| Flutamide-type antiandrogen |
| Flutamide (JP18/USP/INN) <JP/US> |
| Nilutamide (USAN/INN) <US> |
| Bicalutamide (JP18/USP/INN) <JP/US> |
| Enzalutamide (JAN/USAN) <JP/US> |
| Apalutamide (JAN/INN) <JP/US> |
| Darolutamide (JAN/USAN/INN) <JP/US> |
| Deutenzalutamide (USAN) |
| Steroid-type antiandrogen |
| Cyproterone |
| Cyproterone (INN) |
| Cyproterone acetate (JAN/USAN) |
| Abiraterone acetate (JAN/USP) <JP/US> |
| Oxendolone (JAN/USAN/INN) |
| Benorterone (USAN/INN) |
| Topterone (USAN/INN) |
| Zanoterone (USAN/INN) |
| Galeterone (USAN) |
| Clascoterone (USAN) <US> |
| Chlormadinone |
| Chlormadinone (INN) |
| Chlormadinone acetate (JP18/USAN) <JP> |
| Delmadinone |
| Delmadinone (INN) |
| Delmadinone acetate (USAN) |
| Cioteronel (USAN/INN) |
| Clometherone (USAN/INN) |
