KEGG   DGROUP: CYP3A/CYP3A4 substrate
Entry
DG01633                     DGroup                                 
Name
CYP3A/CYP3A4 substrate
Type
Metabolism
Member
CYP3A4 substrate
 DG00011  
Dexamethasone
  D00292  
Dexamethasone (JP18/USP/INN)  <JP/US>
  D00975  
Dexamethasone sodium phosphate (JAN/USP)  <JP/US>
  D01510  
Dexamethasone metasulfobenzoate sodium (JAN)  <JP>
  D01615  
Dexamethasone palmitate (JAN)  <JP>
  D01632  
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN)  <JP>
  D01948  
Dexamethasone valerate (JAN)  <JP>
  D02174  
Dexamethasone acetate (JAN/USP)
  D02591  
Dexamethasone acefurate (USAN/INN)
  D02592  
Dexamethasone beloxil (USAN)
  D07073  
Dexamethasone cipecilate (JAN/INN)  <JP>
  D07796  
Dexamethasone 21-acetate
  D07797  
Dexamethasone isonicotinate
  D07798  
Dexamethasone sodium hemisulfate
  D07799  
Dexamethasone 21-tebutate
  D07800  
Dexamethasone 21-valerate
  D07801  
Dexamethasone phenylpropionate
  D07802  
Dexamethasone phosphate
 D01131  
Lafutidine (JP18/INN)  <JP>
 DG00020  
Omeprazole
  D00455  
Omeprazole (JP18/USP/INN)  <JP/US>
  D01207  
Omeprazole sodium (USAN)
  D05261  
Omeprazole sodium injection (JAN)  <JP>
  D05259  
Omeprazole magnesium (USP)  <US>
 DG00021  
Pantoprazole
  D05353  
Pantoprazole (USAN/INN)
  D02593  
Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN)  <US>
 D00355  
Lansoprazole (JP18/USP/INN)  <JP/US>
 DG00022  
Rabeprazole
  D08463  
Rabeprazole (INN)
  D00724  
Rabeprazole sodium (JP18/USP)  <JP/US>
 DG00023  
Esomeprazole
  D07917  
Esomeprazole (INN)
  D01984  
Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN)  <JP/US>
  D04056  
Esomeprazole sodium (USAN)  <US>
  D09339  
Esomeprazole potassium (USAN)
  D10120  
Esomeprazole strontium (USAN)  <US>
  D11114  
Esomeprazole magnesium dihydrate  <US>
 DG03298  
Dexlansoprazole
  D08903  
Dexlansoprazole (INN/USAN)  <US>
  D12816  
Dexlansoprazole sesquihydrate  <US>
 DG03104  
Vonoprazan
  D11784  
Vonoprazan (USAN/INN)
  D10466  
Vonoprazan fumarate (JAN/USAN)  <JP/US>
 D09742  
Lansoprazole, amoxicillin hydrate and metronidazole
 D10246  
Omeprazole, clarithromycin and amoxicillin
 D08774  
Amoxicillin hydrate, clarithromycin and lansoprazole  <US>
 D10519  
Rabeprazole, amoxicillin and clarithromycin  <JP>
 D10520  
Rabeprazole, amoxicillin and metronidazole  <JP>
 D10775  
Vonoprazan, amoxicillin and clarithromycin  <JP>
 D10774  
Vonoprazan, amoxicillin and metronidazole  <JP>
 D01121  
Rebamipide (JP18/INN)  <JP>
 DG00046  
Alosetron
  D07129  
Alosetron (INN)
  D02829  
Alosetron hydrochloride (USAN)  <US>
 DG00057  
Domperidone
  D01745  
Domperidone (JP18/USAN/INN)  <JP>
  D07868  
Domperidone maleate
 DG01285  
Mosapride
  D01994  
Mosapride citrate hydrate (JP18)  <JP>
  D08236  
Mosapride (INN)
 DG00060  
Ondansetron
  D00456  
Ondansetron (JAN/USP/INN)  <US>
  D00678  
Ondansetron hydrochloride hydrate (JAN/USP)  <JP/US>
 DG00061  
Granisetron
  D04370  
Granisetron (JAN/USAN/INN)  <US>
  D00677  
Granisetron hydrochloride (JAN/USP)  <JP/US>
 DG00064  
Palonosetron
  D07175  
Palonosetron (INN)
  D05343  
Palonosetron hydrochloride (JAN/USP)  <JP/US>
 D10572  
Fosnetupitant and palonosetron hydrochloride
 DG00066  
Aprepitant
  D02968  
Aprepitant (JAN/USP/INN)  <JP/US>
  D10895  
Fosaprepitant (INN)
  D06597  
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN)  <JP/US>
 DG01868  
Rolapitant
  D10742  
Rolapitant (USAN/INN)
  D08988  
Rolapitant hydrochloride (USAN)  <US>
 DG01342  
Naldemedine
  D10188  
Naldemedine (USAN/INN)
  D10478  
Naldemedine tosylate (JAN/USAN)  <JP/US>
 DG03072  
Tenapanor
  D11652  
Tenapanor (USAN/INN)
  D11653  
Tenapanor hydrochloride (JAN/USAN)  <JP/US>
 D02554  
Rifaximin (JAN/USAN/INN)  <JP/US>
 DG00092  
Loperamide
  D08144  
Loperamide (INN)
  D00729  
Loperamide hydrochloride (JAN/USP)  <JP/US>
  D07113  
Loperamide oxide (INN)
 D00246  
Budesonide (JP18/USP/INN)  <JP/US>
 D00689  
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18)  <JP/US>
 D11572  
Beclomethasone dipropionate monohydrate
 DG00103  
Fenfluramine
  D07945  
Fenfluramine (INN)
  D04148  
Fenfluramine hydrochloride (JAN/USAN)  <JP/US>
 D11710  
Phentermine and topiramate  <US>
 D00336  
Glyburide (USP); Glibenclamide (JP18/INN)  <JP/US>
 D10263  
Metformin hydrochloride and saxagliptin hydrochloride  <US>
 DG00119  
Saxagliptin
  D08996  
Saxagliptin (USAN/INN)
  D09753  
Saxagliptin hydrate (JAN)  <JP/US>
  D10262  
Saxagliptin hydrochloride  <US>
 DG01283  
Teneligliptin
  D08616  
Teneligliptin (INN)
  D09756  
Teneligliptin hydrobromide hydrate (JAN)  <JP>
  D11968  
Teneligliptin hydrobromide (JAN)
 D10669  
Sotagliflozin (USAN/INN)  <US>
 D00594  
Repaglinide (JAN/USP/INN)  <JP/US>
 DG00148  
Eliglustat
  D09893  
Eliglustat (USAN/INN)
  D09894  
Eliglustat tartrate (JAN/USAN)  <JP/US>
 DG00155  
Clopidogrel
  D07729  
Clopidogrel (USP/INN)
  D00769  
Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18)  <JP/US>
  D10823  
Clopidogrel hydrochloride
  D10824  
Clopidogrel besilate
 D01896  
Cilostazol (JP18/USP/INN)  <JP/US>
 DG01349  
Vorapaxar
  D09765  
Vorapaxar (USAN/INN)
  D09766  
Vorapaxar sulfate (JAN/USAN)
 D09994  
Selexipag (JAN/USAN/INN)  <JP/US>
 D10513  
Clopidogrel sulfate and aspirin  <JP>
 D10527  
Acetylsalicylic acid and lansoprazole  <JP>
 DG00163  
Argatroban
  C04931  
Argatroban
  D00181  
Argatroban (USP); Argatroban hydrate (JP18)  <JP/US>
 D07086  
Rivaroxaban (JAN/USAN/INN)  <JP/US>
 D03213  
Apixaban (JAN/USAN/INN)  <JP/US>
 DG01976  
Avatrombopag
  D10306  
Avatrombopag (USAN/INN)
  D10307  
Avatrombopag maleate (JAN/USAN)  <JP/US>
 DG01419  
Fostamatinib
  D09347  
Fostamatinib (USAN)
  D09348  
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN)  <JP/US>
 D12396  
Sebetralstat (JAN/USAN/INN)  <JP/US>
 D11330  
Voxelotor (USAN)  <US>
 DG00192  
Quinidine
  D08458  
Quinidine (BAN)
  D00642  
Quinidine gluconate (USP)  <US>
  D00643  
Quinidine polygalacturonate
  D02272  
Quinidine sulfate (USP); Quinidine sulfate hydrate (JP18)  <JP/US>
  D08459  
Quinidine phenylethylbarbiturate
 DG00194  
Disopyramide
  D00303  
Disopyramide (JP18/USAN/INN)  <JP>
  D00637  
Disopyramide phosphate (JAN/USP)  <JP/US>
 DG00196  
Lidocaine
  D00358  
Lidocaine (JP18/USP/INN)  <JP/US>
  D02086  
Lidocaine hydrochloride (JAN/USP)  <JP/US>
  D08127  
Lidocaine hydrochloride monohydrate  <JP/US>
 DG00200  
Propafenone
  D08435  
Propafenone (INN)
  D00640  
Propafenone hydrochloride (JP18/USP)  <JP/US>
 DG00204  
Amiodarone
  D02910  
Amiodarone (USAN/INN)
  D00636  
Amiodarone hydrochloride (JP18/USP)  <JP/US>
 DG00209  
Cibenzoline
  D03492  
Cifenline (USAN); Cibenzoline (INN)
  D01455  
Cifenline succinate (USAN); Cibenzoline succinate (JP18)  <JP>
 DG00246  
Ivabradine
  D07165  
Ivabradine (USAN/INN)
  D08095  
Ivabradine hydrochloride (JAN/USAN)  <JP/US>
 D12265  
Mavacamten (JAN/USAN/INN)  <JP/US>
 DG00250  
Guanfacine
  D08031  
Guanfacine (INN)
  D00606  
Guanfacine hydrochloride (JAN/USP)  <JP/US>
 DG00266  
Bosentan
  D07538  
Bosentan (INN)
  D01227  
Bosentan (USAN); Bosentan hydrate (JAN)  <JP/US>
 D10135  
Macitentan (JAN/USAN)  <JP/US>
 D01115  
Eplerenone (JP18/USAN/INN)  <JP/US>
 D10633  
Finerenone (JAN/USAN/INN)  <JP/US>
 D01213  
Tolvaptan (JP18/USAN/INN)  <JP/US>
 DG00331  
Diltiazem
  D07845  
Diltiazem (INN)
  D00616  
Diltiazem hydrochloride (JP18/USP)  <JP/US>
  D03830  
Diltiazem malate (USAN)
 DG00321  
Carvedilol
  D00255  
Carvedilol (JP18/USP/INN)  <JP/US>
  D03415  
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN)  <US>
 DG00322  
Amlodipine
  D07450  
Amlodipine (USP/INN)
  D00615  
Amlodipine besylate (USP); Amlodipine besilate (JP18)  <JP/US>
  D02914  
Amlodipine maleate (USAN)
  D11881  
Amlodipine benzoate  <US>
 D00319  
Felodipine (JP18/USP/INN)  <JP/US>
 DG00323  
Nicardipine
  D08270  
Nicardipine (INN)
  D00617  
Nicardipine hydrochloride (JP18/USAN)  <JP/US>
 D00437  
Nifedipine (JP18/USP/INN)  <JP/US>
 D00438  
Nimodipine (USP/INN)  <US>
 D00618  
Nisoldipine (JAN/USAN/INN)  <US>
 D00629  
Nitrendipine (JP18/USAN/INN)  <JP>
 D01908  
Nilvadipine (JP18/USAN/INN)  <JP>
 DG00324  
Manidipine
  D08155  
Manidipine (INN)
  D01553  
Manidipine hydrochloride (JP18)  <JP>
 DG00325  
Barnidipine
  D07494  
Barnidipine (INN)
  D01104  
Barnidipine hydrochloride (JAN)  <JP>
 D01173  
Cilnidipine (JP18/INN)  <JP>
 DG00327  
Benidipine
  D07509  
Benidipine (INN)
  D02045  
Benidipine hydrochloride (JP18)  <JP>
 DG00329  
Verapamil
  D02356  
Verapamil (USAN/INN)
  D00619  
Verapamil hydrochloride (JP18/USP)  <JP/US>
 D10932  
Etripamil (USAN/INN)  <US>
 DG00333  
Bepridil
  D07520  
Bepridil (INN)
  D00631  
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN)  <JP>
 D09745  
Valsartan and amlodipine besilate  <JP/US>
 D09743  
Telmisartan and amlodipine besilate (JP18)  <JP/US>
 D10243  
Irbesartan and amlodipine besilate (JP18)  <JP>
 D07569  
Candesartan cilexetil and anmlodipine besylate (JP18)  <JP>
 D10805  
Telmisartan, amlodipine and hydrochlorothiazide  <JP>
 DG00352  
Aliskiren
  D03208  
Aliskiren (USAN/INN)
  D06412  
Aliskiren fumarate (JAN/USAN)  <JP/US>
 D00434  
Simvastatin (JP18/USP/INN)  <JP/US>
 D00359  
Lovastatin (USP/INN)  <US>
 DG00354  
Fluvastatin
  D07983  
Fluvastatin (INN)
  D00892  
Fluvastatin sodium (JAN/USP)  <JP/US>
 DG00355  
Atorvastatin
  D07474  
Atorvastatin (INN)  <US>
  D00887  
Atorvastatin calcium anhydorous
  D02258  
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18)  <JP/US>
  D11095  
Atorvastatin calcium propylene glycol solvate  <US>
 DG00356  
Cerivastatin
  D07661  
Cerivastatin (INN)
  D00889  
Cerivastatin sodium (JAN/USAN)
 DG00362  
Lomitapide
  D09637  
Lomitapide (USAN/INN)
  D09638  
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN)  <JP/US>
 D10385  
Ezetimibe and atorvastatin  <JP>
 D08488  
Amlodipine besilate and atorvastatin calcium  <JP/US>
 D00351  
Ketoconazole (JP18/USP)  <JP/US>
 DG00375  
Terbinafine
  D02375  
Terbinafine (USAN/INN)
  D02219  
Terbinafine hydrochloride (JP18/USP)  <JP/US>
 D05744  
Roflumilast (JAN/USAN/INN)  <US>
 D09544  
Ozenoxacin (JAN/USAN/INN)  <JP>
 DG00410  
Methylprednisolone
  D00407  
Methylprednisolone (JP18/USP/INN)  <JP/US>
  D00751  
Methylprednisolone sodium succinate (JAN/USP)  <JP/US>
  D00979  
Methylprednisolone acetate (JAN/USP)  <JP/US>
  D05000  
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18)
  D05001  
Methylprednisolone sodium phosphate (USAN)
  D05002  
Methylprednisolone suleptanate (USAN/INN)
  D07203  
Methylprednisolone aceponate (INN)
 DG00419  
Mometasone
  D08227  
Mometasone (INN)
  D00690  
Mometasone furoate (JAN/USP)  <JP/US>
  D03325  
Mometasone furoate hydrate (JAN)  <JP/US>
 DG00420  
Fluticasone
  D07981  
Fluticasone (INN)
  D01708  
Fluticasone propionate (JAN/USP)  <JP/US>
  D06315  
Fluticasone furoate (JAN/USAN/INN)  <JP/US>
 D00592  
Dapsone (USP); Diaphenylsulfone (JAN)  <JP/US>
 D10989  
Sofpironium bromide (JAN/USAN/INN)  <JP/US>
 DG00439  
Tacrolimus
  D08556  
Tacrolimus (INN)
  D00107  
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18)  <JP/US>
 DG00719  
Ruxolitinib
  D09959  
Ruxolitinib (USAN/INN)
  D09960  
Ruxolitinib phosphate (JAN/USAN)  <JP/US>
 D11046  
Delgocitinib (JAN/USAN/INN)  <JP/US>
 D00321  
Finasteride (JAN/USP/INN)  <JP/US>
 D00804  
Ivermectin (JAN/USP/INN)  <JP/US>
 DG00974  
Caffeine
  D00528  
Caffeine (USP); Anhydrous caffeine (JP18)  <JP>
  D01453  
Caffeine hydrate (JP18)  <JP>
  D07603  
Caffeine citrate (USP)  <US>
 DG00445  
Methylergometrine
  D08207  
Methylergometrine (INN)
  D00680  
Methylergonovine maleate (USP); Methylergometrine maleate (JP18)  <JP/US>
 DG00446  
Ergometrine
  D07905  
Ergometrine (INN)
  D01163  
Ergonovine maleate (USP); Ergometrine maleate (JP18)
 DG00452  
Bromocriptine
  D03165  
Bromocriptine (USAN/INN)
  D00780  
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18)  <JP/US>
 D00987  
Cabergoline (JP18/USP/INN)  <JP/US>
 D02577  
Flibanserin (USAN/INN)  <US>
 D12123  
Elinzanetant (USAN/INN)  <US>
 D04483  
Ethinylestradiol and norethisterone  <JP/US>
 D04463  
Norgestrel and ethinylestradiol tablets (JP18)  <JP/US>
 D04482  
Ethinylestradiol and levonorgestrel  <JP/US>
 D04484  
Desogestrel and ethinylestradiol  <JP/US>
 D09741  
Drospirenone and ethinylestradiol  <JP/US>
 D03917  
Drospirenone (JAN/USP/INN)  <JP/US>
 DG00461  
Ethinylestradiol
  D00554  
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN)  <JP>
  D07928  
Ethinylestradiol propanesulfonate
 DG00462  
Estradiol
  D00105  
Estradiol (JAN/USP/INN)  <JP/US>
  D01413  
Estradiol valerate (JAN/USP/INN)  <JP/US>
  D01617  
Estradiol dipropionate (JAN)
  D01953  
Estradiol benzoate (JP18/USP)
  D04061  
Estradiol acetate (USAN)  <US>
  D04063  
Estradiol cypionate (USP)  <US>
  D04064  
Estradiol enanthate (USAN)
  D04065  
Estradiol undecylate (USAN/INN)
  D07918  
Estradiol hemihydrate  <US>
  D07919  
Estradiol 17 beta-hemisuccinate
 DG00464  
Estrone
  D00067  
Estrone (JAN/USP/INN)
  D00312  
Estrone sodium sulfate
  D00948  
Estropipate (USP)
 DG00465  
Conjugated estrogen
  D04070  
Estrogens, conjugated (JAN/USP)  <JP/US>
  D05987  
Synthetic conjugated estrogens, B (USAN)
 D00066  
Progesterone (JP18/USP/INN)  <JP/US>
 D01217  
Dydrogesterone (JP18/USP/INN)  <JP>
 D03799  
Dienogest (JAN/USAN/INN)  <JP>
 D09188  
Estradiol and norethindrone  <JP/US>
 D09187  
Estradiol and levonorgestrel  <JP/US>
 D00585  
Mifepristone (JAN/USAN/INN)  <US>
 DG00478  
Oxybutynin
  D00465  
Oxybutynin (USAN/INN)  <US>
  D00722  
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18)  <JP/US>
 DG00479  
Propiverine
  D08441  
Propiverine (INN)
  D01007  
Propiverine hydrochloride (JP18)  <JP>
 DG00480  
Tolterodine
  D00646  
Tolterodine (USAN/INN)
  D01148  
Tolterodine tartrate (JAN/USP)  <US>
 DG00481  
Solifenacin
  D08522  
Solifenacin (INN)
  D01269  
Solifenacin succinate (JAN/USAN/INN)  <JP/US>
 DG00482  
Darifenacin
  D03654  
Darifenacin (USAN/INN)
  D01699  
Darifenacin hydrobromide (JAN/USAN)  <US>
 DG00483  
Fesoterodine
  D07226  
Fesoterodine (INN)
  D08923  
Fesoterodine fumarate (JAN/USAN)  <JP/US>
 D09535  
Mirabegron (JAN/USAN/INN)  <JP/US>
 D06273  
Imidafenacin (JAN/INN)  <JP>
 D10433  
Vibegron (JAN/USAN/INN)  <JP/US>
 DG00484  
Sildenafil
  D08514  
Sildenafil (INN)
  D02229  
Sildenafil citrate (JAN/USP)  <JP/US>
 D02008  
Tadalafil (JAN/USP/INN)  <JP/US>
 DG00487  
Vardenafil
  D08668  
Vardenafil (USAN/INN)
  D02731  
Vardenafil dihydrochoride (USAN)
  D03260  
Vardenafil hydrochloride hydrate (JAN)  <JP/US>
  D09989  
Vardenafil hydrochloride (USP)
 D03217  
Avanafil (USAN/INN)  <US>
 DG00489  
Alfuzosin
  D07124  
Alfuzosin (INN)
  D01692  
Alfuzosin hydrochloride (JAN/USAN)  <US>
 D01965  
Silodosin (JP18/INN)  <JP/US>
 D11389  
Dutasteride and tamsulosin  <US>
 D03820  
Dutasteride (JAN/USP/INN)  <JP/US>
 D12486  
Finasteride and tadalafil
 D03671  
Deflazacort (USAN/INN)  <US>
 D11000  
Vamorolone (USAN/INN)  <US>
 DG02839  
Osilodrostat
  D11061  
Osilodrostat (USAN/INN)
  D11062  
Osilodrostat phosphate (JAN/USAN)  <JP/US>
 DG00513  
Cinacalcet
  D03504  
Cinacalcet (USAN)
  D03505  
Cinacalcet hydrochloride (JAN/USAN)  <JP/US>
 D01322  
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN)
 DG00605  
Clarithromycin
  D00276  
Clarithromycin (JP18/USP/INN)  <JP/US>
  D07710  
Clarithromycin lactobionate
 DG00616  
Ofloxacin
  D00453  
Ofloxacin (JP18/USP/INN)  <JP/US>
  D08291  
Ofloxacin hydrochloride
 DG03066  
Lefamulin
  D11631  
Lefamulin (USAN/INN)
  D11632  
Lefamulin acetate (USAN)
 DG01998  
Gepotidacin
  D10878  
Gepotidacin (USAN/INN)
  D10879  
Gepotidacin mesylate (USAN); Gepotidacin mesilate hydrate (JAN)  <US>
 D00350  
Itraconazole (JP18/USP)  <JP/US>
 D00424  
Rifabutin (JAN/USP/INN)  <JP/US>
 DG00644  
Bedaquiline
  D09872  
Bedaquiline (USAN/INN)
  D09873  
Bedaquiline fumarate (JAN/USAN)  <JP/US>
 D09785  
Delamanid (JAN/USAN)  <JP>
 DG00653  
Saquinavir
  D00429  
Saquinavir (JAN/USP/INN)
  D01160  
Saquinavir mesylate (USP); Saquinavir mesilate (JAN)
 DG00654  
Indinavir
  C07051  
Indinavir
  D03833  
Indinavir (USAN)
  D00897  
Indinavir sulfate (USP)
  D02861  
Indinavir sulfate ethanolate (JAN)
 DG00655  
Nelfinavir
  D08259  
Nelfinavir (INN)
  D00899  
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN)  <US>
 D00894  
Amprenavir (JAN/USAN/INN)
 DG00656  
Fosamprenavir
  D02497  
Fosamprenavir (INN)
  D02867  
Fosamprenavir calcium hydrate (JAN)
  D03835  
Fosamprenavir calcium (USAN)  <US>
  D03837  
Fosamprenavir sodium (USAN)
 DG00659  
Darunavir
  D03656  
Darunavir (USAN/INN)  <US>
  D06478  
Darunavir ethanolate (JAN)  <JP/US>
  D12637  
Darunavir hydrate  <US>
  D12752  
Darunavir propylene glycolate  <US>
 D12269  
Nirmatrelvir and ritonavir  <JP/US>
 D00435  
Nevirapine (JAN/USP/INN)  <JP/US>
 D00896  
Efavirenz (JAN/USP/INN)  <US>
 D04112  
Etravirine (JAN/USAN/INN)  <US>
 DG00667  
Dolutegravir
  D10066  
Dolutegravir (USAN)
  D10113  
Dolutegravir sodium (JAN/USAN)  <JP/US>
 D09012  
Telaprevir (JAN/USAN/INN)
 DG01669  
Daclatasvir
  D10065  
Daclatasvir (USAN)
  D10105  
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN)
 D10745  
Ombitasvir, paritaprevir and ritonavir
 D10827  
Sofosbuvir and velpatasvir  <JP/US>
 D10600  
Dolutegravir, abacavir and lamivudine  <JP/US>
 D10753  
Atazanavir and cobicistat  <US>
 D06670  
Maraviroc (JAN/INN)  <JP/US>
 D04859  
Maribavir (JAN/USAN/INN)  <JP/US>
 DG00675  
Cyclophosphamide
  D07760  
Cyclophosphamide (INN)
  D00287  
Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18)  <JP/US>
 D00343  
Ifosfamide (JAN/USP/INN)  <JP/US>
 DG00689  
Vinblastine
  D08675  
Vinblastine (INN)
  D01068  
Vinblastine sulfate (JP18/USP)  <JP/US>
 DG00692  
Vinorelbine
  D08680  
Vinorelbine (INN)
  D01935  
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN)  <JP/US>
 DG00694  
Docetaxel
  D07866  
Docetaxel (JAN/INN)  <JP/US>
  D02165  
Docetaxel (USP); Docetaxel hydrate (JP18)  <JP/US>
 DG00726  
Irinotecan
  D08086  
Irinotecan (INN)
  D01061  
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18)  <JP/US>
  D10642  
Irinotecan sucrosofate (USAN)
 D06199  
Trabectedin (JAN/USAN/INN)  <JP/US>
 D04645  
Ixabepilone (JAN/USAN/INN)  <US>
 DG00710  
Imatinib
  D08066  
Imatinib (INN)
  D01441  
Imatinib mesylate (USAN); Imatinib mesilate (JAN)  <JP/US>
 DG00714  
Dasatinib
  D03658  
Dasatinib (JAN/INN)  <JP>
  D06414  
Dasatinib (USAN); Dasatinib hydrate (JAN)  <JP/US>
  D12609  
Dasatinib laurylsulfate (USAN)
 DG00716  
Nilotinib
  D08953  
Nilotinib (USAN/INN)  <US>
  D06413  
Nilotinib hydrochloride hydrate (JAN)  <JP/US>
  D12444  
Nilotinib hydrochloride dihydrate (JAN)  <JP>
  D12854  
Nilotinib laurylsulfate (USAN)
  D13008  
Nilotinib D-tartrate (USAN)  <US>
 DG00718  
Bosutinib
  D03252  
Bosutinib (USAN)
  D09728  
Bosutinib hydrate (JAN)  <JP/US>
 DG03004  
Asciminib
  D11403  
Asciminib (USAN/INN)
  D11404  
Asciminib hydrochloride (JAN/USAN)  <JP/US>
 DG00711  
Erlotinib
  D07907  
Erlotinib (INN)
  D04023  
Erlotinib hydrochloride (JAN/USAN)  <JP/US>
 DG03205  
Lazertinib
  D11980  
Lazertinib (USAN/INN)
  D12245  
Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN)  <JP/US>
 DG00721  
Dabrafenib
  D10064  
Dabrafenib (USAN)
  D10104  
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN)  <JP/US>
 D11053  
Encorafenib (JAN/USAN/INN)  <JP/US>
 D09731  
Crizotinib (JAN/USAN/INN)  <JP/US>
 DG01625  
Alectinib
  D10542  
Alectinib (USAN/INN)
  D10450  
Alectinib hydrochloride (JAN)  <JP/US>
 D10866  
Brigatinib (JAN/USAN)  <JP/US>
 DG01414  
Selumetinib
  D09666  
Selumetinib (USAN/INN)
  D10024  
Selumetinib sulfate (JAN/USAN)  <JP/US>
 DG02084  
Ribociclib
  D10883  
Ribociclib (USAN/INN)
  D10979  
Ribociclib succinate (USAN)  <US>
 D06068  
Temsirolimus (JAN/USAN/INN)  <JP/US>
 D02714  
Everolimus (JAN/USAN/INN)  <JP/US>
 D00753  
Sirolimus (JAN/USAN/INN)  <JP/US>
 DG00715  
Lapatinib
  D08108  
Lapatinib (INN)
  D04024  
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN)  <JP/US>
 DG02303  
Neratinib
  D08950  
Neratinib (USAN/INN)
  D10898  
Neratinib maleate  <US>
 DG02968  
Fedratinib
  D10630  
Fedratinib (USAN/INN)
  D11296  
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN)  <JP/US>
 D11768  
Pacritinib (USAN/INN)  <US>
 DG01366  
Momelotinib
  D10315  
Momelotinib (USAN/INN)
  D10358  
Momelotinib dihydrochloride (USAN)
  D10889  
Momelotinib hydrochloride hydrate (JAN)  <JP/US>
 D03218  
Axitinib (JAN/USAN)  <JP/US>
 DG01375  
Tivozanib
  D09683  
Tivozanib (USAN/INN)
  D10190  
Tivozanib hydrochloride (USAN)  <US>
 D12050  
Pirtobrutinib (JAN/USAN)  <JP/US>
 D10927  
Erdafitinib (JAN/USAN/INN)  <JP/US>
 D11417  
Pemigatinib (JAN/USAN/INN)  <JP/US>
 DG00712  
Sunitinib
  D08552  
Sunitinib (INN)
  D06402  
Sunitinib malate (JAN/USAN)  <JP/US>
 D06407  
Vandetanib (JAN/USAN/INN)  <JP/US>
 DG00720  
Regorafenib
  D10138  
Regorafenib (USAN/INN)
  D10137  
Regorafenib hydrate (JAN)  <JP/US>
 D05029  
Midostaurin (JAN/USAN/INN)  <US>
 DG01948  
Gilteritinib
  D10709  
Gilteritinib (USAN/INN)
  D10800  
Gilteritinib fumarate (JAN/USAN)  <JP/US>
 D10926  
Entrectinib (JAN/USAN/INN)  <JP/US>
 DG02960  
Pexidartinib
  D11270  
Pexidartinib (USAN/INN)
  D11271  
Pexidartinib hydrochloride (JAN/USAN)  <US>
 DG02081  
Capmatinib
  D10696  
Capmatinib (USAN/INN)
  D10891  
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN)  <JP/US>
 DG03087  
Tepotinib
  D11717  
Tepotinib (USAN/INN)
  D11073  
Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN)  <JP/US>
 D11713  
Selpercatinib (JAN/USAN/INN)  <JP/US>
 D11454  
Repotrectinib (JAN/USAN)  <JP/US>
 D03259  
Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN)  <JP/US>
 D10954  
Mirvetuximab soravtansine (USAN/INN); Mirvetuximab soravtansine (genetical recombination) (JAN)  <US>
 DG01403  
Panobinostat
  D10319  
Panobinostat (USAN/INN)
  D10019  
Panobinostat lactate (JAN)
 D08870  
Belinostat (USAN/INN)  <US>
 D12483  
Olutasidenib (USAN/INN)  <US>
 D08914  
Eribulin mesylate (USAN); Eribulin mesilate (JP18)  <JP/US>
 D11222  
Selinexor (USAN/INN)  <US>
 D12301  
Adagrasib (USAN/INN)  <US>
 DG03016  
Nirogacestat
  D10960  
Nirogacestat (USAN/INN)
  D11453  
Nirogacestat hydrobromide (USAN)  <US>
 DG00734  
Tamoxifen
  D08559  
Tamoxifen (INN)
  D00966  
Tamoxifen citrate (JP18/USP)  <JP/US>
 DG00735  
Toremifene
  D08620  
Toremifene (INN)
  D00967  
Toremifene citrate (JAN/USAN)  <JP/US>
 D01161  
Fulvestrant (JAN/USP/INN)  <JP/US>
 DG03078  
Elacestrant
  D11671  
Elacestrant (USAN/INN)
  D11672  
Elacestrant hydrochloride (USAN)  <US>
 D10218  
Enzalutamide (JAN/USAN)  <JP/US>
 D11040  
Apalutamide (JAN/INN)  <JP/US>
 D00964  
Letrozole (JAN/USP/INN)  <JP/US>
 D00963  
Exemestane (JAN/USP/INN)  <JP/US>
 D09701  
Abiraterone acetate (JAN/USP)  <JP/US>
 DG02927  
Leniolisib
  D11158  
Leniolisib (USAN/INN)
  D11159  
Leniolisib phosphate (JAN/USAN)  <US>
 D11510  
Mavorixafor (USAN)  <US>
 D00184  
Cyclosporine (USP); Ciclosporin (JP18)  <JP/US>
 DG03109  
Belumosudil
  D11815  
Belumosudil (USAN)
  D11816  
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN)  <JP/US>
 D12285  
Remibrutinib (JAN/USAN/INN)  <US>
 D09033  
Voclosporin (JAN/USAN/INN)  <JP/US>
 DG03018  
Siponimod
  D11460  
Siponimod (USAN/INN)
  D11072  
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN)  <JP/US>
 DG02444  
Etrasimod
  D10930  
Etrasimod (USAN)
  D10931  
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN)  <JP/US>
 DG00742  
Tofacitinib
  D09970  
Tofacitinib (USAN)
  D09783  
Tofacitinib citrate (JAN/USAN)  <JP/US>
 DG02829  
Upadacitinib
  D10994  
Upadacitinib (USAN/INN)
  D10995  
Upadacitinib tartrate (USAN)
  D11048  
Upadacitinib hydrate (JAN)  <JP/US>
 DG03114  
Deuruxolitinib
  D11866  
Deuruxolitinib (USAN)
  D11867  
Deuruxolitinib phosphate (USAN)  <US>
 D11093  
Avacopan (JAN/USAN/INN)  <JP/US>
 D00749  
Leflunomide (JAN/USP/INN)  <JP/US>
 D08976  
Pomalidomide (JAN/USAN/INN)  <JP/US>
 D00969  
Meloxicam (JAN/USP/INN)  <JP/US>
 D11576  
Naproxen and esomeprazole magnesium  <US>
 D00570  
Colchicine (JP18/USP)  <JP/US>
 D11406  
Risdiplam (JAN/USAN/INN)  <JP/US>
 D09365  
Palovarotene (JAN/USAN/INN)  <US>
 D00542  
Halothane (JP18/USP/INN)
 DG00791  
Fentanyl
  D00320  
Fentanyl (JAN/USP/INN)  <JP/US>
  D01399  
Fentanyl citrate (JP18/USP)  <JP/US>
  D10811  
Fentanyl hydrochloride (JAN)
 D03852  
Droperidol and fentanyl citrate
 DG01829  
Esketamine
  D07283  
Esketamine (USAN/INN)
  D10627  
Esketamine hydrochloride (JAN/USAN)  <US>
 DG00801  
Bupivacaine
  D07552  
Bupivacaine (USAN/INN)  <US>
  D01450  
Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18)  <JP/US>
 DG00806  
Ropivacaine
  D08490  
Ropivacaine (INN)
  D04048  
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN)  <JP/US>
 DG00807  
Levobupivacaine
  D08116  
Levobupivacaine (INN)
  D01287  
Levobupivacaine hydrochloride (JAN/USAN)  <JP>
 D02740  
Lidocaine and prilocaine  <JP/US>
 DG00813  
Oxycodone
  D05312  
Oxycodone (USAN/INN)  <US>
  D00847  
Oxycodone hydrochloride (USP)  <US>
  D02175  
Compound oxycodone (JP18)
  D03783  
Oxycodone terephthalate (USP)
  D05462  
Oxycodone hydrochloride hydrate (JP18)  <JP>
 DG00814  
Dihydrocodeine
  D07831  
Dihydrocodeine (INN)
  D01481  
Dihydrocodeine phosphate (JP18)  <JP>
  D03825  
Dihydrocodeine bitartrate (USP)
  D07832  
Dihydrocodeine thiocyanate
 D08695  
dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea  <JP>
 DG00820  
Buprenorphine
  D07132  
Buprenorphine (JAN/INN)  <JP/US>
  D00836  
Buprenorphine hydrochloride (JP18/USP)  <JP/US>
 D09999  
Tramadol hydrochloride and acetaminophen  <JP/US>
 D11573  
Oxycodone and ibuprofen
 DG00824  
Tramadol
  D08623  
Tramadol (INN)
  D01355  
Tramadol hydrochloride (JP18/USP)  <JP/US>
 D00544  
Methoxyflurane (USP/INN)
 DG00833  
Dihydroergotamine
  D07837  
Dihydroergotamine (INN)
  D02211  
Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18)  <US>
  D07838  
Dihydroergotamine tartrate
 DG00834  
Ergotamine
  D07906  
Ergotamine (INN)
  D00679  
Ergotamine tartrate (JP18/USP)  <US>
 D07585  
Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine  <JP>
 DG00837  
Naratriptan
  D08255  
Naratriptan (INN)
  D00674  
Naratriptan hydrochloride (JAN/USP)  <JP/US>
 DG00839  
Almotriptan
  D02824  
Almotriptan (USAN)
  D02825  
Almotriptan malate (USP)  <US>
 DG00840  
Eletriptan
  D07887  
Eletriptan (INN)
  D01973  
Eletriptan hydrobromide (JAN/USAN)  <JP/US>
  D11617  
Eletriptan hydrobromide monohydrate
 D10673  
Ubrogepant (USAN/INN)  <US>
 DG01845  
Rimegepant
  D10662  
Rimegepant (USAN/INN)
  D10663  
Rimegepant sulfate (USAN); Rimegepant sulfate hydrate (JAN)  <JP/US>
 DG03330  
Atogepant
  D11313  
Atogepant (USAN)  <US>
  D13026  
Atogepant hydrate (JAN)
 D00539  
Ethosuximide (JP18/USP/INN)  <JP/US>
 D00252  
Carbamazepine (JP18/USP/INN)  <JP/US>
 D00537  
Topiramate (JAN/USP/INN)  <JP/US>
 D05928  
Stiripentol (JAN/USAN/INN)  <JP>
 D07299  
Lacosamide (JAN/USAN/INN)  <JP/US>
 D10915  
Cannabidiol (JAN/USAN/INN)  <US>
 D11150  
Cenobamate (JAN/USAN/INN)  <US>
 D04300  
Ganaxolone (USAN/INN)  <US>
 DG00864  
Selegiline
  D03731  
Selegiline (USAN/INN)  <US>
  D00785  
Selegiline hydrochloride (JAN/USP)  <JP/US>
 DG01260  
Safinamide
  D10158  
Safinamide (USAN/INN)
  D10191  
Safinamide mesylate (USAN); Safinamide mesilate (JAN)  <JP/US>
 D04641  
Istradefylline (JAN/USAN/INN)  <JP/US>
 DG00885  
Haloperidol
  D00136  
Haloperidol (JP18/USP/INN)  <JP/US>
  D01898  
Haloperidol decanoate (JAN/USP)  <JP/US>
  D08035  
Haloperidol lactate  <US>
 DG00890  
Bromperidol
  D01101  
Bromperidol (JAN/USAN/INN)  <JP>
  D02626  
Bromperidol decanoate (USAN)
 D04820  
Lurasidone hydrochloride (JAN/USAN)  <JP/US>
 D00560  
Pimozide (JP18/USP/INN)  <US>
 DG00897  
Loxapine
  D02340  
Loxapine (USAN/INN)
  D00794  
Loxapine succinate (USP)  <US>
  D08148  
Loxapine hydrochloride
 D00283  
Clozapine (JAN/USP/INN)  <JP/US>
 DG00899  
Quetiapine
  D08456  
Quetiapine (INN)
  D00458  
Quetiapine fumarate (JP18/USP)  <JP/US>
 D00426  
Risperidone (JP18/USP/INN)  <JP/US>
 DG00906  
Aripiprazole
  D01164  
Aripiprazole (JP18/USP/INN)  <JP/US>
  D10355  
Aripiprazole cavoxil (USAN)
  D10364  
Aripiprazole lauroxil (USAN)  <US>
  D10516  
Aripiprazole hydrate (JAN)  <JP/US>
 D02666  
Iloperidone (USAN/INN)  <US>
 DG01305  
Cariprazine
  D09997  
Cariprazine (USAN/INN)
  D09876  
Cariprazine hydrochloride (JAN/USAN)  <US>
 DG03365  
Brexpiprazole
  D10309  
Brexpiprazole (JAN/USAN/INN)  <JP/US>
  D13183  
Brexpiprazole fumarate hydrate (JAN)
 D08969  
Pimavanserin tartrate (USAN)  <US>
 D00293  
Diazepam (JP18/USP/INN)  <JP/US>
 D01253  
Clobazam (JAN/USAN/INN)  <JP/US>
 D08283  
Nordazepam (INN)
 D01293  
Ethyl loflazepate (JP18/INN)  <JP>
 D01514  
Etizolam (JP18/INN)  <JP>
 D01316  
Mexazolam (JAN/INN)  <JP>
 D00387  
Triazolam (JP18/USP/INN)  <JP/US>
 DG00920  
Midazolam
  D00550  
Midazolam (JAN/USP/INN)  <JP/US>
  D00696  
Midazolam hydrochloride (USAN)  <US>
  D05028  
Midazolam maleate (USAN)
 D01744  
Brotizolam (JP18/USAN/INN)  <JP>
 D00457  
Quazepam (JAN/USP/INN)  <JP/US>
 D01372  
Zopiclone (JP18/INN)  <JP>
 DG00922  
Zolpidem
  D08690  
Zolpidem (INN)
  D00706  
Zolpidem tartrate (JP18/USP)  <JP/US>
 D00530  
Zaleplon (JAN/USP/INN)  <US>
 D02624  
Eszopiclone (JAN/USP/INN)  <JP/US>
 D09388  
Tasimelteon (USAN/INN)  <US>
 D11022  
Lemborexant (JAN/USAN/INN)  <JP/US>
 DG00928  
Imipramine
  D08070  
Imipramine (INN)
  D00815  
Imipramine hydrochloride (JP18/USP)  <JP/US>
  D08071  
Imipramine pamoate (USP)  <US>
 DG00929  
Clomipramine
  D07727  
Clomipramine (INN)
  D00811  
Clomipramine hydrochloride (JP18/USP)  <JP/US>
 DG00934  
Amitriptyline
  D07448  
Amitriptyline (INN)
  D00809  
Amitriptyline hydrochloride (JP18/USP)  <JP/US>
 DG00943  
Citalopram
  D07704  
Citalopram (USP/INN)
  D00822  
Citalopram hydrobromide (USP)  <US>
  D07705  
Citalopram hydrochloride
 DG00945  
Sertraline
  D02360  
Sertraline (INN)
  D00825  
Sertraline hydrochloride (JAN/USP)  <JP/US>
 DG00947  
Escitalopram
  D07913  
Escitalopram (INN)
  D02567  
Escitalopram oxalate (JAN/USP)  <JP/US>
 DG00951  
Mianserin
  D08216  
Mianserin (INN)
  D01358  
Mianserin hydrochloride (JAN/USAN)  <JP>
 DG00952  
Trazodone
  D08626  
Trazodone (INN)
  D00820  
Trazodone hydrochloride (JAN/USP)  <JP/US>
 DG02838  
Mirtazapine
  D00563  
Mirtazapine (JAN/USP/INN)  <JP/US>
  D11056  
Mirtazapine hydrate (JAN)
 DG00959  
Venlafaxine
  D08670  
Venlafaxine (INN)
  D00821  
Venlafaxine hydrochloride (JAN/USP)  <JP/US>
  D12403  
Venlafaxine besylate monohydrate  <US>
 D04314  
Gepirone hydrochloride (USAN)  <US>
 DG00963  
Desvenlafaxine
  D07793  
Desvenlafaxine (INN)  <US>
  D02570  
Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN)  <US>
  D11619  
Desvenlafaxine succinate anhydrous
 DG00964  
Vilazodone
  D09698  
Vilazodone (USAN/INN)
  D09699  
Vilazodone hydrochloride (USAN)  <US>
 DG00965  
Vortioxetine
  D10184  
Vortioxetine (USAN)
  D10185  
Vortioxetine hydrobromide (JAN/USAN)  <JP/US>
  D12544  
Vortioxetine hemihydrobromide (USAN)
 D11793  
Zuranolone (JAN/USAN/INN)  <JP/US>
 D01832  
Modafinil (JAN/USP/INN)  <JP/US>
 D03215  
Armodafinil (USAN/INN)  <US>
 DG00983  
Donepezil
  D07869  
Donepezil (JAN/INN)  <JP>
  D00670  
Donepezil hydrochloride (JP18/USP)  <JP/US>
 DG00985  
Galantamine
  D04292  
Galantamine (USAN/INN)
  D02173  
Galantamine hydrobromide (JAN/USP)  <JP/US>
 DG00993  
Cevimeline
  D07667  
Cevimeline (INN)
  D00661  
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN)  <JP/US>
 DG00999  
Methadone
  D08195  
Methadone (BAN)
  D02102  
Methadone hydrochloride (JAN/USP)  <JP/US>
 DG01000  
Levacetylmethadol
  D04716  
Levomethadyl acetate (USAN); Levacetylmethadol (INN)
  D00840  
Levomethadyl acetate hydrochloride (USAN)
 D08575  
Tetrabenazine (JAN/INN)  <JP/US>
 DG03021  
Pitolisant
  D10749  
Pitolisant (USAN/INN)
  D11490  
Pitolisant hydrochloride (JAN/USAN)  <US>
 DG02115  
Valbenazine
  D10675  
Valbenazine (USAN/INN)
  D10999  
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN)  <JP/US>
 DG01015  
Hydroxychloroquine
  D08050  
Hydroxychloroquine (INN)
  D02114  
Hydroxychloroquine sulfate (JAN/USP)  <JP/US>
 DG01019  
Quinine
  D08460  
Quinine (BAN)
  D01663  
Quinine ethylcarbonate (JP18)
  D02261  
Quinine hydrochloride hydrate (JP18)
  D02262  
Quinine sulfate (USP); Quinine sulfate hydrate (JP18)  <US>
  D05681  
Quinine ascorbate (USAN)
  D08461  
Quinine dihydrochloride
 D11252  
Fexinidazole (USAN/INN)  <US>
 D00471  
Praziquantel (JAN/USP/INN)  <JP/US>
 DG01040  
Flunisolide
  C07005  
Flunisolide
  D00324  
Flunisolide (JAN/USP)  <US>
  D04214  
Flunisolide acetate (USAN)
 D01703  
Ciclesonide (JAN/USAN/INN)  <JP/US>
 D08699  
Salmeterol xinafoate and fluticasone propionate  <JP/US>
 DG01051  
Salmeterol
  D05792  
Salmeterol (USAN/INN)
  D00687  
Salmeterol xinafoate (JAN/USP)  <JP/US>
 DG01055  
Procaterol
  D08424  
Procaterol (INN)
  D02404  
Procaterol hydrochloride (USAN)
  D05366  
Procaterol hydrochloride hydrate (JP18)  <JP>
 DG01057  
Indacaterol
  D09318  
Indacaterol (USAN/INN)
  D09319  
Indacaterol maleate (JAN/USAN)  <JP>
  D11009  
Indacaterol acetate (JAN)
 D09595  
Budesonide and formoterol fumarate dihydrate  <JP/US>
 D10501  
Fluticasone furoate and vilanterol trifenatate  <JP/US>
 D10506  
Fluticasone propionate and formoterol fumarate hydrate  <JP>
 D10533  
Umeclidinium bromide and vilanterol  <JP/US>
 D10505  
Glycopyrronium bromide and indacaterol maleate  <JP>
 DG01065  
Pranlukast
  D08408  
Pranlukast (INN)
  D02732  
Pranlukast hydrate (JP18)  <JP>
 DG01066  
Montelukast
  D08229  
Montelukast (INN)
  D00529  
Montelukast sodium (JP18/USP)  <JP/US>
 DG01074  
Ethylmorphine
  D07929  
Ethylmorphine (BAN)
  D02205  
Ethylmorphine hydrochloride hydrate (JP18)
 DG01075  
Hydrocodone
  D08045  
Hydrocodone (INN)
  D03725  
Hydrocodone bitartrate (USP)  <US>
  D04461  
Hydrocodone polistirex (USAN)
  D08046  
Hydrocodone hydrochloride
 DG01076  
Codeine
  C06174  
Codeine
  D00195  
Codeine (USP)
  D02101  
Codeine phosphate (USP); Codeine phosphate hydrate (JP18)  <JP>
  D03579  
Codeine polistirex (USAN)
  D03580  
Codeine sulfate (USP)  <US>
  D07740  
Codeine hydrochloride
 D12312  
Codeine phosphate and chlorpheniramine maleate  <US>
 D04340  
Dextromethorphan hydrobromide and potassium cresolsulfonate  <JP>
 D04313  
Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate  <JP>
 D04447  
Betamethasone and d-chlorpheniramine maleate  <JP>
 D12313  
Chlorpheniramine polistirex and codeine polistirex
 DG01108  
Levocetirizine
  D07402  
Levocetirizine (USAN/INN)
  D08118  
Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN)  <JP/US>
 D00364  
Loratadine (JAN/USP/INN)  <JP/US>
 D01478  
Ebastine (JP18/USAN/INN)  <JP>
 DG01118  
Rupatadine
  D07407  
Rupatadine (USAN/INN)
  D08497  
Rupatadine fumarate (JAN/USAN)  <JP>
 DG01119  
Doxapram
  D07873  
Doxapram (INN)
  D01872  
Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18)  <JP/US>
 DG01135  
Dorzolamide
  D07871  
Dorzolamide (INN)
  D00653  
Dorzolamide hydrochloride (JP18/USP)  <JP/US>
 D10512  
Brinzolamide and timolol maleate  <JP>
 D08493  
Dorzolamide hydrochloride and timolol maleate (JP18)  <JP/US>
 D06405  
Nalfurafine hydrochloride (JAN/USAN)  <JP>
 DG01307  
Rilmazafone
  D08481  
Rilmazafone (INN)
  D01564  
Rilmazafone hydrochloride hydrate (JP18)  <JP>
 DG01333  
Sarpogrelate
  D08508  
Sarpogrelate (INN)
  D01624  
Sarpogrelate hydrochloride (JP18)  <JP>
 DG01430  
Paclitaxel
  D00491  
Paclitaxel (JAN/USP/INN)  <JP/US>
  D05333  
Paclitaxel poliglumex (USAN/INN)
 DG03177  
Imlunestrant
  D12216  
Imlunestrant (USAN)
  D12217  
Imlunestrant tosylate (USAN); Imlunestrant tosilate (JAN)  <JP/US>
 D01098  
Maxacalcitol (JAN/USAN/INN)  <JP>
 D01145  
Azelnidipine (JP18/INN)  <JP>
 D01176  
Blonanserin (JAN/INN)  <JP>
 D01418  
Tamibarotene (JAN/USAN/INN)  <JP>
 D01468  
Nemonapride (JAN/INN)  <JP>
 D04052  
Epinephrine and lidocaine hydrochloride  <JP/US>
 D04446  
Betamethasone acetate and betamethasone sodium phosphate  <JP/US>
 D04813  
Lidocaine hydrochloride and epinephrine bitartrate  <JP/US>
 D08856  
Anamorelin hydrochloride (JAN/USAN)  <JP>
 D09594  
Olmesartan medoxomil and azelnidipine  <JP>
 D10524  
Azilsartan and amlodipine besilate  <JP>
 D10525  
Valsartan and cilnidipine  <JP>
 D10897  
Teneligliptin and canagliflozin  <JP>
 D12611  
Vornorexant hydrate (JAN)  <JP>
 DG03280  
Dordaviprone
  D12733  
Dordaviprone (USAN/INN)
  D12734  
Dordaviprone hydrochloride (JAN/USAN)  <US>
 DG03287  
Brensocatib
  D12120  
Brensocatib (USAN/INN)
  D12746  
Brensocatib hydrate (JAN)  <US>
 D11628  
Benzhydrocodone and acetaminophen  <US>
 D11656  
Azelastine hydrochloride and fluticasone propionate  <US>
 D11706  
Omeprazole and sodium bicarbonate  <US>
 D11851  
Butalbital, acetaminophen, caffeine and codeine phosphate  <US>
 D11860  
Butalbital, aspirin, caffeine and codeine  <US>
 D12130  
Drospirenone, ethinyl estradiol and levomefolate calcium  <US>
 D12497  
Drospirenone and estradiol  <US>
 D12756  
Vonoprazan and amoxicillin  <US>
 D13120  
Avutometinib and defactinib  <US>
 DG01850  
Benzhydrocodone
  D10612  
Benzhydrocodone (USAN/INN)
  D10692  
Benzhydrocodone hydrochloride (USAN)
 DG01977  
Dihydroergotoxine
  D07839  
Dihydroergotoxine
  D02268  
Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18)
 D01562  
Aranidipine (JAN/INN)
 D01855  
Mozavaptane hydrochloride (JAN)
 D04338  
Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride
 D08697  
Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate
 D11553  
Lidocaine and tetracaine
 D11616  
Aspirin and omeprazole
Hydrocortisone
 D00088  
Hydrocortisone (JP18/USP/INN)  <JP/US>
 D00165  
Hydrocortisone acetate (JP18/USP)  <US>
 D00976  
Hydrocortisone cypionate
 D00977  
Hydrocortisone sodium phosphate (JP18/USP)  <JP>
 D00978  
Hydrocortisone sodium succinate (JP18/USP)  <JP/US>
 D01442  
Hydrocortisone succinate (JP18)
 D01619  
Hydrocortisone butyrate (JP18/USP)  <JP/US>
 D01886  
Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN)  <JP>
 D02288  
Hydrocortisone valerate (USP)  <US>
 D04467  
Hydrocortisone hemisuccinate (USP)
 D06876  
Hydrocortisone aceponate (INN)
 D09796  
Hydrocortisone caproate (JAN)
D00472  
Prednisolone (JP18/USP/INN)  <JP/US>
D11858  
Omeprazole magnesium, amoxicillin and rifabutin  <US>
Cisapride
 D00274  
Cisapride (USP/INN)
 D02092  
Cisapride (JAN)
Dolasetron
 D07867  
Dolasetron (INN)
 D00725  
Dolasetron mesylate (USP)
Naloxegol
 D10479  
Naloxegol (USAN/INN)
 D10375  
Naloxegol oxalate (USAN)  <US>
D10865  
Bexagliflozin (USAN)  <US>
D04768  
Lonafarnib (JAN/USAN/INN)  <JP/US>
D09017  
Ticagrelor (JAN/USAN/INN)  <JP/US>
D00297  
Digitoxin (JAN/USP/INN)
Dronedarone
 D02537  
Dronedarone (INN)
 D03914  
Dronedarone hydrochloride (USP)  <US>
Ranolazine
 D05700  
Ranolazine (USAN/INN)  <US>
 D05701  
Ranolazine hydrochloride (USAN)
D09572  
Riociguat (JAN/USAN/INN)  <JP/US>
D12963  
Macitentan and tadalafil  <JP/US>
Conivaptan
 D07748  
Conivaptan (INN)
 D01236  
Conivaptan hydrochloride (JAN/USAN)
Lercanidipine
 D08111  
Lercanidipine (INN)
 D01849  
Lercanidipine hydrochloride (JAN/USAN)
D11776  
Sparsentan (JAN/USAN/INN)  <US>
D10711  
Pemafibrate (JAN)  <JP>
Erythromycin
 D00140  
Erythromycin (JP18/USP/INN)  <JP/US>
 D00851  
Erythromycin estolate (USP); Erythromycin estorate (JAN)
 D01361  
Erythromycin ethylsuccinate (JP18/USP)  <JP/US>
 D02009  
Erythromycin lactobionate (JP18/USP)  <JP/US>
 D02184  
Erythromycin stearate (JP18/USP)  <JP>
 D02523  
Erythromycin acistrate (USAN)
 D02524  
Erythromycin gluceptate (USP)
 D02525  
Erythromycin propionate (USAN)
 D03098  
Berythromycin (USAN/INN)
 D04054  
Erythromycin salnacedin (USAN)
 D07909  
Erythromycin thiocyanate
 D07910  
Erythromycin stinoprate (INN)
D10461  
Dienogest and estradiol valerate  <US>
D12586  
Mifepristone and misoprostol  <JP>
D12137  
Elagolix, estradiol and norethisterone  <US>
D01710  
Roxithromycin (JP18/USAN/INN)  <JP>
D01078  
Telithromycin (JAN/USAN/INN)
D00427  
Ritonavir (JAN/USP/INN)  <JP/US>
Ensitrelvir
 D12619  
Ensitrelvir (USAN/INN)
 D12353  
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN)  <JP>
Delavirdine
 D07782  
Delavirdine (INN)
 D00895  
Delavirdine mesylate (USAN); Delavirdine mesilate (JAN)
Rilpivirine
 D09720  
Rilpivirine (JAN/USAN/INN)  <JP>
 D09958  
Rilpivirine hydrochloride (JAN/USAN)  <JP/US>
D10624  
Doravirine (JAN/USAN/INN)  <JP/US>
Simeprevir
 D10081  
Simeprevir (JAN/USAN)
 D10469  
Simeprevir sodium (JAN)
D10093  
Asunaprevir (JAN/USAN)
D10625  
Elbasvir (JAN/USAN/INN)
Grazoprevir
 D11565  
Grazoprevir (USAN/INN)
 D10639  
Grazoprevir (USAN); Grazoprevir hydrate (JAN)
D10582  
Dasabuvir, ombitasvir, paritaprevir and ritonavir
D10882  
Daclatasvir, asunaprevir and beclabuvir
D11521  
Lamivudine, nevirapine and zidovudine
D10571  
Rilpivirine hydrochloride, tenofovir disoproxil fumarate and emtricitabine  <US>
D10756  
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil  <US>
D02498  
Lopinavir and ritonavir  <JP/US>
D10832  
Darunavir and cobicistat  <JP/US>
D10835  
Emtricitabine and tenofovir alafenamide  <JP/US>
D10755  
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide  <JP/US>
D10836  
Emtricitabine, rilpivirine and tenofovir alafenamide  <JP/US>
D11282  
Dolutegravir sodium and rilpivirine hydrochloride  <JP/US>
D11382  
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide  <JP/US>
D11396  
Doravirine, lamivudine and tenofovir disoproxil  <US>
D10564  
Amenamevir (JAN/INN)  <JP>
Lenacapavir
 D12161  
Lenacapavir (USAN/INN)
 D12162  
Lenacapavir sodium (JAN/USAN)  <JP/US>
Vincristine
 D08679  
Vincristine (INN)
 D02197  
Vincristine sulfate (JP18/USP)  <JP/US>
Vindesine
 D06304  
Vindesine (USAN/INN)
 D01769  
Vindesine sulfate (JAN/USAN)  <JP>
Cabazitaxel
 D09755  
Cabazitaxel (USAN/INN)
 D10452  
Cabazitaxel acetonate (JAN)  <JP/US>
Ponatinib
 D09950  
Ponatinib (USAN/INN)
 D09951  
Ponatinib hydrochloride (JAN/USAN)  <JP/US>
D10766  
Osimertinib mesylate (USAN); Osimertinib mesilate (JAN)  <JP/US>
Mobocertinib
 D12001  
Mobocertinib (USAN/INN)
 D11969  
Mobocertinib succinate (JAN)
D10551  
Ceritinib (JAN/USAN/INN)  <JP/US>
D11012  
Lorlatinib (JAN/USAN/INN)  <JP/US>
D10688  
Abemaciclib (JAN/USAN/INN)  <JP/US>
Tucatinib
 D11141  
Tucatinib (USAN/INN)  <US>
 D12442  
Tucatinib ethanolate (JAN)
Sevabertinib
 D13098  
Sevabertinib (USAN)
 D13116  
Sevabertinib hydrate (JAN)  <US>
D11977  
Fruquintinib (JAN/USAN)  <JP/US>
D10223  
Ibrutinib (JAN/USAN)  <JP/US>
Acalabrutinib
 D10893  
Acalabrutinib (JAN/USAN/INN)  <JP>
 D11720  
Acalabrutinib maleate (USAN)
 D12704  
Acalabrutinib maleate hydrate (JAN)  <JP/US>
D11422  
Zanubrutinib (JAN/USAN/INN)  <JP/US>
D10560  
Idelalisib (JAN/USAN/INN)  <US>
Copanlisib
 D10867  
Copanlisib (USAN/INN)
 D10797  
Copanlisib hydrochloride (USAN)
 D10798  
Copanlisib hydrochloride hydrate (JAN)
Lenvatinib
 D09919  
Lenvatinib (USAN/INN)
 D09920  
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN)  <JP/US>
Quizartinib
 D09955  
Quizartinib (USAN/INN)
 D09956  
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN)  <JP/US>
Larotrectinib
 D11137  
Larotrectinib (USAN/INN)
 D11138  
Larotrectinib sulfate (JAN/USAN)  <JP/US>
D11371  
Capivasertib (JAN/USAN)  <JP/US>
D10761  
Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN)  <JP/US>
D06637  
Romidepsin (JAN/USAN/INN)  <JP/US>
Sonidegib
 D10119  
Sonidegib (USAN/INN)
 D10729  
Sonidegib phosphate (USAN)  <US>
D09730  
Olaparib (JAN/USAN/INN)  <JP/US>
Vorasidenib
 D11834  
Vorasidenib (USAN/INN)
 D11835  
Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN)  <JP/US>
D12055  
Sotorasib (JAN/USAN)  <JP/US>
D12975  
Nerandomilast (JAN/USAN/INN)  <US>
Dantrolene
 D02347  
Dantrolene (USAN/INN)
 D02274  
Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18)  <JP/US>
D03844  
Phenytoin, phenobarbital and caffeine and sodium benzoate
D00538  
Zonisamide (JP18/USP/INN)  <JP/US>
Perampanel
 D08964  
Perampanel (JAN/USAN)
 D10780  
Perampanel hydrate (JAN)  <JP/US>
D00225  
Alprazolam (JP18/USP/INN)  <JP/US>
D02615  
Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital
D00311  
Estazolam (JP18/USP/INN)  <JP/US>
D10082  
Suvorexant (JAN/USAN)  <JP/US>
Daridorexant
 D11886  
Daridorexant (USAN/INN)
 D11887  
Daridorexant hydrochloride (JAN/USAN)  <JP>
D10964  
Omaveloxolone (USAN/INN)  <US>
Mefloquine
 D04895  
Mefloquine (USAN/INN)
 D00831  
Mefloquine hydrochloride (JP18/USP)  <JP/US>
D02484  
Artemether and lumefantrine  <JP/US>
Dexchlorpheniramine
 D07803  
Dexchlorpheniramine (INN)
 D00668  
Dexchlorpheniramine maleate (USP); d-Chlorpheniramine maleate (JP18)  <JP/US>
D00234  
Astemizole (JAN/USP/INN)
D00521  
Terfenadine (JAN/USAN/INN)
D11700  
Elexacaftor, ivacaftor and tezacaftor  <US>
D13024  
Vanzacaftor, tezacaftor and deutivacaftor  <US>
D09881  
Cobicistat (JAN/USAN/INN)  <US>
Isavuconazonium
 D10644  
Isavuconazonium (USAN)
 D10643  
Isavuconazonium sulfate (JAN/USAN)  <JP/US>
Colforsin
 D03584  
Colforsin (USAN/INN)
 D01697  
Colforsin daropate hydrochloride (JAN)  <JP>
Taletrectinib
 D12363  
Taletrectinib (USAN/INN)
 D12364  
Taletrectinib adipate (JAN/USAN)  <JP/US>
D10892  
Esaxerenone (JAN/INN)  <JP>
D03009  
Atrasentan hydrochloride (USAN)  <US>
Temsavir
 D10734  
Temsavir (USAN/INN)
 D10707  
Fostemsavir (USAN)
 D10708  
Fostemsavir tromethamine (USAN)  <US>
Ensartinib
 D11346  
Ensartinib (USAN)
 D11356  
Ensartinib hydrochloride (USAN)  <US>
D11873  
Rilzabrutinib (JAN/USAN/INN)  <US>
D12419  
Ziftomenib (USAN/INN)  <US>
D12860  
Suzetrigine (USAN/INN)  <US>
D11966  
Cabotegravir and rilpivirine  <US>
D01425  
Lopinavir (JAN/USP/INN)
D05152  
Netupitant (USAN/INN)
D09987  
Vaniprevir (JAN/USAN/INN)
D12506  
Sunvozertinib (USAN/INN)
D12253  
Aficamten (USAN/INN)
 » expand
Class
Metabolizing enzyme substrate
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