| Gefitinib (JP18/USAN/INN) <JP/US> |
| Erlotinib |
| Erlotinib (INN) |
| Erlotinib hydrochloride (JAN/USAN) <JP/US> |
| Afatinib |
| Afatinib (USAN/INN) |
| Afatinib dimaleate (USAN); Afatinib maleate (JAN) <JP/US> |
| Osimertinib mesylate (USAN); Osimertinib mesilate (JAN) <JP/US> |
| Rociletinib (USAN/INN) |
| Olmutinib |
| Olmutinib (USAN/INN) |
| Olmutinib hydrochloride (USAN) |
| Dacomitinib |
| Dacomitinib (INN) |
| Dacomitinib (USAN); Dacomitinib hydrate (JAN) <JP/US> |
| Icotinib |
| Lazertinib |
| Lazertinib (USAN) |
| Lazertinib mesilate hydrate (JAN) |
| Aumolertinib |
| Aumolertinib (USAN/INN) |
| Aumolertinib mesylate (USAN) |
| Cetuximab (USAN/INN); Cetuximab (genetical recombination) (JAN) <JP/US> |
| Panitumumab (USAN/INN); Panitumumab (genetical recombination) (JAN) <JP/US> |
| Necitumumab (USAN/INN); Necitumumab (genetical recombination) (JAN) <JP/US> |
| Amivantamab (USAN/INN); Amivantamab (genetical recombination) (JAN) <US> |
| Tuxobertinib (USAN/INN) |
| Sunvozertinib (USAN/INN) |
| Tigozertinib (USAN) |
| Pebezertinib (USAN) |