KEGG   DRUG: Ruxoprubart
Entry
D12857                      Drug                                   
Name
Ruxoprubart (USAN)
Formula
C6482H10004N1712O2024S44
Exact mass
145620.0226
Mol weight
145709.98
Sequence
(Heavy chain)
QVQLVQSGAE VAKPGASVKM SCKASGYTFT NYWIHWVKQR PGQGLEWIGY INPNTGYNDY
NQKFKDKATL TADKSSSTVY MQLSSLTSED TAVYYCARGG QLGLRRAMDY WGQGTLVTVS
SASTKGPSVF PLAPSSKSTS GGTAALGCLV KDYFPEPVTV SWNSGALTSG VHTFPAVLQS
SGLYSLSSVV TVPSSSLGTQ TYICNVNHKP SNTKVDKKVE PKSCDKTHTC PPCPAPELLG
GPSVFLFPPK PKDTLMISRT PEVTCVVVDV SHEDPEVKFN WYVDGVEVHN AKTKPREEQY
ASTYRVVSVL TVLHQDWLNG KEYKCKVSNK ALPAPIEKTI SKAKGQPREP QVYTLPPSRD
ELTKNQVSLT CLVKGFYPSD IAVEWESNGQ PENNYKTTPP VLDSDGSFFL YSKLTVDKSR
WQQGNVFSCS VMHEALHNHY TQKSLSLSPG K
(Light chain)
DVQITQSPSY LSASPGDTIT ITCRASKSIS KYLAWYQDKP GKTNKLLIYS GSTLQSGIPS
RFSGSGSGTE FTLTISSLQP DDFAMYYCQQ HDEYPWTFGQ GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H148-H204, H224-L214, H230-H'230, H233-H'233, H265-H325, H371-H429, H'22-H'96, H'148-H'204, H'224-L'214, H'265-H'325, H'371-H'429, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Anti complement factor B antibody
  Type
Monoclonal antibody
Comment
Treatment of complement mediated diseases
Target
CFB [HSA:629] [KO:K01335]
  Pathway
hsa04610  Complement and coagulation cascades
Brite
Target-based classification of drugs [BR:br08310]
 Peptidases and inhibitors
  Serine peptidases
   Chymotrypsin family
    CFB
     D12857  Ruxoprubart (USAN)
Other DBs
CAS: 2842046-67-5
PubChem: 497621270
LinkDB

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