KEGG   DRUG: Velaprumig
Entry
D13359                      Drug                                   
Name
Velaprumig (USAN/INN)
Formula
C4457H6895N1215O1451S28
Exact mass
101550.5276
Mol weight
101612.58
Sequence
(A chain)
DIVLTQSPAT LSVSPGERAT ISCRASQRVS SSTYSYMHWY QQKPGQPPKL LIKYASNLES
GVPARFSGSG SGTDFTLTIS SVEPEDFATY YCQHSWEIPP TTGGGTKLEI KRGGGGSGGG
GSGGGGSQVQ LVQSGAEVVK PGASVKLSCK ASGYIFTSYY MYWVKQAPGQ GLEWIGEINP
SNGDTNFNEK FKSKATLTVD KSASTAYMEL SSLRSEDTAV YYCTRSDGRN DMDSWGQGTL
VTVSSGGGGS GGGGSGGGGS QVQLVQSGGG PVKPGGSLRL SCAASGFMFR AYSMNWVRQA
PGKGLEWVSS ISSSGRYIHY ADSVKGRFTI SRDNAKNSLY LQMNSLRAED TAVYYCARET
VMAGKALDYW GQGTLVTVSS ASTKGPSVFP LAPSSKSTSE GTAALGCLVK DYFPEPVTVS
WNSGALTSGV HTFPAVLQSS GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKKVEP
KSS
(B chain)
DIVLTQSPAT LSVSPGERAT ISCRASQRVS SSTYSYMHWY QQKPGQPPKL LIKYASNLES
GVPARFSGSG SGTDFTLTIS SVEPEDFATY YCQHSWEIPP TFGGGTKLEI KRGGGGSGGG
GSGGGGSQVQ LVQSGAEVVK PGASVKLSCK ASGYIFTSYY MYWVKQAPGQ GLEWIGEINP
SNGDTNFNEK FKSKATLTVD KSASTAYMEL SSLRSEDTAV YYCTRSDGRN DMDSWGQGTL
VTVSSGSTSG SGKPGSGEGS TKGDIVLTQS PGTLSLSPGE TATLSCRASQ SVGSNLAWYQ
QKPGQAPRLL IYGASTGATG VPARFSGSRS GTDFTLTITS LQPEDFATYY CQQYYSFLAK
TFGQGTQLEI KRTVAAPSVF IFPPSDEQLK SGTASVVCLL NNFYPREAKV QWKVDNALQS
GNSQESVTEQ DSKDSTYSLS NTLTLSKADY EKHKVYACEV THQGLSSPVT KSFNRGES
(Disulfide bridge: A23-A92, A149-A223, A282-A356, A407-A463, B23-B92, B149-B223, B286-B351, B398-B458)
  Type
Peptide
Efficacy
Immunosuppressant, Anti-CD40 ligand antibody
  Type
Bispecific antibody
Comment
Treatment of thyroid eye disease (TED, Graves' ophthalmopathy)
Target
TNFSF5 (CD40L, CD154) [HSA:959] [KO:K03161]
ALB [HSA:213] [KO:K16141]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04514  Cell adhesion molecule (CAM) interaction
hsa04660  T cell receptor signaling pathway
hsa04672  Intestinal immune network for IgA production
Brite
Target-based classification of drugs [BR:br08310]
 Not elsewhere classified
  Organismal systems
   Circulatory system
    ALB
     D13359  Velaprumig (USAN/INN)
Other DBs
CAS: 2988741-17-7
PubChem: 530451558
LinkDB

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