSPGQSIT ISCTGTSSDV GGYNFVSWYQ QHPGKAPKLM IYDVSDRPSG VSDRFSGSKS
GNTASLIISG LQADDEADYY CSSYGSSSTH VIFGGGTKVT VL
(Light chain)
DILLTQSPVI LSVSPGERVS FSCRASQSIG TNIHWYQQRT NGSPRLLIKY ASESISGIPS
RFSGSGSGTD FTLSINSVES EDIADYYCQQ NNNWPTTFGA GTKLELKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H95, H146-H202, H222-L214, H231-H'231, H263-H323, H369-H427, H480-H554, H613-H681, H'22-H'95, H'146-H'202, H'222-L'214, H'263-H'323, H'369-H'427, H'480-H'554, H'613-H'681, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody, bispecific antibody
Target
EGFR [HSA:1956] [KO:K04361]
ERBB3 (HER3) [HSA:2065] [KO:K05084]
  Pathway
hsa04012  ErbB signaling pathway
hsa04151  PI3K-Akt signaling pathway
hsa05200  Pathways in cancer
Brite
Target-based classification of drugs [BR:br08310]
 Protein kinases
  Receptor tyrosine kinases (RTK)
   EGFR family
    EGFR
     D13052  Izalontamab (USAN/INN)
    ERBB3 (HER3)
     D13052  Izalontamab (USAN/INN)
Other DBs
CAS: 2559704-24-2
PubChem: 505917325
LinkDB

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