Homo sapiens (human): 1132
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Entry
1132 CDS
T01001
Symbol
CHRM4, HM4, M4R
Name
(RefSeq) cholinergic receptor muscarinic 4
KO
K04132
muscarinic acetylcholine receptor M4
Organism
hsa
Homo sapiens (human)
Pathway
hsa04080
Neuroactive ligand-receptor interaction
hsa04725
Cholinergic synapse
hsa04810
Regulation of actin cytoskeleton
Drug target
Acetylcholine (
DG01133
):
D00999
<JP/US>
Aclatonium (
DG01291
):
D01955
Aclidinium bromide:
D08837
<JP/US>
Anisotropine methylbromide:
D00232
Atropine (
DG00052
):
D00113
D02069
<JP/US>
Atropine oxide (
DG01243
):
D03011
D07477
Batefenterol (
DG01627
):
D10545
D10546
Benapryzine hydrochloride:
D03076
Benzatropine (
DG00859
):
D00778
<US>
D07511
Benzetimide (
DG01301
):
D03087
D07513
Benzilone:
D03088
Bethanechol (
DG00991
):
D01000
<JP/US>
Bevonium:
D01532
Biperiden (
DG00852
):
D00779
D02246
<JP>
D02247
<JP>
Blarcamesine (
DG03048
):
D11383
D11549
Bornaprine:
D07302
Butropium bromide:
D01491
Butylscopolamine:
D01451
<JP>
Carbachol:
D00524
<US>
Carpronium (
DG01289
):
D01175
<JP>
D09752
<JP>
Chlorpromazine (
DG00867
):
D00270
D00789
<JP/US>
D03274
D04034
<JP>
D09819
Choline alfoscerate:
D07349
Cimetropium bromide:
D07099
Clidinium bromide:
D00716
Cyclopentolate (
DG01141
):
D01002
<JP/US>
D07759
Darotropium bromide:
D09402
Dexetimide (
DG00856
):
D03711
D07804
Diethazine (
DG01921
):
D02603
D07823
Difemerine:
D07079
Dihexyverine (
DG00033
):
D03824
D07821
Diphenidol (
DG02880
):
D01318
<JP>
D03858
D03859
Diphenylpiperidinomethyldioxolan iodide:
D01600
Diponium bromide:
D01463
Elantrine:
D03970
Elucaine:
D03979
Emraclidine:
D12468
Etomidoline:
D01359
Etybenzatropine:
D04087
Eucatropine hydrochloride:
D04116
Fenpiverinium:
D07070
Fentonium:
D07951
Flutropium bromide:
D02417
Glycopyrronium (
DG02467
):
D10939
<JP/US>
Heteronium bromide:
D04434
Homatropine (
DG01142
):
D01004
Homatropine methylbromide:
D02070
Hyoscyamine (
DG00053
):
D00147
D00719
D01648
D04479
Ipratropium bromide:
D02212
<JP/US>
Mazaticol (
DG00857
):
D03264
D08157
Mebeverine (
DG00030
):
D04868
D08160
Mepenzolate (
DG00040
):
D00720
<JP>
Methacholine:
D04970
<JP/US>
Methantheline (
DG00036
):
D00721
Methscopolamine bromide:
D00715
<US>
Methylatropine (
DG01242
):
D01077
D03814
Methylbenactyzium bromide:
D01315
Methylscopolamine:
D01976
<JP>
Metixene (
DG00853
):
D01871
D08209
Metoquizine:
D05012
Milameline hydrochloride:
D05035
Otilonium bromide:
D07083
Oxapium iodide:
D01815
Oxitropium bromide:
D01946
Oxybutynin (
DG00478
):
D00465
<US>
D00722
<JP/US>
Parapenzolate bromide:
D05360
Pentapiperium methylsulfate:
D05418
Penthienate:
D07081
Phencarbamide:
D05452
Phenglutarimide:
D07301
Pipenzolate:
D07084
Piperidolate (
DG00034
):
D01165
<JP>
D08382
Pipethanate (
DG01255
):
D01521
D08384
Pipethanate ethobromide:
D01987
Pirenzepine (
DG00026
):
D01297
D05276
<JP>
D08389
Piroheptine (
DG01272
):
D01231
<JP>
D08395
Poldine:
D05535
Pridinol (
DG00774
):
D02064
<JP>
D08418
D08419
Prifinium bromide:
D01377
Procyclidine (
DG00854
):
D00782
D08425
Profenamine (
DG00855
):
D01118
D03276
D08426
Propantheline (
DG00035
):
D00481
<JP>
Propenzolate hydrochloride:
D05628
Propiverine (
DG00479
):
D01007
<JP>
D08441
Rapacuronium bromide:
D05703
Rocuronium bromide:
D00765
<JP/US>
Scopolamine (
DG00065
):
D00138
<US>
D02071
Tazomeline citrate:
D06015
Tematropium methylsulfate:
D06061
Tiemonium (
DG01254
):
D08595
Tiemonium iodide:
D01201
Timepidium bromide (
DG00041
):
D02535
<JP>
Tofenacin hydrochloride:
D06175
Toquizine:
D06192
Triampyzine sulfate:
D06217
Trihexyphenidyl (
DG00851
):
D00787
<JP/US>
D08638
Tropatepine (
DG00858
):
D07303
D08653
Tropicamide:
D00397
<JP/US>
Umeclidinium (
DG01253
):
D10180
Umeclidinium bromide:
D10181
<JP/US>
Valethamate:
D01538
Xanomeline (
DG01300
):
D06330
D06331
Brite
KEGG Orthology (KO) [BR:
hsa00001
]
09130 Environmental Information Processing
09133 Signaling molecules and interaction
04080 Neuroactive ligand-receptor interaction
1132 (CHRM4)
09140 Cellular Processes
09142 Cell motility
04810 Regulation of actin cytoskeleton
1132 (CHRM4)
09150 Organismal Systems
09156 Nervous system
04725 Cholinergic synapse
1132 (CHRM4)
09180 Brite Hierarchies
09183 Protein families: signaling and cellular processes
04030 G protein-coupled receptors [BR:
hsa04030
]
1132 (CHRM4)
G protein-coupled receptors [BR:
hsa04030
]
Rhodopsin family
Biogenic amine
Acetylcholine (muscarinic)
1132 (CHRM4)
BRITE hierarchy
SSDB
Ortholog
Paralog
Gene cluster
GFIT
Motif
Pfam:
7tm_1
7TM_GPCR_Srsx
7tm_4
Motif
Other DBs
NCBI-GeneID:
1132
NCBI-ProteinID:
NP_000732
OMIM:
118495
HGNC:
1953
Ensembl:
ENSG00000180720
UniProt:
P08173
Structure
PDB
LinkDB
All DBs
Position
11:complement(46383789..46391776)
Genome browser
AA seq
479 aa
AA seq
DB search
MANFTPVNGSSGNQSVRLVTSSSHNRYETVEMVFIATVTGSLSLVTVVGNILVMLSIKVN
RQLQTVNNYFLFSLACADLIIGAFSMNLYTVYIIKGYWPLGAVVCDLWLALDYVVSNASV
MNLLIISFDRYFCVTKPLTYPARRTTKMAGLMIAAAWVLSFVLWAPAILFWQFVVGKRTV
PDNQCFIQFLSNPAVTFGTAIAAFYLPVVIMTVLYIHISLASRSRVHKHRPEGPKEKKAK
TLAFLKSPLMKQSVKKPPPGEAAREELRNGKLEEAPPPALPPPPRPVADKDTSNESSSGS
ATQNTKERPATELSTTEATTPAMPAPPLQPRALNPASRWSKIQIVTKQTGNECVTAIEIV
PATPAGMRPAANVARKFASIARNQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMV
LVNTFCQSCIPDTVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR
NT seq
1440 nt
NT seq
+upstream
nt +downstream
nt
atggccaacttcacacctgtcaatggcagctcgggcaatcagtccgtgcgcctggtcacg
tcatcatcccacaatcgctatgagacggtggaaatggtcttcattgccacagtgacaggc
tccctgagcctggtgactgtcgtgggcaacatcctggtgatgctgtccatcaaggtcaac
aggcagctgcagacagtcaacaactacttcctcttcagcctggcgtgtgctgatctcatc
ataggcgccttctccatgaacctctacaccgtgtacatcatcaagggctactggcccctg
ggcgccgtggtctgcgacctgtggctggccctggactacgtggtgagcaacgcctccgtc
atgaaccttctcatcatcagctttgaccgctacttctgcgtcaccaagcctctcacctac
cctgcccggcgcaccaccaagatggcaggcctcatgattgctgctgcctgggtactgtcc
ttcgtgctctgggcgcctgccatcttgttctggcagtttgtggtgggtaagcggacggtg
cccgacaaccagtgcttcatccagttcctgtccaacccagcagtgacctttggcacagcc
attgctgccttctacctgcctgtggtcatcatgacggtgctgtacatccacatctccctg
gccagtcgcagccgagtccacaagcaccggcccgagggcccgaaggagaagaaagccaag
acgctggccttcctcaagagcccactaatgaagcagagcgtcaagaagcccccgcccggg
gaggccgcccgggaggagctgcgcaatggcaagctggaggaggcccccccgccagcgctg
ccaccgccaccgcgccccgtggctgataaggacacttccaatgagtccagctcaggcagt
gccacccagaacaccaaggaacgcccagccacagagctgtccaccacagaggccaccacg
cccgccatgcccgcccctcccctgcagccgcgggccctcaacccagcctccagatggtcc
aagatccagattgtgacgaagcagacaggcaatgagtgtgtgacagccattgagattgtg
cctgccacgccggctggcatgcgccctgcggccaacgtggcccgcaagttcgccagcatc
gctcgcaaccaggtgcgcaagaagcggcagatggcggcccgggagcgcaaagtgacacga
acgatctttgccattctgctagccttcatcctcacctggacgccctacaacgtcatggtc
ctggtgaacaccttctgccagagctgcatccctgacacggtgtggtccattggctactgg
ctctgctacgtcaacagcaccatcaaccctgcctgctatgctctgtgcaacgccaccttt
aaaaagaccttccggcacctgctgctgtgccagtatcggaacatcggcactgccaggtag
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