KEGG   DRUG: Cenzestotug
Entry
D13258                      Drug                                   
Name
Cenzestotug (USAN/INN)
Formula
C6380H9886N1706O1992S42
Exact mass
143617.2994
Mol weight
143705.80
Sequence
(Heavy chain)
QVQLVESGGG VVQPGRSLRI SCAVSGFSLT SYGVLWVRQA PGKGLEWLGV IWSGGSTDYN
AAFISRLTIS RDNSKSTVYF QMNSLRAEDT AVYYCAREEF GYWGQGTLVT VSSASTKGPS
VFPLAPSSKS TSGGTAALGC LVKDYFPEPV TVSWNSGALT SGVHTFPAVL QSSGLYSLSS
VVTVPSSSLG TQTYICNVNH KPSNTKVDKK VEPKSCDKTH TCPPCPAPEL LGGPSVFLFP
PKPKDTLMIS RTPEVTCVVV DVSHEDPEVK FNWYVDGVEV HNAKTKPREE QYNSTYRVVS
VLTVLHQDWL NGKEYKCKVS NKALPAPIEK TISKAKGQPR EPQVYTLPPS REEMTKNQVS
LTCLVKGFYP SDIAVEWESN GQPENNYKTT PPVLDSDGSF FLYSKLTVDK SRWQQGNVFS
CSVMHEALHN HYTQKSLSLS PGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRASQDIN NYLNWYQQKP GGAVKLLIYY TSRLHTGVPS
RFSGSGSGTD FTLTISSLQP EDIATYYCQQ TNTLPWTFGG GTKLEVKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H95, H140-H196, H216-L214, H222-H'222, H225-H'225, H257-H317, H363-H421, H'22-H'95, H'140-H'196, H'216-L'214, H'257-H'317, H'363-H'421, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Comment
Treatment of solid tumors
Target
TNFRSF4 (CD134, OX40) [HSA:7293] [KO:K05142]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Signaling molecules and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF4 (CD134, OX40)
     D13258  Cenzestotug (USAN/INN)
Other DBs
CAS: 3014361-58-8
PubChem: 527701161
LinkDB

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