KEGG   DRUG: Acapatamab
Entry
D12121                      Drug                                   
Name
Acapatamab (USAN)
Formula
C4691H7162N1262O1462S38
Exact mass
105781.4262
Mol weight
105847.18
Sequence
QVQLVESGGG LVKPGESLRL SCAASGFTFS DYYMYWVRQA PGKCLEWVAI ISDGGYYTYY
SDIIKGRFTI SRDNAKNSLY LQMNSLKAED TAVYYCARGF PLLRHGAMDY WGQGTLVTVS
SGGGGSGGGG SGGGGSDIQM TQSPSSLSAS VGDRVTITCK ASQNVDTNVA WYQQKPGQAP
KSLIYSASYV YWDVPSRFSG SASGTDFTLT ISSVQSEDFA TYYCQQYDQQ LITFGCGTKL
EIKSGGGGSE VQLVESGGGL VQPGGSLKLS CAASGFTFNK YAMNWVRQAP GKGLEWVARI
RSKYNNYATY YADSVKDRFT ISRDDSKNTA YLQMNNLKTE DTAVYYCVRH GNFGNSYISY
WAYWGQGTLV TVSSGGGGSG GGGSGGGGSQ TVVTQEPSLT VSPGGTVTLT CGSSTGAVTS
GNYPNWVQQK PGQAPRGLIG GTKFLAPGTP ARFSGSLLGG KAALTLSGVQ PEDEAEYYCV
LWYSNRWVFG GGTKLTVLGG GGDKTHTCPP CPAPELLGGP SVFLFPPKPK DTLMISRTPE
VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPCEEQYGS TYRCVSVLTV LHQDWLNGKE
YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSREEM TKNQVSLTCL VKGFYPSDIA
VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ QGNVFSCSVM HEALHNHYTQ
KSLSLSPGKG GGGSGGGGSG GGGSGGGGSG GGGSGGGGSD KTHTCPPCPA PELLGGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP CEEQYGSTYR
CVSVLTVLHQ DWLNGKEYKC KVSNKALPAP IEKTISKAKG QPREPQVYTL PPSREEMTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPGK
(Disulfide birdge: 22-96, 44-236, 159-224, 271-347, 411-479, 508-765, 511-768, 543-603, 574-584, 649-707, 800-860, 831-841, 906-964)
  Type
Peptide
Efficacy
Antineoplastic, PSMA antibody
  Type
Bispecific antibody
Comment
Treatment of prostate cancer
Target
FOLH1 (PSMA) [HSA:2346] [KO:K14592]
CD3E [HSA:916] [KO:K06451]
  Pathway
hsa04658  Th1 and Th2 cell differentiation
hsa04659  Th17 cell differentiation
hsa04660  T cell receptor signaling pathway
hsa04981  Folate transport and metabolism
hsa05215  Prostate cancer
Brite
Target-based classification of drugs [BR:br08310]
 Peptidases and inhibitors
  Metallo peptidases
   Family M28
    FOLH1 (PSMA)
     D12121  Acapatamab (USAN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3E
     D12121  Acapatamab (USAN)
Other DBs
PubChem: 497620534
LinkDB

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