KEGG   DRUG: Forimtamig
Entry
D12724                      Drug                                   
Name
Forimtamig (USAN/INN)
Formula
C8551H13244N2300O2698S58
Exact mass
193175.3647
Mol weight
193294.32
Sequence
(A chain)
EVQLLESGGG LVQPGGSLRL SCAASGFTFS KYAMAWVRQA PGKGLEWVAS ISTGGVNTYY
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCATHT GDYFDYWGQG TMVTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVEDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDEKVEPKSC DGGGGSGGGG SQAVVTQEPS
LTVSPGGTVT LTCGSSTGAV TTSNYANWVQ EKPGQAFRGL IGGTNKRAPG TPARFSGSLL
GGKAALTLSG AQPEDEAEYY CALWYSNLWV FGGGTKLTVL SSASTKGPSV FPLAPSSKST
SGGTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ SSGLYSLSSV VTVPSSSLGT
QTYICNVNHK PSNTKVDKKV EPKSCDKTHT CPPCPAPEAA GGPSVFLFPP KPKDTLMISR
TPEVTCVVVD VSHEDPEVKF NWYVDGVEVH NAKTKPREEQ YNSTYRVVSV LTVLHQDWLN
GKEYKCKVSN KALGAPIEKT ISKAKGQPRE PQVYTLPPCR DELTKNQVSL WCLVKGFYPS
DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSKLTVDKS RWQQGNVFSC SVMHEALHNH
YTQKSLSLSP GK
(B chain)
EVQLLESGGG LVQPGGSLRL SCAASGFTFS KYAMAWVRQA PGKGLEWVAS ISTGGVNTYY
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCATHT GDYFDYWGQG TMVTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVEDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDEKVEPKSC DKTHTCPPCP APEAAGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK PREEQYNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKALGA PIEKTISKAK GQPREPQVCT LPPSRDELTK
NQVSLSCAVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLVSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(C chain)
EVQLLESGGG LVQPGGSLRL SCAASGFQFS SYAMNWVRQA PGKGLEWVSR IRSKYNNYAT
YYADSVKGRF TISRDDSKNT LYLQMNSLRA EDTAVYYCVR HTTFPSSYVS YYGYWGQGTL
VTVSSASVAA PSVFIFPPSD EQLKSGTASV VCLLNNFYPR EAKVQWKVDN ALQSGNSQES
VTEQDSKDST YSLSSTLTLS KADYEKHKVY ACEVTHQGLS SPVTKSFNRG EC
(D chain)
EIVLTQSPGT LSLSPGERAT LSCRASQSVS ISGINLMNWY QQKPGQQPKL LIYHASILAS
GIPDRFSGSG SGTDFTLTIS RLEPEDFAVY YCQQTRESPL TFGQGTRLEI KRTVAAPSVF
IFPPSDRKLK SGTASVVCLL NNFYPREAKV QWKVDNALQS GNSQESVTEQ DSKDSTYSLS
STLTLSKADY EKHKVYACEV THQGLSSPVT KSFNRGEC
(Disulfide bridge: A22-A96, A144-A200, A220-D218, A253-A321, A369-A425, A445-C232, A451-B226, A454-B229, A486-A546, A579-B34, A592-A650, B22-B96, B144-B200, B220-D'218, B261-B321, B367-B425, C22-C98, C152-C212, D23-D92, D138-D198, D'23-D'92, D'138-D'198)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Bispecific antibody
Target
GPRC5D [HSA:55507] [KO:K04621]
CD3E [HSA:916] [KO:K06451]
  Pathway
hsa04640  Hematopoietic cell lineage
hsa04658  Th1 and Th2 cell differentiation
hsa04659  Th17 cell differentiation
hsa04660  T cell receptor signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 G Protein-coupled receptors
  Metabotropic glutamate receptor family
   Orphan GPRC5
    GPRC5D
     D12724  Forimtamig (USAN/INN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3E
     D12724  Forimtamig (USAN/INN)
Other DBs
CAS: 2649379-96-2
PubChem: 497621137
LinkDB

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