KEGG   DGROUP: CYP3A4 inhibitor
Entry
DG01522                     DGroup                                 
Name
CYP3A4 inhibitor
Type
Metabolism
Member
D00282  
Clotrimazole (JP18/USP/INN)  <JP/US>
Cimetidine
 D00295  
Cimetidine (JP18/USP/INN)  <JP/US>
 D03503  
Cimetidine hydrochloride (USP)  <US>
D10246  
Omeprazole, clarithromycin and amoxicillin  <US>
D08774  
Amoxicillin hydrate, clarithromycin and lansoprazole  <US>
D10519  
Rabeprazole, amoxicillin and clarithromycin  <JP>
D10775  
Vonoprazan, amoxicillin and clarithromycin  <JP>
Aprepitant
 D02968  
Aprepitant (JAN/USP/INN)  <JP/US>
 D10895  
Fosaprepitant (INN)
 D06597  
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN)  <JP/US>
D09394  
Fidaxomicin (JAN/USAN)  <JP/US>
Teneligliptin
 D08616  
Teneligliptin (INN)
 D09756  
Teneligliptin hydrobromide hydrate (JAN)  <JP>
 D11968  
Teneligliptin hydrobromide (JAN)
Berotralstat
 D11673  
Berotralstat (USAN/INN)
 D11674  
Berotralstat hydrochloride (JAN/USAN)  <JP/US>
Verapamil
 D02356  
Verapamil (USAN/INN)
 D00619  
Verapamil hydrochloride (JP18/USP)  <JP/US>
D00351  
Ketoconazole (JP18/USP)  <JP/US>
Fluconazole
 D00322  
Fluconazole (JP18/USP/INN)  <JP/US>
 D01429  
Fosfluconazole (JAN/INN)  <JP>
D01980  
Luliconazole (JAN/USAN/INN)  <JP/US>
Bromocriptine
 D03165  
Bromocriptine (USAN/INN)
 D00780  
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18)  <JP/US>
Ethinylestradiol
 D00554  
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN)  <JP>
 D07928  
Ethinylestradiol propanesulfonate
Midecamycin
 D01339  
Midecamycin (JP18/INN)
 D01636  
Midecamycin acetate (JP18)
Josamycin
 D01235  
Josamycin (JP18/USAN/INN)
 D05351  
Josamycin propionate (JP18)
D01322  
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN)
Clarithromycin
 D00276  
Clarithromycin (JP18/USP/INN)  <JP/US>
 D07710  
Clarithromycin lactobionate
D00854  
Quinupristin and dalfopristin
D00350  
Itraconazole (JP18/USP)  <JP/US>
D02555  
Posaconazole (JAN/USAN/INN)  <JP/US>
Indinavir
 C07051  
Indinavir
 D03833  
Indinavir (USAN)
 D00897  
Indinavir sulfate (USP)
 D02861  
Indinavir sulfate ethanolate (JAN)
Nelfinavir
 D08259  
Nelfinavir (INN)
 D00899  
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN)  <US>
Fosamprenavir
 D02497  
Fosamprenavir (INN)
 D02867  
Fosamprenavir calcium hydrate (JAN)
 D03835  
Fosamprenavir calcium (USAN)  <US>
 D03837  
Fosamprenavir sodium (USAN)
Atazanavir
 D07471  
Atazanavir (INN)
 D01276  
Atazanavir sulfate (JAN/USAN)  <US>
Darunavir
 D03656  
Darunavir (USAN/INN)  <US>
 D06478  
Darunavir ethanolate (JAN)  <JP/US>
 D12637  
Darunavir hydrate  <US>
 D12752  
Darunavir propylene glycolate  <US>
D09012  
Telaprevir (JAN/USAN/INN)
D10582  
Dasabuvir, ombitasvir, paritaprevir and ritonavir
D10745  
Ombitasvir, paritaprevir and ritonavir
D00753  
Sirolimus (JAN/USAN/INN)  <JP/US>
D00961  
Bicalutamide (JP18/USP/INN)  <JP/US>
D00960  
Anastrozole (JP18/USP/INN)  <JP/US>
D00184  
Cyclosporine (USP); Ciclosporin (JP18)  <JP/US>
D05928  
Stiripentol (JAN/USAN/INN)  <JP>
D04641  
Istradefylline (JAN/USAN/INN)  <JP/US>
Fluvoxamine
 D07984  
Fluvoxamine (INN)
 D00824  
Fluvoxamine maleate (JP18/USP)  <JP/US>
D08837  
Aclidinium bromide (JAN/USAN/INN)  <JP/US>
D00707  
Fomepizole (JAN/USAN/INN)  <JP/US>
D09799  
Carotegrast methyl (JAN)  <JP>
 » expand
Class
Metabolizing enzyme inhibitor
 DG02852  CYP3A/CYP3A4 inhibitor
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