KEGG   Homo sapiens (human): 6869
Entry
6869              CDS       T01001                                 
Symbol
TACR1, NK1R, NKIR, SPR, TAC1R
Name
(RefSeq) tachykinin receptor 1
  KO
K04222  tachykinin receptor 1
Organism
hsa  Homo sapiens (human)
Pathway
hsa04020  Calcium signaling pathway
hsa04080  Neuroactive ligand-receptor interaction
hsa04082  Neuroactive ligand signaling
Network
nt06528  Calcium signaling
nt06544  Neuroactive ligand signaling
  Element
N01640  GPCR-PLCB-ITPR signaling pathway
N01915  Tachykinin receptor signaling
Drug target
Aprepitant (DG00066): D02968<JP/US> D06597<JP/US> D10895
Befetupitant: D03221
Casopitant: D06574
Elinzanetant: D12123
Ezlopitant: D04122
Maropitant citrate: D04860
Netupitant (DG02843): D05152 D11065 D11370<JP>
Orvepitant (DG01315): D09650 D09651
Rolapitant (DG01868): D08988<US> D10742
Serlopitant: D09378
Telmapitant: D10391
Tradipitant: D11728
Vestipitant mesylate: D06293
Vofopitant dihydrochloride: D06317
Brite
KEGG Orthology (KO) [BR:hsa00001]
 09130 Environmental Information Processing
  09132 Signal transduction
   04020 Calcium signaling pathway
    6869 (TACR1)
  09133 Signaling molecules and interaction
   04080 Neuroactive ligand-receptor interaction
    6869 (TACR1)
   04082 Neuroactive ligand signaling
    6869 (TACR1)
 09180 Brite Hierarchies
  09183 Protein families: signaling and cellular processes
   04030 G protein-coupled receptors [BR:hsa04030]
    6869 (TACR1)
G protein-coupled receptors [BR:hsa04030]
 Rhodopsin family
  Peptide
   Tachykinin
    6869 (TACR1)
SSDB
Motif
Pfam: 7tm_1 7tm_4
Other DBs
NCBI-GeneID: 6869
NCBI-ProteinID: NP_001049
OMIM: 162323
HGNC: 11526
Ensembl: ENSG00000115353
UniProt: P25103
Structure
LinkDB
Position
2:complement(75046463..75199520)
AA seq 407 aa
MDNVLPVDSDLSPNISTNTSEPNQFVQPAWQIVLWAAAYTVIVVTSVVGNVVVMWIILAH
KRMRTVTNYFLVNLAFAEASMAAFNTVVNFTYAVHNEWYYGLFYCKFHNFFPIAAVFASI
YSMTAVAFDRYMAIIHPLQPRLSATATKVVICVIWVLALLLAFPQGYYSTTETMPSRVVC
MIEWPEHPNKIYEKVYHICVTVLIYFLPLLVIGYAYTVVGITLWASEIPGDSSDRYHEQV
SAKRKVVKMMIVVVCTFAICWLPFHIFFLLPYINPDLYLKKFIQQVYLAIMWLAMSSTMY
NPIIYCCLNDRFRLGFKHAFRCCPFISAGDYEGLEMKSTRYLQTQGSVYKVSRLETTIST
VVGAHEEEPEDGPKATPSSLDLTSNCSSRSDSKTMTESFSFSSNVLS
NT seq 1224 nt   +upstreamnt  +downstreamnt
atggataacgtcctcccggtggactcagacctctccccaaacatctccactaacacctcg
gaacccaatcagttcgtgcaaccagcctggcaaattgtcctttgggcagctgcctacacg
gtcattgtggtgacctctgtggtgggcaacgtggtagtgatgtggatcatcttagcccac
aaaagaatgaggacagtgacgaactattttctggtgaacctggccttcgcggaggcctcc
atggctgcattcaatacagtggtgaacttcacctatgctgtccacaacgaatggtactac
ggcctgttctactgcaagttccacaacttctttcccatcgccgctgtcttcgccagtatc
tactccatgacggctgtggcctttgataggtacatggccatcatacatcccctccagccc
cggctgtcagccacagccaccaaagtggtcatctgtgtcatctgggtcctggctctcctg
ctggccttcccccagggctactactcaaccacagagaccatgcccagcagagtcgtgtgc
atgatcgaatggccagagcatccgaacaagatttatgagaaagtgtaccacatctgtgtg
actgtgctgatctacttcctccccctgctggtgattggctatgcatacaccgtagtggga
atcacactatgggccagtgagatccccggggactcctctgaccgctaccacgagcaagtc
tctgccaagcgcaaggtggtcaaaatgatgattgtcgtggtgtgcaccttcgccatctgc
tggctgcccttccacatcttcttcctcctgccctacatcaacccagatctctacctgaag
aagtttatccagcaggtctacctggccatcatgtggctggccatgagctccaccatgtac
aaccccatcatctactgctgcctcaatgacaggttccgtctgggcttcaagcatgccttc
cggtgctgccccttcatcagcgccggcgactatgaggggctggaaatgaaatccacccgg
tatctccagacccagggcagtgtgtacaaagtcagccgcctggagaccaccatctccaca
gtggtgggggcccacgaggaggagccagaggacggccccaaggccacaccctcgtccctg
gacctgacctccaactgctcttcacgaagtgactccaagaccatgacagagagcttcagc
ttctcctccaatgtgctctcctag

KEGG   Homo sapiens (human): 6865
Entry
6865              CDS       T01001                                 
Symbol
TACR2, NK2R, NKNAR, SKR, TAC2R
Name
(RefSeq) tachykinin receptor 2
  KO
K04223  tachykinin receptor 2
Organism
hsa  Homo sapiens (human)
Pathway
hsa04020  Calcium signaling pathway
hsa04080  Neuroactive ligand-receptor interaction
hsa04082  Neuroactive ligand signaling
Network
nt06528  Calcium signaling
nt06544  Neuroactive ligand signaling
  Element
N01640  GPCR-PLCB-ITPR signaling pathway
N01915  Tachykinin receptor signaling
Brite
KEGG Orthology (KO) [BR:hsa00001]
 09130 Environmental Information Processing
  09132 Signal transduction
   04020 Calcium signaling pathway
    6865 (TACR2)
  09133 Signaling molecules and interaction
   04080 Neuroactive ligand-receptor interaction
    6865 (TACR2)
   04082 Neuroactive ligand signaling
    6865 (TACR2)
 09180 Brite Hierarchies
  09183 Protein families: signaling and cellular processes
   04030 G protein-coupled receptors [BR:hsa04030]
    6865 (TACR2)
G protein-coupled receptors [BR:hsa04030]
 Rhodopsin family
  Peptide
   Tachykinin
    6865 (TACR2)
SSDB
Motif
Pfam: 7tm_1 7TM_GPCR_Srsx 7tm_4
Other DBs
NCBI-GeneID: 6865
NCBI-ProteinID: NP_001048
OMIM: 162321
HGNC: 11527
Ensembl: ENSG00000075073
UniProt: P21452
Structure
LinkDB
Position
10:complement(69403903..69416918)
AA seq 398 aa
MGTCDIVTEANISSGPESNTTGITAFSMPSWQLALWATAYLALVLVAVTGNAIVIWIILA
HRRMRTVTNYFIVNLALADLCMAAFNAAFNFVYASHNIWYFGRAFCYFQNLFPITAMFVS
IYSMTAIAADRYMAIVHPFQPRLSAPSTKAVIAGIWLVALALASPQCFYSTVTMDQGATK
CVVAWPEDSGGKTLLLYHLVVIALIYFLPLAVMFVAYSVIGLTLWRRAVPGHQAHGANLR
HLQAMKKFVKTMVLVVLTFAICWLPYHLYFILGSFQEDIYCHKFIQQVYLALFWLAMSST
MYNPIIYCCLNHRFRSGFRLAFRCCPWVTPTKEDKLELTPTTSLSTRVNRCHTKETLFMA
GDTAPSEATSGEAGRPQDGSGLWFGYGLLAPTKTHVEI
NT seq 1197 nt   +upstreamnt  +downstreamnt
atggggacctgtgacattgtgactgaagccaatatctcatctggccctgagagcaacacc
acgggcatcacagccttctccatgcccagctggcaactggcactgtgggccacagcctac
ctggccctggtgctggtggccgtgacgggtaatgccatcgtcatctggatcatcctggcc
catcggaggatgcgcacagtcaccaactacttcatcgtcaatctggcgctggctgacctc
tgcatggctgccttcaatgccgccttcaactttgtctatgccagccacaacatctggtac
tttggccgtgccttctgctacttccagaacctcttccccatcacagccatgtttgtcagc
atctactccatgaccgccattgctgccgacaggtacatggccatcgtccaccccttccag
cctcggctttcagctcccagcaccaaggcggttattgctggcatctggctggtggctctc
gccctggcctcccctcagtgcttctactccaccgtcaccatggaccagggtgccaccaag
tgcgtggtggcctggcccgaagacagcgggggcaagacgctcctcctgtaccacctcgtg
gtgatcgccctcatctacttcctgccgctcgcggtgatgtttgtagcctacagcgtcatc
ggcctcacgctctggaggcgcgcagtgcccggacatcaggcgcacggtgccaacctgcgc
cacctgcaggccatgaagaagtttgtgaagaccatggtgctggtggtgctgacgtttgcc
atctgctggctgccctaccacctctacttcatcctgggcagcttccaggaggacatctac
tgccacaagttcatccagcaagtctacctggcactcttctggttggccatgagctctacc
atgtacaatcccatcatctactgctgtctcaaccacaggtttcgctctggattccggctt
gccttccgctgctgcccatgggtcacacccaccaaggaagataagctcgagctgactccc
acgacctccctctccacgagagtcaacaggtgtcacactaaggagactttgttcatggct
ggggacacagccccctccgaggctaccagtggggaggcggggcgtccccaggatggatca
gggctatggtttgggtatggtttgcttgcccccaccaaaactcatgttgaaatttga

KEGG   Homo sapiens (human): 6870
Entry
6870              CDS       T01001                                 
Symbol
TACR3, HH11, NK-3R, NK3, NK3R, NKR, TAC3R, TAC3RL
Name
(RefSeq) tachykinin receptor 3
  KO
K04224  tachykinin receptor 3
Organism
hsa  Homo sapiens (human)
Pathway
hsa04020  Calcium signaling pathway
hsa04080  Neuroactive ligand-receptor interaction
hsa04082  Neuroactive ligand signaling
Network
nt06323  KISS1-GnRH-LH/FSH-E2 signaling
nt06528  Calcium signaling
nt06544  Neuroactive ligand signaling
  Element
N00882  TAC3-TACR3-PLC-PKC signaling pathway
N01640  GPCR-PLCB-ITPR signaling pathway
N01915  Tachykinin receptor signaling
Disease
H00255  Hypogonadotropic hypogonadism
Drug target
Elinzanetant: D12123
Fezolinetant: D11976<US>
Pavinetant: D11345
Talnetant hydrochloride: D05996
Brite
KEGG Orthology (KO) [BR:hsa00001]
 09130 Environmental Information Processing
  09132 Signal transduction
   04020 Calcium signaling pathway
    6870 (TACR3)
  09133 Signaling molecules and interaction
   04080 Neuroactive ligand-receptor interaction
    6870 (TACR3)
   04082 Neuroactive ligand signaling
    6870 (TACR3)
 09180 Brite Hierarchies
  09183 Protein families: signaling and cellular processes
   04030 G protein-coupled receptors [BR:hsa04030]
    6870 (TACR3)
G protein-coupled receptors [BR:hsa04030]
 Rhodopsin family
  Peptide
   Tachykinin
    6870 (TACR3)
SSDB
Motif
Pfam: 7tm_1 7TM_GPCR_Srsx 7tm_4 Ourmia_CP
Other DBs
NCBI-GeneID: 6870
NCBI-ProteinID: NP_001050
OMIM: 162332
HGNC: 11528
Ensembl: ENSG00000169836
UniProt: P29371
Structure
LinkDB
Position
4:complement(103586031..103719985)
AA seq 465 aa
MATLPAAETWIDGGGGVGADAVNLTASLAAGAATGAVETGWLQLLDQAGNLSSSPSALGL
PVASPAPSQPWANLTNQFVQPSWRIALWSLAYGVVVAVAVLGNLIVIWIILAHKRMRTVT
NYFLVNLAFSDASMAAFNTLVNFIYALHSEWYFGANYCRFQNFFPITAVFASIYSMTAIA
VDRYMAIIDPLKPRLSATATKIVIGSIWILAFLLAFPQCLYSKTKVMPGRTLCFVQWPEG
PKQHFTYHIIVIILVYCFPLLIMGITYTIVGITLWGGEIPGDTCDKYHEQLKAKRKVVKM
MIIVVMTFAICWLPYHIYFILTAIYQQLNRWKYIQQVYLASFWLAMSSTMYNPIIYCCLN
KRFRAGFKRAFRWCPFIKVSSYDELELKTTRFHPNRQSSMYTVTRMESMTVVFDPNDADT
TRSSRKKRATPRDPSFNGCSRRNSKSASATSSFISSPYTSVDEYS
NT seq 1398 nt   +upstreamnt  +downstreamnt
atggccactctcccagcagcagaaacctggatagacgggggtggaggcgtgggtgcagac
gccgtgaacctgaccgcctcgctagctgccggggcggccacgggggcagttgagactggg
tggctgcaactgctggaccaagctggcaacctctcctcctccccttccgcgctgggactg
cctgtggcttcccccgcgccctcccagccctgggccaacctcaccaaccagttcgtgcag
ccgtcctggcgcatcgcgctctggtccctggcgtatggtgtggtggtggcagtggcagtt
ttgggaaatctcatcgtcatctggatcatcctggcccacaagcgcatgaggactgtcacc
aactacttccttgtgaacctggctttctccgacgcctccatggccgccttcaacacgttg
gtcaatttcatctacgcgcttcatagcgagtggtactttggcgccaactactgccgcttc
cagaacttctttcctatcacagctgtgttcgccagcatctactccatgacggccattgcg
gtggacaggtatatggctattattgatcccttgaaacccagactgtctgctacagcaacc
aagattgtcattggaagtatttggattctagcatttctacttgccttccctcagtgtctt
tattccaaaaccaaagtcatgccaggccgtactctctgctttgtgcaatggccagaaggt
cccaaacaacatttcacttaccatattatcgtcattatactggtgtactgtttcccattg
ctcatcatgggtattacatacaccattgttggaattactctctggggaggagaaatccca
ggagatacctgtgacaagtatcatgagcagctaaaggccaaaagaaaggttgtcaaaatg
atgattattgttgtcatgacatttgctatctgctggctgccctatcatatttacttcatt
ctcactgcaatctatcaacaactaaatagatggaaatacatccagcaggtctacctggct
agcttttggctggcaatgagctcaaccatgtacaatcccatcatctactgctgtctgaat
aaaagatttcgagctggcttcaagagagcatttcgctggtgtcctttcatcaaagtttcc
agctatgatgagctagagctcaagaccaccaggtttcatccaaaccggcaaagcagtatg
tacaccgtgaccagaatggagtccatgacagtcgtgtttgaccccaacgatgcagacacc
accaggtccagtcggaagaaaagagcaacgccaagagacccaagtttcaatggctgctct
cgcaggaattccaaatctgcctccgccacttcaagtttcataagctcaccctatacctct
gtggatgaatattcttaa

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