KEGG   DRUG: エチニルエストラジオール・ノルエチステロン
エントリ  
D04483            Mixture   Drug                                   
一般名   
エチニルエストラジオール・ノルエチステロン;
Ethinylestradiol and norethisterone;
Norethindrone and ethinyl estradiol
商品名   
  後発品
米国の商品 
  後発品
ALYACEN 1/35 (A-S Medication Solutions), ARANELLE (Teva Pharmaceuticals USA), AUROVELA 1.5/30 (Aurobindo Pharma Limited), AUROVELA 1/20 (Aurobindo Pharma Limited), AUROVELA 24 FE (Aurobindo Pharma Limited), AUROVELA FE (Aurobindo Pharma Limited), AUROVELA FE 1/20 (Aurobindo Pharma Limited), BALZIVA (Teva Pharmaceuticals USA), BLISOVI 24 FE (Lupin Pharmaceuticals), BLISOVI FE 1.5/30 (Lupin Pharmaceuticals), BLISOVI FE 1/20 (Lupin Pharmaceuticals), BRIELLYN (Glenmark Pharmaceuticals), CHARLOTTE 24FE (Glenmark Pharmaceuticals), CYONANZ (Aurobindo Pharma Limited), DASETTA 1/35 (Northstar Rx LLC), DASETTA 7/7/7 (Northstar Rx LLC), FEIRZA 1.5/30 TM (Xiromed LLC), FEIRZA 1/20 (Xiromed LLC), FINZALA (Teva Pharmaceuticals USA), FYAVOLV (Lupin Pharmaceuticals), GALBRIELA (Xiromed), GEMMILY (Xiromed), HAILEY 1.5/30 (Glenmark Pharmaceuticals), HAILEY 24 FE (Glenmark Pharmaceuticals), HAILEY FE 1.5/30 (Glenmark Pharmaceuticals), HAILEY FE 1/20 (Glenmark Pharmaceuticals), JINTELI (Teva Pharmaceuticals USA), JUNEL (A-S Medication Solutions), JUNEL (PD-Rx Pharmaceuticals), JUNEL (Proficient Rx LP), JUNEL (RedPharm Drug), JUNEL (Teva Pharmaceuticals USA), JUNEL FE (Direct_Rx), JUNEL FE (Teva Pharmaceuticals USA), JUNEL FE 1.5/30 (Proficient Rx LP), JUNEL FE 1/20 (Preferred Pharmaceuticals), KAITLIB FE (Lupin Pharmaceuticals), LARIN 1.5/30 (Northstar Rx LLC), LARIN 1/20 (Northstar Rx LLC), LARIN 24 FE (Northstar Rx LLC), LARIN FE 1.5/30 (Northstar Rx LLC), LARIN FE 1/20 (Northstar Rx LLC), LAYOLIS FE (Actavis Pharma), LEENA (Mayne Pharma), LOESTRIN (Teva Women's Health LLC), LUIZZA 1.5/30 (Xiromed LLC), MELODETTA 24 FE (Amneal Pharmaceuticals NY LLC), MERZEE (Lupin Pharmaceuticals), MICROGESTIN 1.5/30 (Dr. Reddy's Laboratories), MICROGESTIN 1.5/30 (Mayne Pharma), MICROGESTIN 1/20 (Dr.Reddy's Laboratories), MICROGESTIN 1/20 (Mayne Pharma), MICROGESTIN 24 FE (Mayne Pharma), MICROGESTIN FE 1.5/30 (Dr. Reddy's Laboratories), MICROGESTIN FE 1.5/30 (Mayne Pharma), MICROGESTIN FE 1.5/30 (Proficient Rx LP), MICROGESTIN FE 1/20 (Dr. Reddy's Laboratories), MICROGESTIN FE 1/20 (Mayne Pharma), NECON (Dr. Reddy's Laboratories), NECON (Mayne Pharma), NEXESTA FE (Aurobindo Pharma Limited), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (A-S Medication Solutions), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Amneal Pharmaceuticals NY LLC), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Glenmark Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Glenmark Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Mylan Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Mylan Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Mylan Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Mylan Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Nivagen Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL (Xiromed), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Amneal Pharmaceuticals NY LLC), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Glenmark Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Glenmark Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Mylan Pharmaceuticals), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL, AND FERROUS FUMARATE (Amneal Pharmaceuticals NY LLC), NORETHINDRONE ACETATE AND ETHINYL ESTRADIOL, AND FERROUS FUMARATE (Northstar Rx LLC), NORETHINDRONE AND ETHINYL ESTRADIOL (Glenmark Pharmaceuticals), NORETHINDRONE AND ETHINYL ESTRADIOL (Naari Pte Limited), NORETHINDRONE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Mylan Pharmaceuticals), NORETHINDRONE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Mylan Pharmaceuticals), NORETHINDRONE AND ETHINYL ESTRADIOL AND FERROUS FUMARATE (Naari Pte Limited), NORTREL (A-S Medication Solutions), NORTREL (Teva Pharmaceuticals USA), NORTREL 7/7/7 (Proficient Rx LP), NORTREL 7/7/7 (Teva Pharmaceuticals USA), NYLIA 1/35 (Aurobindo Pharma Limited), NYLIA 7/7/7 (A-S Medication Solutions), NYLIA 7/7/7 (Aurobindo Pharma Limited), OSHIH (Aurobindo Pharma Limited), PHILITH (Northstar Rx LLC), RHUZDAH (Aurobindo Pharma Limited), TARINA 24 FE (Afaxys Pharma), TARINA FE 1/20 EQ (Afaxys Pharma), TAYSOFY (Amneal Pharmaceuticals LLC), TILIA FE (Dr. Reddy's Laboratories), TILIA FE (Mayne Pharma), TRI-LEGEST FE (Teva Pharmaceuticals USA), VYFEMLA (Lupin Pharmaceuticals), WERA (Northstar Rx LLC), WYMZYA FE (Lupin Pharmaceuticals), XARAH FE (Xiromed LLC), XELRIA FE (Xiromed LLC), ZENCHENT FE (Amneal Pharmaceuticals NY LLC)
成分    
エチニルエストラジオール [DR:D00554], (ノルエチステロン [DR:D00182] | 酢酸ノルエチステロン [DR:D00953])
クラス   
代謝酵素基質薬
 DG01633  CYP3A/CYP3A4基質薬
  DG02913  CYP3A4基質薬
コード   
薬効分類: 2482 2549
ATCコード: G03AA05 G03AB04 G03FA01 G03FB05
商品: D04483<JP/US>
効能    
避妊薬, 月経障害治療薬
コメント  
卵胞ホルモン・黄体ホルモン配合
エチニルエストラジオールは主にCYP3A4により代謝される。
代謝    
Enzyme: CYP3A4 [HSA:1576]
相互作用  

階層分類  
医療用医薬品の薬効分類 [BR:jp08301]
 2  個々の器官系用医薬品
  24  ホルモン剤(抗ホルモン剤を含む)
   248  混合ホルモン剤
    2482  卵胞ホルモン、黄体ホルモン混合製剤
     D04483  エチニルエストラジオール・ノルエチステロン
  25  泌尿生殖器官及び肛門用薬
   254  避妊剤
    2549  その他の避妊剤
     D04483  エチニルエストラジオール・ノルエチステロン
医療用医薬品のATC分類 [BR:jp08303]
 G 泌尿生殖器系と性ホルモン
  G03 性ホルモンと生殖器系モジュレーター
   G03A 全身用ホルモン避妊薬
    G03AA プロゲストゲンとエストロゲン、抱合型
     G03AA05 ノルエチステロンとエチニルエストラジオール
      D04483  エチニルエストラジオール・ノルエチステロン <JP/US>
    G03AB プロゲストゲンとエストロゲン、連続型
     G03AB04 ノルエチステロンとエチニルエストラジオール
      D04483  エチニルエストラジオール・ノルエチステロン <JP/US>
   G03F プロゲストゲンとエストロゲンの配合
    G03FA プロゲストゲンとエストロゲン、抱合型
     G03FA01 ノルエチステロンとエストロゲン
      D04483  エチニルエストラジオール・ノルエチステロン <JP/US>
    G03FB プロゲストゲンとエストロゲン、連続型
     G03FB05 ノルエチステロンとエストロゲン
      D04483  エチニルエストラジオール・ノルエチステロン <JP/US>
医療用医薬品のUSP分類 [BR:jp08302]
 避妊薬
  混合型経口避妊薬
   エチニルエストラジオール・ノルエチステロン
    D04483  エチニルエストラジオール・ノルエチステロン
医薬品グループ [BR:jp08330]
 代謝酵素基質薬
  DG01633  CYP3A/CYP3A4基質薬
   DG02913  CYP3A4基質薬
    D04483  エチニルエストラジオール・ノルエチステロン
薬物代謝酵素とトランスポーター [jp08309.html]
 薬物代謝酵素
  D04483
リンク   
PubChem: 17398126
LinkDB    

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