| Carboxamide antiepileptic |
| Carbamazepine (JP18/USP/INN) <JP/US> |
| Oxcarbazepine (JAN/USP/INN) <US> |
| Rufinamide (JAN/USP/INN) <JP/US> |
| Eslicarbazepine |
| Eslicarbazepine (USAN/INN) |
| Eslicarbazepine acetate (USAN) <US> |
| Lamotrigine (JAN/USP/INN) <JP/US> |
| Zonisamide (JP18/USP/INN) <JP/US> |
| Lacosamide (JAN/USAN/INN) <JP/US> |
| Piracetam antiepileptic |
| Levetiracetam (JAN/USP/INN) <JP/US> |
| Brivaracetam (JAN/USAN/INN) <US> |
| Seletracetam (USAN/INN) |
| AMPA receptor antagonist |
| Topiramate (JAN/USP/INN) <JP/US> |
| Perampanel |
| Perampanel (USAN) |
| Perampanel hydrate (JAN) <JP/US> |
| Tezampanel (USAN) |
| Zonampanel (INN/USAN) |
| Hydantoin antiepileptic |
| Ethotoin (JAN/USP/INN) <JP> |
| Phenytoin |
| Phenytoin (JP18/USP/INN) <JP/US> |
| Phenytoin sodium (USP); Phenytoin sodium for injection (JP18) <JP/US> |
| Mephenytoin (USP/INN) |
| Fosphenytoin |
| Fosphenytoin (INN) |
| Fosphenytoin sodium (USP) <US> |
| Fosphenytoin sodium hydrate (JAN) <JP> |
| Albutoin (USAN/INN) |
| Methetoin (USAN/INN) |
| GABA mimetic antiepileptic |
| gamma-Aminobutyric acid (JAN) <JP> |
| Vigabatrin (JAN/USP/INN) <JP/US> |
| Progabide (USAN/INN) |
| Tiagabine |
| Tiagabine (INN) |
| Tiagabine hydrochloride (USP) <US> |
| Gabapentin |
| Gabapentin (JAN/USP/INN) <JP/US> |
| Gabapentin enacarbil (JAN/USAN/INN) <JP/US> |
| Pregabalin (JAN/USAN/INN) <JP/US> |
| Ezogabine (USAN); Retigabine (INN) |
| Tolgabide (USAN/INN) |
| Fatty acid antiepileptic |
| Valproic acid |
| Valproic acid (USP) <US> |
| Divalproex sodium (USP); Valproate semisodium (INN) <US> |
| Valproate sodium (USAN); Sodium valproate (JP18) <JP/US> |
| Calcium valproate |
| Valpromide (INN) |
| Valrocemide (USAN/INN) |
| Isovaleramide (USAN) |
| Milacemide hydrochloride (USAN) |
| Barbiturate antiepileptic |
| Mephobarbital (JAN/USP); Methylphenobarbital (INN) |
| Phenobarbital |
| Phenobarbital (JP18/USP/INN) <JP> |
| Phenobarbital sodium (JAN/USP/INN) <JP/US> |
| Phenobarbital diethylamine |
| Primidone (JP18/USP/INN) <JP/US> |
| Barbexaclone (INN) |
| Metharbital (JAN/INN) |
| Eterobarb (USAN/INN) |
| Benzodiazepine derivative, antiepileptic |
| Clonazepam (JP18/USP/INN) <JP/US> |
| Clobazam (JAN/USAN/INN) <JP/US> |
| Nitrazepam (JP18/USAN/INN) <JP> |
| Midazolam |
| Midazolam (JAN/USP/INN) <JP/US> |
| Midazolam hydrochloride (USAN) <US> |
| Midazolam maleate (USAN) |
| Diazepam (JP18/USP/INN) <JP/US> |
| Lorazepam (JP18/USP/INN) <JP/US> |
| Oxazolidine antiepileptic |
| Paramethadione (INN) |
| Trimethadione (JP18/INN) <JP> |
| Dimethadione (USAN/INN) |
| Succinimide antiepileptic |
| Ethosuximide (JP18/USP/INN) <JP/US> |
| Phensuximide (USP/INN) |
| Methsuximide (USP); Mesuximide (INN) <US> |
| Sulthiame (USAN); Sultiame (JP18) <JP> |
| Stiripentol (JAN/USAN/INN) <JP> |
| Acetylpheneturide (JAN) <JP> |
| Potassium bromide (JP18/USP) <JP> |
| Sodium bromide (JP18) <JP> |
| Phenytoin and phenobarbital <JP> |