KEGG   DRUG: イムボタマブ
エントリ  
D12567                      Drug                                   
一般名   
イムボタマブ;
Imvotamab (USAN/INN)
組成式   
C43154H66961N11627O13563S349
質量    
976243.9933
分子量   
976849.57
配列    
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFI SYTMHWVRQA PGQGLEWMGY INPRSGYTHY
NQKLKDKATL TADKSASTAY MELSSLRSED TAVYYCARSA YYDYDGFAYW GQGTLVTVSS
GGGGSGGGGS GGGGSDIQMT QSPSSLSASV GDRVTITCSA SSSVSYMNWY QQKPGKAPKR
LIYDTSKLAS GVPSRFSGSG SGTDFTLTIS SLQPEDFATY YCQQWSSNPP TFGGGTKVEI
KGGGGSGGGG SGGGGSQEDE RIVLVDNKCK CARITSRIIR SSEDPNEDIV ERNIRIIVPL
NNRENISDPT SPLRTRFVYH LSDLCKKCDP TEVELDNQIV TATQSNICDE DSATETCYTY
DRNKCYTAVV PLVYGGETKM VETALTPDAC YPDGGGGSGG GGSGGGGSDA HKSEVAHRFK
DLGEENFKAL VLIAFAQYLQ QCPFEDHVKL VNEVTEFAKT CVADESAENC DKSLHTLFGD
KLCTVATLRE TYGEMADCCA KQEPERNECF LQHKDDNPNL PRLVRPEVDV MCTAFHDNEE
TFLKKYLYEI ARRHPYFYAP ELLFFAKRYK AAFTECCQAA DKAACLLPKL DELRDEGKAS
SAKQRLKCAS LQKFGERAFK AWAVARLSQR FPKAEFAEVS KLVTDLTKVH TECCHGDLLE
CADDRADLAK YICENQDSIS SKLKECCEKP LLEKSHCIAE VENDEMPADL PSLAADFVES
KDVCKNYAEA KDVFLGMFLY EYARRHPDYS VVLLLRLAKT YETTLEKCCA AADPHECYAK
VFDEFKPLVE EPQNLIKQNC ELFKQLGEYK FQNALLVRYT KKVPQVSTPT LVEVSRNLGK
VGSKCCKHPE AKRMPCAEDY LSVVLNQLCV LHEKTPVSDR VTKCCTESLV NRRPCFSALE
VDETYVPKEF NAETFTFHAD ICTLSEKERQ IKKQTALVEL VKHKPKATKE QLKAVMDDFA
AFVEKCCKAD DKETCFAEEG KKLVAASQAA LGL
(heavy chain A-J)
EVQLVQSGAE VKKPGESLKI SCKGSGYSFT SYWIGWVRQM PGKGLEWMGI IYPGDSDTRY
SPSFQGQVTI SADKSITTAY LQWSSLKASD TAMYYCARHP SYGSGSPNFD YWGQGTLVTV
SSGSASAPTL FPLVSCENSP SDTSSVAVGC LAQDFLPDSI TFSWKYKNNS DISSTRGFPS
VLRGGKYAAT SQVLLPSKDV MQGTDEHVVC KVQHPNGNKE KNVPLPVIAE LPPKVSVFVP
PRDGFFGNPR KSKLICQATG FSPRQIQVSW LREGKQVGSG VTTDQVQAEA KESGPTTYKV
TSTLTIKESD WLSQSMFTCR VDHRGLTFQQ NASSMCVPDQ DTAIRVFAIP PSFASIFLTK
STKLTCLVTD LTTYDSVTIS WTRQNGEAVK THTNISESHP NATFSAVGEA SICEDDWNSG
ERFTCTVTHT DLPSPLKQTI SRPKGVALHR PDVYLLPPAR EQLNLRESAT ITCLVTGFSP
ADVFVQWMQR GQPLSPEKYV TSAPMPEPQA PGRYFAHSIL TVSEEEWNTG ETYTCVVAHE
ALPNRVTERT VDKSTGKPTL YNVSLVMSDT AGTCY
(Light chain a-j)
DIVMTQTPLS SPVTLGQPAS ISCRSSQSLV YSDGNTYLSW LQQRPGQPPR LLIYKISNRF
SGVPDRFSGS GAGTDFTLKI SRVEAEDVGV YYCVQATQFP LTFGGGTKVE IKRTVAAPSV
FIFPPSDEQL KSGTASVVCL LNNFYPREAK VQWKVDNALQ SGNSQESVTE QDSKDSTYSL
SSTLTLSKAD YEKHKVYACE VTHQGLSSPV TKSFNRGEC
(Disulfide bridge: H22-H96, H158-H222, H269-H357, H271-hA574, H325-hJ574, H328-H348, H365-H390, H461-H470, H483-H499, H498-H509, H532-H577, H576-H585, H608-H654, H653-H771, H673-H687, H686-H697, H724-H769, H768-H777, H800-H846, H845-H856, H869-H885, H884-H895, H922-H967, H966-H975, hA22-hA96, hA136-La219, hA150-hA210, hA256-hA319, hA336-hB336, hA366-hA425, hA413-hB413, hA473-hA535, hB22-hB96, hB136-Lb219, hB150-hB210, hB256-hB319, hB366-hB425, hB473-hB535, hB574-hC425, hB473-hB535, hB574-hC574, hC22-hC96, hC136-Lc219, hC22-hC96, hC136-Lc219, hC150-hC210, hC256-hC319, hC336-hD336, hC366-hC425, hC413-hD413, hC473-hC535, hD22-hD96, hD136-Ld219, hD150-hD210, hD256-hD319, hD366-hD425, hD473-hD535, hD574-hE574, hE22-hE96, hE136-Le219, hE150-hE210, hE256-hE319, hE336-hF336, hE366-hE425, hE413-hF413, hE473-hE535, hF22-hF96, hF136-Lf219, hF150-Hf210, hF256-hF319, hF256-hF319, hF366-hF425, hF473-hF535, hF574-hG574, hG22-hG96, hG136-Lg219, hG150-hG210, hG256-hG319, hG336-hH336, hG366-hG425, hG413-hH413, hG473-hG535, hH22-hH96, hH136-Lh219, hH150-hH210, hH256-hH319, hH366-hH425, hH473-hH535, hH574-hI574, hI22-hI96, hI136-hJ219, hI150-hI210, hI256-hI319, hI336-hJ336, hI366-hI425, hI413-hJ413, hI473-hI535, hJ136-Lj219, hJ150-hJ210, hJ256-hJ319, hJ366-hJ425, hJ473-hJ535, La23-La93, La139-La199, Lb23-Lb93, Lb139-Lb199, Lc23-Lc93, Lc139-Lc199, Ld23-Ld93, Ld139-Ld199, Le23-Le93, Le139-Le199, Lf23-Lf93, Lf139-Lf199, Lg23-Lg93, Lg139-Lg199, Lh23-Lh93, Lh139-Lh199, Li23-Li93, Li139-Li199, Lj23-Lj93, Lj139-Lj199)
  タイプ
Peptide
効能    
抗悪性腫瘍薬
  タイプ
モノクローナル抗体
ターゲット 
CD20 [HSA:931] [KO:K06466]
CD3E [HSA:916] [KO:K06451]
  パスウェイ
hsa04640  造血細胞系譜
階層分類  
ターゲットに基づく医薬品分類 [BR:jp08310]
 細胞表面分子とリガンド
  その他の細胞表面分子
   CD 分子
    CD3E
     D12567  イムボタマブ
    CD20
     D12567  イムボタマブ
リンク   
CAS: 2573121-53-4
PubChem: 497620980
LinkDB    

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