KEGG   DRUG: Nivisnebart
Entry
D13210                      Drug                                   
Name
Nivisnebart (USAN/INN)
Formula
C6450H10038N1740O2025S48
Exact mass
145806.2580
Mol weight
145896.38
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT KYYMSWVRQA PGQGLEWMGI INPIGGSTSY
AQKFQGRVTM TRDTSTSTVY MELSSLRSED TAVYYCARDP SGIALAGPAS RGYQGMDVWG
QGTTVTVSSA STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH
TFPAVLQSSG LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP
CPAPEAAGGP SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK
TKPREEQYNS TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PASIEKTISK AKGQPREPQV
YTLPPSRDEL TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS
KLTVDKSRWQ QGNVFSCSVM HEALHNHYTQ KSLSLSPGK
(Light chain)
EIVMTQSPAT LSVSPGERAT LSCRASQSVS SNLAWYQQKP GQAPRLLIYG ASTRATGIPA
RFSGSGSGTE FTLTISSLQS EDFAVYYCQQ ARLGPWTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H156-H212, H232-L214, H238-H'238, H241-H'241, H273-H333, H379-H437, H'22-H'96, H'156-H'212, H'232-L'214, H'273-H'333, H'379-H'437, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Neurodegenerative diseases agent, Anti-sortilin antibody
  Type
Monoclonal antibody
Comment
Treatment of Alzheimer's disease and Parkinson's disease
Target
SORT1 [HSA:6272] [KO:K12388]
  Pathway
hsa04722  Neurotrophin signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Not elsewhere classified
  Cellular process
   Membrane trafficking
    SORT1
     D13210  Nivisnebart (USAN/INN)
Other DBs
CAS: 2923556-87-8
LinkDB

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