KEGG   DRUG: Etalanetug
Entry
D12848                      Drug                                   
Name
Etalanetug (USAN)
Formula
C6626H10212N1732O2112S40
Exact mass
149117.3759
Mol weight
149208.98
Sequence
(Heavy chain)
EVQLLESGGG LVQPGGSLRL SCAASGYTFT TYWITWVRQA PGKGLEWVSD IYPGSSISNY
NEKFKSRFTI SVDNSKNTLY LQMNSLRAED TAVYYCARED GYDAWFAYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP CPAPELLGGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPREEQYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSRDEL
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPG
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRSSQSIL HSNGNTYLEW YQQKPGKAPK LLISKVSNRF
SGVPSRFSGS GSGTDFTLTI SSLQPEDFAT YYCFQGSHVP FTFGQGTKLE IKRTVAAPSV
FIFPPSDEQL KSGTASVVCL LNNFYPREAK VQWKVDNALQ SGNSQESVTE QDSKDSTYSL
SSTLTLSKAD YEKHKVYACE VTHQGLSSPV TKSFNRGEC
(Disulfide bridge: H22-H96, H146-H202, H222-L219, H228-H'228, H231-H'231, H263-H323, H369-H427, H'22-H'96, H'146-H'202, H'222-L'219, H'263-H'323, H'369-H'427, L23-L93, L139-L199, L'23-L'93, L'139-L'199)
  Type
Peptide
Efficacy
Dementia therapeutic agent, Anti-tau protein antibody
  Type
Monoclonal antibody
Comment
Treatment of Alzheimer's disease
Target
MAPT (TAU) [HSA:4137] [KO:K04380]
  Pathway
hsa04010  MAPK signaling pathway
hsa05010  Alzheimer disease
Brite
Target-based classification of drugs [BR:br08310]
 Not elsewhere classified
  Cellular process
   Cytoskeleton
    MAPT (TAU)
     D12848  Etalanetug (USAN)
Other DBs
CAS: 2690265-18-8
PubChem: 497621261
LinkDB

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