KEGG   DRUG: スペバタミグ
エントリ  
D13158                      Drug                                   
一般名   
スペバタミグ;
Spevatamig (USAN/INN)
組成式   
C6450H9972N1714O2013S44
質量    
145055.8343
分子量   
145145.41
配列    
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFIFS SFGMHWVRKA PGKGLEWVAY ISSGRSTMYY
ADSVKGRFTI SRDNSKNTLY LQMNSLTAED TAVYYCARGG FYGNSLDYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSKVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP CPAPELLGGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPREEQYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV CTLPPSRDEL
TKNQVSLSCA VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLVS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPGK
(heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT SYWMHWVREA PGQGLEWIGN IDPSDSETHY
AQKFQGRVTL TVDKSTSTVY MELSSLRSED TAVYYCAGTD LAYWGQGTLV TVSSASTKGP
SVFPLAPSSC STSGGTAALG CLVKDYFPEP VTVSWNSGAL TSEVHTFPAV LQSSGLYSLS
SVVTVPSSSL GTQTYICNVN HKPSNTKVDK KVEPKSSDKT HTCPPCPAPE LLGGPSVFLF
PPKPKDTLMI SRTPEVTCVV VDVSHEDPEV KFNWYVDGVE VHNAKTKPRE EQYNSTYRVV
SVLTVLHQDW LNGKEYKCKV SNKALPAPIE KTISKAKGQP REPQVYTLPP CRDELTKNQV
SLWCLVKGFY PSDIAVEWES NGQPENNYKT TPPVLDSDGS FFLYSKLTVD KSRWQQGNVF
SCSVMHEALH NHYTQKSLSL SPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCKSSLSLL NSGNQKNYLT WYQEKPGKAP KLLIYWASTR
ESGVPSRFSG SGSGTDFTLT ISSLQPEDFA TYSCQNAYSY PLTFGQGTKV EIKRTVAAPE
VFIFPPSDEQ LKSGTASVVC LLNNFYPREA KVQWKVDNAL QSGNSQESVT EQDSKDSTYS
LSSTLTLSKA DYEKHKVYAC EVTHQGLSSP VTKSFNRGEC
(light chain)
EIVLTQSPGT LSLSPGERAT LSCHASQNIN VWLSWYQKKP GQAPRLLIYK ASNLHTGIPD
RFSGSGSGTD FTLTISRLEP EDFAVYYCQQ GQSYPFTFGQ GTKVEIKRTV AAPKVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSCN RGES
(Disulfide bridge: H22-H96, H146-H202, H222-L220, H228-l223, H231-h226, H351-h351, H263-H323, H369-H427, h22-h96, h130-l209, h141-h197, h258-h318, h364-h422, L23-L94, L140-L200, l23-l88, l134-l194)
  タイプ
Peptide
効能    
抗悪性腫瘍薬
  タイプ
二重特異性抗体
ターゲット 
CLDN18 [HSA:51208] [KO:K06087]
CD47 [HSA:961] [KO:K06266]
  パスウェイ
hsa04514  細胞接着分子 (CAM) の相互作用
hsa04530  密着結合
hsa04670  白血球の内皮細胞間隙遊走
階層分類  
ターゲットに基づく医薬品分類 [BR:jp08310]
 細胞表面分子とリガンド
  その他の細胞表面分子
   CD 分子
    CD47
     D13158  スペバタミグ
   その他
    CLDN18
     D13158  スペバタミグ
リンク   
CAS: 2928515-36-8
PubChem: 518520878
LinkDB    

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