| Nitrogen mustard analog |
| Isophosphoramide mustard analog |
| Cyclophosphamide |
| Cyclophosphamide (INN) |
| Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18) <JP/US> |
| Ifosfamide (JAN/USP/INN) <JP/US> |
| Trofosfamide (INN) |
| Palifosfamide |
| Palifosfamide (USAN/INN) |
| Palifosfamide tromethamine (USAN) |
| Canfosfamide hydrochloride (USAN) |
| Perfosfamide (USAN/INN) |
| Chlorambucil (JAN/USP/INN) <US> |
| Melphalan |
| Melphalan (JP18/USP/INN) <JP> |
| Melphalan hydrochloride <US> |
| Chlormethine |
| Chlormethine (INN) |
| Mechlorethamine hydrochloride (USP) <US> |
| Prednimustine (USAN/INN) |
| Bendamustine |
| Bendamustine (INN) |
| Bendamustine hydrochloride (JAN/USAN) <JP/US> |
| Bendamustine hydrochloride hydrate (JAN) <JP> |
| Uracil mustard (USAN); Uramustine (INN) |
| Estramustine |
| Estramustine (USAN/INN) |
| Estramustine phosphate sodium (USAN) |
| Estramustine phosphate sodium hydrate (JAN) <JP> |
| Nitrogen mustard N-oxide hydrochloride (JAN) |
| Spiromustine (USAN/INN) |
| Methanesulfonate derivative |
| Busulfan (JP18/USP/INN) <JP/US> |
| Treosulfan (USAN/INN) |
| Mannosulfan (INN) |
| Improsulfan tosilate (JAN) |
| Piposulfan (USAN/INN) |
| Ethylene imine |
| Thiotepa type ethylene imine |
| Thiotepa (JAN/USP/INN) <JP/US> |
| Azetepa (USAN/INN) |
| Benzodepa (USAN/INN) |
| Meturedepa (USAN/INN) |
| Uredepa (USAN/INN) |
| Triaziquone (INN) |
| Carboquone (JAN/INN) |
| Apaziquone (USAN/INN) |
| Diaziquone (USAN/INN) |
| Nitrosourea |
| Carmustine (JAN/USP/INN) <JP/US> |
| Lomustine (USP/INN) <US> |
| Semustine (USAN/INN) |
| Streptozocin (JAN/USAN/INN) <JP/US> |
| Fotemustine (INN/BAN) |
| Nimustine |
| Nimustine (INN) |
| Nimustine hydrochloride (JAN) <JP> |
| Ranimustine (JAN/INN) <JP> |
| Pentamustine (USAN); Neptamustine (INN) |
| Epoxide |
| Etoglucid (INN) |
| Asperlin (USAN) |
| Epipropidine (USAN/INN) |
| Teroxirone (USAN) |
| Omtriptolide sodium (USAN) |
| Dianhydrogalactitol (USAN/INN) |
| Mitobronitol (JAN/INN) |
| Pipobroman (JAN/USAN/INN) |
| Temozolomide (JP18/USAN/INN) <JP/US> |
| Dacarbazine |
| Dacarbazine (JAN/USP/INN) <JP/US> |
| Dacarbazine citrate |
| Laromustine (USAN) |