KEGG   DRUG: Ixotatug
Entry
D13271                      Drug                                   
Name
Ixotatug (USAN/INN)
Formula
C6444H9918N1718O2006S44
Exact mass
144873.4597
Mol weight
144962.95
Sequence
(Heavy chain)
EVQLLESGGG LVQPGGSMRL SCAASGFTFS NYWMNWVRQA PGKGLEWVAQ IRLKSDNYAT
HYADSVKGRF TISRDDSKNT VYLQMNSLRA EDTGVYYCND GPPSGSWGQG TLLTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDKKVEPKSC DKTHTCPPCP APELLGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK PREEQYNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKALPA PIEKTISKAK GQPREPQVYT LPPSRDELTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRISENIY SYLAWYQQKP GKAPKLLVYN AKILVEGVPS
RFSGSGSGTD FTLTISSLQP EDFGTYYCQH HYTVPWTFGQ GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H98, H144-H200, H220-L214, H226-H'226, H229-H'229, H261-H321, H367-H425, H'22-H'98, H'144-H'200, H'220-L'214, H'261-H'321, H'367-H'425, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic, Anti-claudin 6 antibody
  Type
Monoclonal antibody
Target
CLDN6 [HSA:9074] [KO:K06087]
  Pathway
hsa04514  Cell adhesion molecule (CAM) interaction
hsa04530  Tight junction
hsa04670  Leukocyte transendothelial migration
Other DBs
CAS: 3018936-99-4
PubChem: 527701174
LinkDB

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