KEGG   DRUG: Coramitug
Entry
D13140                      Drug                                   
Name
Coramitug (USAN/INN)
Formula
C6574H10152N1736O2042S48
Exact mass
147625.0513
Mol weight
147716.56
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLKL SCAASGFTFS SYTMSWVRQT PEKRLELVAE INNSGDTTYY
PDTVKGRFTI SRDNAKNTLY LQMSSLKSED TAMYYCARHY YYGGGYGGWF FDVWGQGTLV
TVSSASTKGP SVFPLAPSSK STSGGTAALG CLVKDYFPEP VTVSWNSGAL TSGVHTFPAV
LQSSGLYSLS SVVTVPSSSL GTQTYICNVN HKPSNTKVDK RVEPKSCDKT HTCPPCPAPE
LLGGPSVFLF PPKPKDTLMI SRTPEVTCVV VDVSHEDPEV KFNWYVDGVE VHNAKTKPRE
EQYNSTYRVV SVLTVLHQDW LNGKEYKCKV SNKALPAPIE KTISKAKGQP REPQVYTLPP
SREEMTKNQV SLTCLVKGFY PSDIAVEWES NGQPENNYKT TPPVLDSDGS FFLYSKLTVD
KSRWQQGNVF SCSVMHEALH NHYTQKSLSL SPGK
(Light chain)
DIVMTQSPLS LPVTPGEPAS ISCRSSKSLL HSNGNTYLYW FLQKPGQSPQ LLIYRVSNLA
SGVPSRFSGS GSGTDFTLKI SRVEAEDVGV YYCMQHLEYP LTFGQGTKLE IKRTVAAPSV
FIFPPSDEQL KSGTASVVCL LNNFYPREAK VQWKVDNALQ SGNSQESVTE QDSKDSTYSL
SSTLTLSKAD YEKHKVYACE VTHQGLSSPV TKSFNRGEC
(Disulfide bridge: H22-H96, H151-H207, H227-L219, H233-H'233, H236-H'236, H268-H328, H374-H432, H'22-H'96, H'151-H'207, H'227-L'219, H'268-H'328, H'374-H'432, L23-L93, L139-L199, L'23-L'93, L'139-L'199)
  Type
Peptide
Efficacy
Anti-transthyretin misfolded
  Type
Monoclonal antibody
Comment
Treatment of hereditary or wild-type ATTR CM
Target
TTR [HSA:7276] [KO:K20731]
  Pathway
hsa04918  Thyroid hormone synthesis
Brite
Target-based classification of drugs [BR:br08310]
 Transporters
  Other transporters
   Others
    TTR
     D13140  Coramitug (USAN/INN)
Other DBs
CAS: 2626841-92-5
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