DGROUP: Lapatinib
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Entry
DG00715 DGroup
Name
Lapatinib
Type
Chemical
Member
D08108
Lapatinib (INN)
D04024
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN) <JP/US>
Class
Antineoplastic
DG01918
Tyrosine kinase inhibitor
DG01917
Receptor tyrosine kinase inhibitor
DG03158
HER2 inhibitor
Metabolizing enzyme substrate
DG02918
CYP2C8 substrate
DG01639
CYP2C19 substrate
DG01633
CYP3A/CYP3A4 substrate
DG02913
CYP3A4 substrate
DG02925
CYP3A5 substrate
Transporter substrate
DG01665
ABCB1 substrate
DG01913
ABCG2 substrate
Remark
ATC code:
L01EH01
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