KEGG   DRUG: Nezastomig
Entry
D12566                      Drug                                   
Name
Nezastomig (USAN)
Formula
C6488H9983N1723O2024S43
Exact mass
145792.9201
Mol weight
145882.89
Sequence
(Heavy chain)
QVQLVESGGG VVQPGRSLRL SCAASGFTFS SYGMHWVRQA PGKGLEWVAF MSYDGSNKFY
SDSVKGRFTI SRDNSRKMLF LQMNNLRAED TAVYYCARDQ YYDFLTDHGV FDYWGQGTLV
TVSSASTKGP SVFPLAPCSR STSESTAALG CLVKDYFPEP VTVSWNSGAL TSGVHTFPAV
LQSSGLYSLS SVVTVPSSSL GTKTYTCNVD HKPSNTKVDK RVESKYGPPC PPCPAPPVAG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS QEDPEVQFNW YVDGVEVHNA KTKPREEQFN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKG LPSSIEKTIS KAKGQPREPQ VYTLPPSQEE
MTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SRLTVDKSRW
QEGNVFSCSV MHEALHNHYT QKSLSLSLGK
(heavy chain)
QVQLQESGPG LVKPSETLSL TCTVSGGSIS SYYWSWIRQP PGKGLEWIGY IYYSGITHYN
PSLKSRVTIS VDTSKIQFSL KLSSVTAADT AVYYCARWGV RRDYYYYGMD VWGQGTTVTV
SSASTKGPSV FPLAPCSRST SESTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ
SSGLYSLSSV VTVPSSSLGT KTYTCNVDHK PSNTKVDKRV ESKYGPPCPP CPAPPVAGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSQE DPEVQFNWYV DGVEVHNAKT KPREEQFNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKGLP SSIEKTISKA KGQPREPQVY TLPPSQEEMT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSR LTVDKSRWQE
GNVFSCSVMH EALHNRFTQK SLSLSPGK
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCRASQSVS SSYLAWYQQK PGQAPRLLIY GASSRATGIP
DRFSGSGSGT DFTLTISRLE PEDFAVYYCQ QYGSSPWTFG QGTKVEIKRT VAAPSVFIFP
PSDEQLKSGT ASVVCLLNNF YPREAKVQWK VDNALQSGNS QESVTEQDSK SDTYSLSSTL
TLSKADYEKH KVYACEVTHQ GLSSPVTKSF NRGEC
(Disulfide bridge: H22-H96, H138-L215, H151-H207, H230-h228, H223-h231, H264-H324, H370-H428, h22-h95, h136-L'215, h149-h205, h262-h322, h368-h426, L23-L89, L135-L195, L'23-L'89, L'135-L'195)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Bispecific antibody
Comment
Treatment of prostate cancer
Target
FOLH1 (PSMA) [HSA:2346] [KO:K14592]
CD28 [HSA:940] [KO:K06470]
  Pathway
hsa04514  Cell adhesion molecule (CAM) interaction
hsa04660  T cell receptor signaling pathway
hsa04672  Intestinal immune network for IgA production
hsa04981  Folate transport and metabolism
hsa05215  Prostate cancer
Brite
Target-based classification of drugs [BR:br08310]
 Peptidases and inhibitors
  Metallo peptidases
   Family M28
    FOLH1 (PSMA)
     D12566  Nezastomig (USAN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD28
     D12566  Nezastomig (USAN)
Other DBs
CAS: 2657613-60-8
PubChem: 497620979
LinkDB

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