KEGG   DRUG: レミグロミグ
エントリ  
D13162                      Drug                                   
一般名   
レミグロミグ;
Remigromig (USAN)
組成式   
C8812H13568N2370O2812S62
質量    
199565.4238
分子量   
199688.36
配列    
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFDFT AYAMHWVRQA PGKGLEWVAS IYPSGGYTAY
ADSVKGRFTI SADTSKNTAY LQMNSLRAED TAVYYCARRS YYFALDYWGQ GTLVTVSSGG
GGSDIQMTQS PSSLSASVGD RVTITCRASQ SVSSAVAWYQ QKPGKAPKLL IYSASSLYSG
VPSRFSGSRS GTDFTLTISS LQPEDFATYY CQQYWAYYSP ITFGQGTKVE IKGGGGSGGG
GSEPKSSDKT HTCPPCPAPE AAGGPSVFLF PPKPKDTLMI SRTPEVTCVV VDVSHEDPEV
KFNWYVDGVE VHNAKTKPRE EQYNSTYRVV SVLTVLHQDW LNGKEYKCKV SNKALPASIE
KTISKAKGQP REPMVFDLPP SREEMTKNQV SLWCMVKGFY PSDIAVEWES NGQPENNYKT
TPPVLDSDGS FFLYSKLTVD KSRWQQGNVF SCSVMHEALH NHYTQKSLSL SPGKGGGSGG
GSGGGSGGGS GSTGEVQLVE SGGGLVQPGG SLRLSCAASG FTLSSYSMHW VRQAPGKGLE
WVAYISSYDS ITDYADSVKG RFTISADTSK NTAYLQMNSL RAEDTAVYYC ARPAVGHMAF
DYWGQGTLVT VSSASTKGPS VFPLAPSSKS TSGGTAALGC LVKDYFPEPV TVSWNSGALT
SGVHTFPAVL QSSGLYSLSS VVTVPSSSLG TQTYICNVNH KPSNTKVDKK VEPKSCDKTH
T
(heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFDFS SSSIHWVRQA PGKGLEWVAS ISSSYGYTYY
ADSVKGRFTI SADTSKNTAY LQMNSLRAED TAVYYCARSW AMDYWGQGTL VTVSSGGGGS
DIQMTQSPSS LSASVGDRVT ITCRASQSVS SAVAWYQQKP GKAPKLLIYS ASDLYSGVPS
RFSGSRSGTD FTLTISSLQP EDFATYYCQQ YAGAGLITFG QGTKVEIKGG GGSGGGGSEP
KSSDKTHTCP PCPAPEAAGG PSVFLFPPKP KDTLMISRTP EVTCVVVDVS HEDPEVKFNW
YVDGVEVHNA KTKPREEQYN STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPASIEKTIS
KAKGQPREPQ VYTLPPIREL MTSNQVSLSC AVKGFYPSDI AVEWESNGQP ENNYKTTPPV
LDSDGSFFLV SKLTVDKSRW QQGNVFSCSV MHEALHNHYT QKSLSLSPGK GGGSGGGSGG
GSGGGSGSTG EVQLVESGGG LVQPGGSLRL SCAASGFTLS SYSMHWVRQA PGKGLEWVAY
ISSYDSITDY ADSVKGRFTI SADTSKNTAY LQMNSLRAED TAVYYCARPA VGHMAFDYWG
QGTLVTVSSA STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH
TFPAVLQSSG LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHT
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRASQSVS SAVAWYQQKP GKAPKLLIYS ASSLYSGVPS
RFSGSRSGTD FTLTISSLQP EDFATYYCQQ WYNAPITFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H146-H211, H2534-h249, H256-h252, H288-H348, H394-H452, H516-H590, H640-H696, H716-L214, h22-h96, h143-h208, h284-h344, h390-h448, h51-h586, h636-h692, h712-L'214, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  タイプ
Peptide
効能    
網膜疾患治療薬
  タイプ
多重特異性抗体
ターゲット 
LRP5 [HSA:4041] [KO:K03068]
SFRP4 [HSA:6424] [KO:K02185]
  パスウェイ
hsa04150  mTOR シグナル伝達経路
hsa04310  Wnt シグナル伝達経路
hsa04928  副甲状腺ホルモンの合成、分泌、作用
hsa05022  神経変性のパスウェイ - 多疾患
階層分類  
ターゲットに基づく医薬品分類 [BR:jp08310]
 他に分類されないもの
  環境情報処理
   Wnt シグナリング
    SFRP4
     D13162  レミグロミグ
リンク   
CAS: 3059389-31-7
PubChem: 518520882
LinkDB    

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