KEGG   DRUG: Mavrostobart
Entry
D13146                      Drug                                   
Name
Mavrostobart (USAN/INN)
Formula
C6540H10048N1718O2045S42
Exact mass
146716.3345
Mol weight
146806.84
Sequence
(Heavy chain)
EVQLVESGGG LVQPGQSLKL SCKASGYAFS SYWMNWVKQR PGKGLEWIGQ IYPGDGDTYY
SGKFKGRATL SADKSKNTAY LQLNNLRAED TAVYYCAREA IYYGNYVFTY WGQGTLVTVS
SASTKGPSVF PLAPCSRSTS ESTAALGCLV KDYFPEPVTV SWNSGALTSG VHTFPAVLQS
SGLYSLSSVV TVPSSSLGTK TYTCNVDHKP SNTKVDKRVE SKYGPPCPPC PAPEFLGGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSQE DPEVQFNWYV DGVEVHNAKT KPREEQFNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKGLP SSIEKTISKA KGQPREPQVY TLPPSQEEMT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSR LTVDKSRWQE
GNVFSCSVMH EALHNHYTQK SLSLSLGK
(Light chain)
DIVMTQSPSL LSASLGDRVT ISCKSSQSLL NSSNQKNYLA WYQQKPGQSP KLLVYFASTR
DSGVPDRFSG SGSGTDFTLT ISSLEPEDFA TYFCQQHYST PLTFGAGTKL EIKRTVAAPS
VFIFPPSDEQ LKSGTASVVC LLNNFYPREA KVQWKVDNAL QSGNSQESVT EQDSKDSTYS
LSSTLTLSKA DYEKHKVYAC EVTHQGLSSP VTKSFNRGEC
(Disulfide bridge: H22-H96, H135-H148, H204-L220, H227-H'227, H230-H'230, H262-H322, H368-H426, H'22-H'96, H'135-H'148, H'204-L'220, H'262-H'322, H'368-H'426, L23-L94, L140-L200, L'23-L'94, L'140-L'200)
  Type
Peptide
Efficacy
Antineoplastic, Anti-CD73 antibody
  Type
Monoclonal antibody
Target
NT5E (CD73) [HSA:4907] [KO:K19970]
  Pathway
hsa00230  Purine metabolism
hsa00240  Pyrimidine metabolism
hsa00760  Nicotinate and nicotinamide metabolism
hsa01232  Nucleotide metabolism
Brite
Target-based classification of drugs [BR:br08310]
 Enzymes
  Hydrolases (EC3)
   Phosphatases
    NT5E (CD73)
     D13146  Mavrostobart (USAN/INN)
Other DBs
CAS: 2928515-12-0
PubChem: 518038668
LinkDB

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