KEGG   DRUG: Trosunilimab
Entry
D13087                      Drug                                   
Name
Trosunilimab (USAN/INN)
Formula
C6380H9862N1690O2002S44
Exact mass
143592.9557
Mol weight
143681.63
Sequence
(Heavy chain)
EVQLVQSGAE VKKPGSSVKV SCKASGFNIK NTYMHWVRQA PGQGLEWIGR IDPAKGHTEY
APKFLGRVTI TADESTNTAY MELSSLRSED TAVYYCYYVD VWGQGTTVTV SSASTKGPSV
FPLAPSSKST SGGTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ SSGLYSLSSV
VTVPSSSLGT QTYICNVNHK PSNTKVDKKV EPKSCDKTHT CPPCPAPELL GGPSVFLFPP
KPKDTLMISR TPEVTCVVVD VSHEDPEVKF NWYVDGVEVH NAKTKPREEQ YNSTYRVVSV
LTVLHQDWLN GKEYKCKVSN KALPAPIEKT ISKAKGQPRE PQVYTLPPSR EEMTKNQVSL
TCLVKGFYPS DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSKLTVDKS RWQQGNVFSC
SVMHEALHNH YTQKSLSLSP GK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCHASQDIS DNIGWLQQKP GKSFKLLIYH GTNLEDGVPS
RFSGSGSGTD YTLTISSLQP EDFATYYCVQ YAQFPWTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H139-H195, H215-L214, H221-H'221, H224-H'224, H256-H316, H362-H420, H'22-H'96, H'139-H'195, H'215-L'214, H'256-H'316, H'362-H'420, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Immunomodulator, Anti-alpha4/beta7 integrin antibody
  Type
Monoclonal antibody
Comment
Treatment of HIV infection
Target
ITGA4/ITGB7 [HSA:3676 3695] [KO:K06483 K06590]
  Pathway
hsa04510  Focal adhesion
hsa04512  ECM-receptor interaction
hsa04514  Cell adhesion molecules
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Cell adhesion molecules: other families
   Integrins
    ITGA4/ITGB7
     D13087  Trosunilimab (USAN/INN)
Other DBs
CAS: 2550297-60-2
PubChem: 508750757
LinkDB

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