Homo sapiens (human): 1909
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Entry
1909 CDS
T01001
Symbol
EDNRA, ET-A, ETA, ETA-R, ETAR, ETRA, MFDA, hET-AR
Name
(RefSeq) endothelin receptor type A
KO
K04197
endothelin receptor type A
Organism
hsa
Homo sapiens (human)
Pathway
hsa04020
Calcium signaling pathway
hsa04022
cGMP-PKG signaling pathway
hsa04024
cAMP signaling pathway
hsa04080
Neuroactive ligand-receptor interaction
hsa04270
Vascular smooth muscle contraction
hsa04924
Renin secretion
hsa05200
Pathways in cancer
Network
nt06325
Hormone/cytokine signaling
nt06528
Calcium signaling
Element
N01640
GPCR-PLCB-ITPR signaling pathway
N01792
EDN-EDNR signaling pathway
Disease
H02126
Mandibulofacial dysostosis with alopecia
Drug target
Ambrisentan:
D07077
<JP/US>
Aprocitentan:
D11441
<US>
Atrasentan hydrochloride:
D03009
Bosentan (
DG00266
):
D01227
<JP/US>
D07538
Centhaquine (
DG03144
):
D11974
D11975
Clazosentan (
DG03076
):
D07682
<JP>
D11664
Edonentan:
D03953
Fandosentan potassium:
D04128
Macitentan:
D10135
<JP/US>
Sitaxentan (
DG00267
):
D07171
D08517
Sparsentan:
D11776
<US>
Zibotentan:
D07741
Brite
KEGG Orthology (KO) [BR:
hsa00001
]
09130 Environmental Information Processing
09132 Signal transduction
04020 Calcium signaling pathway
1909 (EDNRA)
04024 cAMP signaling pathway
1909 (EDNRA)
04022 cGMP-PKG signaling pathway
1909 (EDNRA)
09133 Signaling molecules and interaction
04080 Neuroactive ligand-receptor interaction
1909 (EDNRA)
09150 Organismal Systems
09152 Endocrine system
04924 Renin secretion
1909 (EDNRA)
09153 Circulatory system
04270 Vascular smooth muscle contraction
1909 (EDNRA)
09160 Human Diseases
09161 Cancer: overview
05200 Pathways in cancer
1909 (EDNRA)
09180 Brite Hierarchies
09183 Protein families: signaling and cellular processes
04030 G protein-coupled receptors [BR:
hsa04030
]
1909 (EDNRA)
G protein-coupled receptors [BR:
hsa04030
]
Rhodopsin family
Peptide
Endothelin
1909 (EDNRA)
BRITE hierarchy
SSDB
Ortholog
Paralog
Gene cluster
GFIT
Motif
Pfam:
7tm_1
7TM_GPCR_Srsx
DUF4149
Motif
Other DBs
NCBI-GeneID:
1909
NCBI-ProteinID:
NP_001948
OMIM:
131243
HGNC:
3179
Ensembl:
ENSG00000151617
UniProt:
P25101
Structure
PDB
LinkDB
All DBs
Position
4:147481097..147544954
Genome browser
AA seq
427 aa
AA seq
DB search
METLCLRASFWLALVGCVISDNPERYSTNLSNHVDDFTTFRGTELSFLVTTHQPTNLVLP
SNGSMHNYCPQQTKITSAFKYINTVISCTIFIVGMVGNATLLRIIYQNKCMRNGPNALIA
SLALGDLIYVVIDLPINVFKLLAGRWPFDHNDFGVFLCKLFPFLQKSSVGITVLNLCALS
VDRYRAVASWSRVQGIGIPLVTAIEIVSIWILSFILAIPEAIGFVMVPFEYRGEQHKTCM
LNATSKFMEFYQDVKDWWLFGFYFCMPLVCTAIFYTLMTCEMLNRRNGSLRIALSEHLKQ
RREVAKTVFCLVVIFALCWFPLHLSRILKKTVYNEMDKNRCELLSFLLLMDYIGINLATM
NSCINPIALYFVSKKFKNCFQSCLCCCCYQSKSLMTSVPMNGTSIQWKNHDQNNHNTDRS
SHKDSMN
NT seq
1284 nt
NT seq
+upstream
nt +downstream
nt
atggaaaccctttgcctcagggcatccttttggctggcactggttggatgtgtaatcagt
gataatcctgagagatacagcacaaatctaagcaatcatgtggatgatttcaccactttt
cgtggcacagagctcagcttcctggttaccactcatcaacccactaatttggtcctaccc
agcaatggctcaatgcacaactattgcccacagcagactaaaattacttcagctttcaaa
tacattaacactgtgatatcttgtactattttcatcgtgggaatggtggggaatgcaact
ctgctcaggatcatttaccagaacaaatgtatgaggaatggccccaacgcgctgatagcc
agtcttgcccttggagaccttatctatgtggtcattgatctccctatcaatgtatttaag
ctgctggctgggcgctggccttttgatcacaatgactttggcgtatttctttgcaagctg
ttcccctttttgcagaagtcctcggtggggatcaccgtcctcaacctctgcgctcttagt
gttgacaggtacagagcagttgcctcctggagtcgtgttcagggaattgggattcctttg
gtaactgccattgaaattgtctccatctggatcctgtcctttatcctggccattcctgaa
gcgattggcttcgtcatggtaccctttgaatataggggtgaacagcataaaacctgtatg
ctcaatgccacatcaaaattcatggagttctaccaagatgtaaaggactggtggctcttc
gggttctatttctgtatgcccttggtgtgcactgcgatcttctacaccctcatgacttgt
gagatgttgaacagaaggaatggcagcttgagaattgccctcagtgaacatcttaagcag
cgtcgagaagtggcaaaaacagttttctgcttggttgtaatttttgctctttgctggttc
cctcttcatttaagccgtatattgaagaaaactgtgtataacgagatggacaagaaccga
tgtgaattacttagtttcttactgctcatggattacatcggtattaacttggcaaccatg
aattcatgtataaaccccatagctctgtattttgtgagcaagaaatttaaaaattgtttc
cagtcatgcctctgctgctgctgttaccagtccaaaagtctgatgacctcggtccccatg
aacggaacaagcatccagtggaagaaccacgatcaaaacaaccacaacacagaccggagc
agccataaggacagcatgaactga
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