KEGG   DGROUP: Tyrosine kinase inhibitor
Entry
DG01918                     DGroup                                 
Name
Tyrosine kinase inhibitor
Type
Target
Member
BCR-ABL inhibitor
 DG00710  
Imatinib
  D08066  
Imatinib (INN)
  D01441  
Imatinib mesylate (USAN); Imatinib mesilate (JAN)  <JP/US>
 DG00714  
Dasatinib
  D03658  
Dasatinib (JAN/INN)  <JP>
  D06414  
Dasatinib (USAN); Dasatinib hydrate (JAN)  <JP/US>
 DG00716  
Nilotinib
  D08953  
Nilotinib (USAN/INN)
  D06413  
Nilotinib hydrochloride hydrate (JAN)  <JP/US>
  D12444  
Nilotinib hydrochloride dihydrate (JAN)
 DG00718  
Bosutinib
  D03252  
Bosutinib (USAN)
  D09728  
Bosutinib hydrate (JAN)  <JP/US>
 DG00722  
Ponatinib
  D09950  
Ponatinib (USAN/INN)
  D09951  
Ponatinib hydrochloride (JAN/USAN)  <JP/US>
 DG03004  
Asciminib
  D11403  
Asciminib (USAN/INN)
  D11404  
Asciminib hydrochloride (JAN/USAN)  <JP/US>
Receptor tyrosine kinase inhibitor
 DG03162  
EGFR inhibitor
  D01977  
Gefitinib (JP18/USAN/INN)  <JP/US>
  DG00711  
Erlotinib
   D07907  
Erlotinib (INN)
   D04023  
Erlotinib hydrochloride (JAN/USAN)  <JP/US>
  DG00717  
Afatinib
   D09724  
Afatinib (USAN/INN)
   D09733  
Afatinib dimaleate (USAN); Afatinib maleate (JAN)  <JP/US>
  D10766  
Osimertinib mesylate (USAN); Osimertinib mesilate (JAN)  <JP/US>
  D10858  
Rociletinib (USAN/INN)
  DG02916  
Olmutinib
   D10859  
Olmutinib (USAN/INN)
   D11115  
Olmutinib hydrochloride (USAN)
  DG01793  
Dacomitinib
   D09883  
Dacomitinib (INN)
   D10514  
Dacomitinib (USAN); Dacomitinib hydrate (JAN)  <JP/US>
  D11251  
Icotinib
  D03455  
Cetuximab (USAN/INN); Cetuximab (genetical recombination) (JAN)  <JP/US>
  D05350  
Panitumumab (USAN/INN); Panitumumab (genetical recombination) (JAN)  <JP/US>
  D10018  
Necitumumab (USAN/INN); Necitumumab (genetical recombination) (JAN)  <JP/US>
  D11894  
Amivantamab (USAN/INN); Amivantamab (genetical recombination) (JAN)  <US>
  DG03205  
Lazertinib
   D11980  
Lazertinib (USAN)
   D12245  
Lazertinib mesilate hydrate (JAN)
  DG03209  
Aumolertinib
   D12258  
Aumolertinib (USAN)
   D12259  
Aumolertinib mesylate (USAN)
  D12457  
Tuxobertinib (USAN/INN)
 DG03158  
HER2 inhibitor
  DG00715  
Lapatinib
   D08108  
Lapatinib (INN)
   D04024  
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN)  <JP/US>
  DG02303  
Neratinib
   D08950  
Neratinib (USAN/INN)
   D10898  
Neratinib maleate  <US>
  DG03240  
Tucatinib
   D11141  
Tucatinib (USAN/INN)  <US>
   D12442  
Tucatinib ethanolate (JAN)
  D03257  
Trastuzumab (USAN/INN); Trastuzumab (genetical recombination) (JAN); Trastuzumab (genetical recombination) [Trastuzumab biosimilar 1] (JAN); Trastuzumab (genetical recombination) [Trastuzumab biosimilar 2] (JAN); Trastuzumab (genetical recombination) [Trastuzumab biosimilar 3] (JAN)  <JP/US>
  D05446  
Pertuzumab (USAN/INN); Pertuzumab (genetical recombination) (JAN)  <JP/US>
  D09980  
Trastuzumab emtansine (USAN/INN); Trastuzumab emtansine (genetical recombination) (JAN)  <JP/US>
  D11529  
Trastuzumab deruxtecan (USAN/INN); Trastuzumab deruxtecan (genetical recombination) (JAN)  <JP/US>
  D11375  
Trastuzumab duocarmazine (USAN/INN)
  D10446  
Margetuximab (USAN)  <US>
  D11560  
Trastuzumab and hyaluronidase  <US>
 DG03203  
VEGFR inhibitor
  D03218  
Axitinib (JAN/USAN)  <JP/US>
  DG01360  
Cediranib
   D08881  
Cediranib (USAN/INN)
   D08883  
Cediranib maleate (JAN/USAN)
  DG01375  
Tivozanib
   D09683  
Tivozanib (USAN/INN)
   D10190  
Tivozanib hydrochloride (USAN)  <US>
 DG03208  
FGFR inhibitor
  D10927  
Erdafitinib (JAN/USAN/INN)  <US>
  D11417  
Pemigatinib (JAN/USAN/INN)  <JP/US>
  DG03062  
Infigratinib
   D11589  
Infigratinib (USAN/INN)
   D11611  
Infigratinib phosphate (USAN)  <US>
  D11725  
Futibatinib (JAN/USAN/INN)
 DG00712  
Sunitinib
  D08552  
Sunitinib (INN)
  D06402  
Sunitinib malate (JAN/USAN)  <JP/US>
 D05380  
Pazopanib hydrochloride (JAN/USAN)  <JP/US>
 D06407  
Vandetanib (JAN/USAN/INN)  <JP/US>
 DG00720  
Regorafenib
  D10138  
Regorafenib (USAN/INN)
  D10137  
Regorafenib hydrate (JAN)  <JP/US>
 D10229  
Masitinib (INN)
 DG01670  
Cabozantinib
  D10062  
Cabozantinib (USAN)
  D10095  
Cabozantinib s-malate (USAN); Cabozantinib malate (JAN)  <JP/US>
 DG01362  
Lenvatinib
  D09919  
Lenvatinib (USAN/INN)
  D09920  
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN)  <JP/US>
 D05029  
Midostaurin (JAN/USAN/INN)  <US>
 DG01364  
Quizartinib
  D09955  
Quizartinib (USAN/INN)
  D09956  
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN)  <JP>
 DG02923  
Larotrectinib
  D11137  
Larotrectinib (USAN/INN)
  D11138  
Larotrectinib sulfate (JAN/USAN)  <JP/US>
 DG01948  
Gilteritinib
  D10709  
Gilteritinib (USAN/INN)
  D10800  
Gilteritinib fumarate (JAN/USAN)  <JP/US>
 DG02081  
Capmatinib
  D10696  
Capmatinib (USAN/INN)
  D10891  
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN)  <JP/US>
 D11279  
Avapritinib (USAN/INN)  <US>
 D11353  
Ripretinib (USAN)  <US>
 DG03087  
Tepotinib
  D11717  
Tepotinib (USAN/INN)
  D11073  
Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN)  <JP/US>
 DG01262  
Motesanib
  D06678  
Motesanib (USAN)
  D08947  
Motesanib diphosphate (USAN); Motesanib phosphate (JAN)
 DG01357  
Varlitinib
  D09689  
Varlitinib (USAN/INN)
  D09690  
Varlitinib tosylate (USAN)
 DG01361  
Crenolanib
  D10102  
Crenolanib (USAN)
  D10103  
Crenolanib besylate (USAN)
 DG01363  
Toceranib
  D08503  
Toceranib (USAN)
  D08544  
Toceranib phosphate (USAN)
 DG01367  
Golvatinib
  D10224  
Golvatinib (USAN)
  D10465  
Golvatinib tartrate (USAN)
 DG01373  
Brivanib
  D09589  
Brivanib (USAN)
  D08878  
Brivanib alaninate (JAN/USAN/INN)
 DG02966  
Rivoceranib
  D11288  
Rivoceranib (USAN/INN)
  D11289  
Rivoceranib mesylate (USAN)
 DG03015  
Nazartinib
  D11430  
Nazartinib (USAN/INN)
  D11434  
Nazartinib mesylate (USAN)
 DG03045  
Sitravatinib
  D11140  
Sitravatinib (USAN/INN)
  D11541  
Sitravatinib malate (USAN)
 DG03093  
Dubermatinib
  D11732  
Dubermatinib (USAN/INN)
  D11733  
Dubermatinib tartrate (USAN)
 DG03101  
Tesevatinib
  D11772  
Tesevatinib (USAN/INN)
  D11773  
Tesevatinib tosylate (USAN)
 DG03112  
Naquotinib
  D10958  
Naquotinib (USAN/INN)
  D10886  
Naquotinib mesylate (USAN); Naquotinib mesilate (JAN)
 DG03148  
Mobocertinib
  D12001  
Mobocertinib (USAN/INN)
  D11969  
Mobocertinib succinate (JAN)  <US>
 DG03234  
Tasurgratinib
  D12404  
Tasurgratinib (INN)
  D12405  
Tasurgratinib succinate (JAN)
 D03350  
Canertinib dihydrochloride (USAN)
 D04025  
Mubritinib (USAN/INN)
 D04696  
Lestaurtinib (USAN/INN)
 D05399  
Pelitinib (USAN/INN)
 D05819  
Semaxanib (USAN/INN)
 D06005  
Tandutinib (USAN/INN)
 D06285  
Vatalanib (USAN/INN)
 D08907  
Dovitinib lactate (USAN); Dovitinib lactate hydrate (JAN)
 D09618  
Foretinib (USAN/INN)
 D09635  
Linifanib (USAN/INN)
 D09945  
Pegdinetanib (USAN/INN)
 D10173  
Tivantinib (JAN/USAN/INN)
 D10862  
Altiratinib (USAN)
 D11136  
Glesatinib (USAN/INN)
 D11139  
Savolitinib (USAN/INN)
 D11368  
Mavelertinib (USAN/INN)
 D11438  
Bemcentinib (USAN/INN)
 D11461  
Derazantinib hydrochloride (USAN)
 D11737  
Fisogatinib (USAN/INN)
 D12432  
Zurletrectinib (USAN)
ALK inhibitor
 D09731  
Crizotinib (JAN/USAN/INN)  <JP/US>
 D10551  
Ceritinib (JAN/USAN/INN)  <JP/US>
 DG01625  
Alectinib
  D10542  
Alectinib (USAN/INN)
  D10450  
Alectinib hydrochloride (JAN)  <JP/US>
 D10866  
Brigatinib (JAN/USAN)  <JP/US>
 D11012  
Lorlatinib (JAN/USAN/INN)  <JP/US>
 DG02996  
Ensartinib
  D11346  
Ensartinib (USAN)
  D11356  
Ensartinib hydrochloride (USAN)
BTK inhibitor
 D10223  
Ibrutinib (JAN/USAN)  <JP/US>
 DG03089  
Acalabrutinib
  D10893  
Acalabrutinib (JAN/USAN/INN)  <JP/US>
  D11720  
Acalabrutinib maleate (USAN)
 D11422  
Zanubrutinib (JAN/USAN/INN)  <US>
 D11070  
Tirabrutinib hydrochloride (JAN)  <JP>
 DG01863  
Spebrutinib
  D10730  
Spebrutinib (USAN/INN)
  D10731  
Spebrutinib besylate (USAN)
 DG03023  
Vecabrutinib
  D11428  
Vecabrutinib (USAN/INN)
  D11502  
Vecabrutinib succinate (USAN)
 D11478  
Branebrutinib (USAN)
 D12160  
Orelabrutinib (USAN/INN)
 D11457  
Fenebrutinib (USAN/INN)
 D11873  
Rilzabrutinib (USAN/INN)
 D12158  
Elsubrutinib (USAN/INN)
 D12213  
Tolebrutinib (USAN/INN)
 D12285  
Remibrutinib (USAN/INN)
 D12383  
Edralbrutinib (USAN/INN)
 D12467  
Evobrutinib (USAN/INN)
D11768  
Pacritinib (USAN/INN)  <US>
Sorafenib
 D08524  
Sorafenib (USAN/INN)
 D06272  
Sorafenib tosylate (USAN); Sorafenib tosilate (JAN)  <JP/US>
Nintedanib
 D10481  
Nintedanib (USAN/INN)
 D10396  
Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN)  <JP/US>
D10926  
Entrectinib (JAN/USAN/INN)  <JP/US>
D11713  
Selpercatinib (JAN/USAN/INN)  <JP/US>
Pralsetinib
 D11712  
Pralsetinib (USAN/INN)  <US>
 D12354  
Pralsetinib hydrate (JAN)
Tozasertib
 D08279  
Tozasertib (USAN)
 D08344  
Tozasertib lactate (USAN)
Rebastinib
 D10334  
Rebastinib (USAN)
 D10399  
Rebastinib Tosylate (USAN)
Saracatinib
 D09664  
Saracatinib (USAN/INN)
 D09665  
Saracatinib difumarate (USAN)
Defactinib
 D10618  
Defactinib (USAN/INN)
 D10619  
Defactinib hydrochloride (USAN)
Amuvatinib
 D09864  
Amuvatinib (USAN/INN)
 D09865  
Amuvatinib hydrochloride (USAN)
Gusacitinib
 D11676  
Gusacitinib (USAN/INN)
 D11677  
Gusacitinib hydrochloride (USAN)
Zeteletinib
 D12330  
Zeteletinib (USAN)
 D12331  
Zeteletinib adipate (USAN)
Taletrectinib
 D12363  
Taletrectinib (USAN/INN)
 D12364  
Taletrectinib adipate (USAN)
D10202  
Bafetinib (USAN)
D11209  
Entospletinib (USAN/INN)
D11454  
Repotrectinib (USAN)
D11786  
Vodobatinib (USAN)
D12476  
Tuspetinib (USAN)
 » expand
Class
Antineoplastic
LinkDB

» Japanese version

DBGET integrated database retrieval system