KEGG   DRUG: Dusigitumab
Entry
D10352                      Drug                                   
Name
Dusigitumab (USAN/INN)
Formula
C6372H9824N1700O2016S54
Exact mass
144142.3386
Mol weight
144231.98
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT SYDINWVRQA TGQGLEWMGW MNPNSGNTGY
AQKFQGRVTM TRNTSISTAY MELSSLRSED TAVYYCARDP YYYYYGMDVW GQGTTVTVSS
ASTKGPSVFP LAPCSRSTSE STAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSNFGTQT YTCNVDHKPS NTKVDKTVER KCCVECPPCP APPVAGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVQFNWYVDG VEVHNAKTKP REEQFNSTFR
VVSVLTVVHQ DWLNGKEYKC KVSNKGLPAP IEKTISKTKG QPREPQVYTL PPSREEMTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPMLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPGK
(Light chain)
QSVLTQPPSV SAAPGQKVTI SCSGSSSNIE NNHVSWYQQL PGTAPKLLIY DNNKRPSGIP
DRFSGSKSGT SATLGITGLQ TGDEADYYCE TWDTSLSAGR VFGGGTKLTV LGQPKAAPSV
TLFPPSSEEL QANKATLVCL ISDFYPGAVT VAWKADSSPV KAGVETTTPS KQSNNKYAAS
SYLSLTPEQW KSHRSYSCQV THEGSTVEKT VAPTECS
(Disulfide bridge: H22-H96, H134-L216, H147-H203, H222-H'222, H223-H'223, H226-H'226, H229-H'229, H260-H320, H366-H424, H'22-H'96, H'134-L'216, H'147-H'203, H'260-H'320, H'366-H'424, L22-L89, L139-L198, L'22-L'89, L'139-L'198)
  Type
Peptide
Efficacy
Antineoplastic, Anti-insulin-like growth factor 2 antibody
  Type
Monoclonal antibody
Target
IGF2 [HSA:3481] [KO:K13769]
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Growth factors (RTK-binding)
    IGF2
     D10352  Dusigitumab (USAN/INN)
Other DBs
CAS: 1204390-13-5
PubChem: 172232445
LinkDB

» Japanese version   » Back

DBGET integrated database retrieval system