| C00220 |
Methylene blue; Methylthioninium chloride |
(P) unclassified |
| D00131 |
Disulfiram (JP19/USP/INN); Antabuse (TN) |
(P) CYP inhibition: CYP1A2 |
| D00186 |
Ciprofloxacin (JP19/USP/INN); Cipro (TN); Otiprio (TN) |
(P) CYP inhibition: CYP1A2 |
| D00210 |
Norfloxacin (JP19/USP/INN); Noroxin (TN) |
(P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 |
| D00224 |
Allopurinol (JP19/USP/INN); Zyloprim (TN) |
(P) CYP inhibition: CYP1A2 |
| D00310 |
Enoxacin (USAN/INN); Penetrex (TN) |
(P) CYP inhibition: CYP1A2 |
| D00318 |
Famotidine (JP19/USP/INN); Fluxid (TN); Pepcid (TN) |
(P) CYP inhibition: CYP1A2 |
| D00371 |
Theophylline (JP19); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) |
(P) Enzyme: CYP1A2 |
| D00528 |
Caffeine (USP); Anhydrous caffeine (JP19); Anhydrous caffeine (TN); Respia (TN) |
(P) Enzyme: CYP1A2 |
| D00707 |
Fomepizole (JAN/USAN/INN); Antizol (TN) |
(P) CYP inhibition: CYP1A2 |
| D00809 |
Amitriptyline hydrochloride (JP19/USP); Elavil (TN) |
(P) unclassified |
| D00811 |
Clomipramine hydrochloride (JP19/USP); Anafranil (TN) |
(P) unclassified |
| D00815 |
Imipramine hydrochloride (JP19/USP); Tofranil (TN) |
(P) unclassified |
| D00824 |
Fluvoxamine maleate (JP19/USP); Luvox (TN) |
(P) CYP inhibition: CYP1A2 |
| D00903 |
Diclofenac potassium (USP); Cambia (TN); Cataflam (TN); Zipsor (TN) |
(P) unclassified |
| D00904 |
Diclofenac sodium (JP19/USP); Solaraze (TN); Voltaren (TN) |
(P) unclassified |
| D00960 |
Anastrozole (JP19/USP/INN); Arimidex (TN) |
(P) CYP inhibition: CYP1A2 |
| D01028 |
Ticlopidine hydrochloride (JP19/USP); Ticlid (TN) |
(P) CYP inhibition: CYP1A2 |
| D01153 |
Pazufloxacin (JAN/INN) |
(P) CYP inhibition: CYP1A2 |
| D01224 |
Phenylpropanolamine hydrochloride (JAN/USP) |
(P) CYP inhibition: CYP1A2 |
| D01453 |
Caffeine hydrate (JP19); Caffeine monohydrate |
(P) Enzyme: CYP1A2 |
| D01531 |
Pipemidic acid hydrate (JP19); Karunomazin (TN) |
(P) CYP inhibition: CYP1A2 |
| D01712 |
Theophylline sodium acetate (JAN) |
(P) Enzyme: CYP1A2 |
| D02216 |
Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP19); Ciloxan (TN); Cipro (TN); Proquin XR (TN) |
(P) CYP inhibition: CYP1A2 |
| D02312 |
Methylene blue (USP); Methylthioninium chloride; Provayblue (TN) |
(P) CYP inhibition: CYP1A2 |
| D02748 |
Peginterferon alfa-2b (USAN/INN); Peginterferon alfa-2b (genetical recombination) (JAN); Pegintron (TN); Sylatron (TN) |
(P) CYP inhibition: CYP1A2 |
| D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP inhibition: CYP1A2 |
| D05024 |
Mibefradil dihydrochloride (USAN); Posicor (TN) |
(P) CYP inhibition: CYP1A2 |
| D05382 |
Pazufloxacin mesilate (JP19); Pazufloxacin methanesulfonate; Pasil (TN) |
(P) CYP inhibition: CYP1A2 |
| D05429 |
Aminophylline hydrate (JP19) |
(P) Enzyme: CYP1A2 |
| D05461 |
Enoxacin hydrate (JP19) |
(P) CYP inhibition: CYP1A2 |
| D05466 |
Phenylpropanolamine polistirex (USAN) |
(P) CYP inhibition: CYP1A2 |
| D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 |
| D06103 |
Theophylline (USP); Theophylline monohydrate; Accurbron (TN) |
(P) Enzyme: CYP1A2 |
| D06104 |
Theophylline sodium glycinate (USP); Asbron (TN) |
(P) Enzyme: CYP1A2 |
| D07448 |
Amitriptyline (INN); Laroxyl (TN) |
(P) unclassified |
| D07564 |
Allopurinol sodium; Aloprim (TN) |
(P) CYP inhibition: CYP1A2 |
| D07603 |
Caffeine citrate (USP); Cafcit (TN) |
(P) Enzyme: CYP1A2 |
| D07702 |
Ciprofloxacin lactate; Ciproxin (TN) |
(P) CYP inhibition: CYP1A2 |
| D07727 |
Clomipramine (INN); Anafranil (TN) |
(P) unclassified |
| D07816 |
Diclofenac (USAN/INN); Solaraze (TN); Zorvolex (TN) |
(P) unclassified |
| D07817 |
Diclofenac diethylamine; Voltaren Emulgel (TN) |
(P) unclassified |
| D07818 |
Diclofenac epolamine; Diclofenac hydroxyethylpyrrolidine; Flector (TN) |
(P) unclassified |
| D07819 |
Diclofenac calcium; Voltaren Actingo Extra (TN) |
(P) unclassified |
| D07984 |
Fluvoxamine (INN) |
(P) CYP inhibition: CYP1A2 |
| D08070 |
Imipramine (INN); Tofranil (TN) |
(P) unclassified |
| D08071 |
Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) |
(P) unclassified |
| D08217 |
Mibefradil (INN) |
(P) CYP inhibition: CYP1A2 |
| D08287 |
Norfloxacin nicotinate; Quinabic soluble powder (TN) [veterinary] |
(P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 |
| D08368 |
Phenylpropanolamine (INN); Fansia (TN) |
(P) CYP inhibition: CYP1A2 |
| D08379 |
Pipemidic acid (INN); Nuril (TN) |
(P) CYP inhibition: CYP1A2 |
| D08594 |
Ticlopidine (INN) |
(P) CYP inhibition: CYP1A2 |
| D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP inhibition: CYP1A2 |
| D10537 |
Methylthioninium chloride hydrate (JAN); Methylene blue (TN) |
(P) CYP inhibition: CYP1A2 |
| D10822 |
Ciprofloxacin hydrate (JAN); Ciprofloxacin hemiheptahydrate |
(P) CYP inhibition: CYP1A2 |
| D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) unclassified |
| D11027 |
Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) |
(P) unclassified |
| D11062 |
Osilodrostat phosphate (JAN/USAN); Isturisa (TN) |
(P) unclassified |
| D11708 |
Givosiran sodium (JAN); Givlaari (TN) |
(P) unclassified |
| D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) CYP inhibition: CYP1A2 |
| D12364 |
Taletrectinib adipate (JAN/USAN); Ibtrozi (TN) |
(P) unclassified |