KEGG   DGROUP: Lapatinib
Entry
DG00715                     DGroup                                 
Name
Lapatinib
Type
Chemical
Member
D08108  
Lapatinib (INN)
D04024  
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN)  <JP/US>
Class
Antineoplastic
 DG01918  Tyrosine kinase inhibitor
  DG01917  Receptor tyrosine kinase inhibitor
   DG03158  HER2 inhibitor
Metabolizing enzyme substrate
 DG02918  CYP2C8 substrate
 DG01639  CYP2C19 substrate
 DG01633  CYP3A/CYP3A4 substrate
  DG02913  CYP3A4 substrate
 DG02925  CYP3A5 substrate
Transporter substrate
 DG01665  ABCB1 substrate
 DG01913  ABCG2 substrate
Remark
ATC code: L01EH01
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