| General anesthetics |
| Inhalational anaesthetics |
| Ether (JP18/USP) |
| Halogenated hydrocarbons |
| Halothane (JP18/USP/INN) |
| Enflurane (JP18/USP/INN) |
| Isoflurane (JP18/USP/INN) <JP/US> |
| Desflurane (JAN/USP/INN) <JP/US> |
| Sevoflurane (JP18/USAN/INN) <JP/US> |
| Methoxyflurane (USP/INN) |
| Aliflurane (USAN/INN) |
| Fluroxene (USAN) |
| Norflurane (USAN/INN) |
| Roflurane (USAN/INN) |
| Teflurane (USAN/INN) |
| Nitrous oxide (JP18/USP) <JP/US> |
| Nitrous oxide and oxygen |
| Barbiturate anesthetics |
| Methohexital |
| Methohexital (USP/INN) |
| Methohexital sodium (USP) <US> |
| Hexobarbital (JAN/INN) |
| Thiopental |
| Thiopental |
| Thiopental sodium (JP18/USP/INN) <JP> |
| Thiamylal |
| Thiamylal |
| Thiamylal sodium (JP18) <JP> |
| Opioid anesthetics |
| Fentanyl |
| Fentanyl (JAN/USP/INN) <JP/US> |
| Fentanyl citrate (JP18/USP) <JP/US> |
| Fentanyl hydrochloride (JAN) |
| Alfentanil |
| Alfentanil (INN) |
| Alfentanil hydrochloride (USP) |
| Sufentanil |
| Sufentanil (USAN/INN) |
| Sufentanil citrate (USP) <US> |
| Phenoperidine (INN) |
| Anileridine |
| Anileridine (USP/INN) |
| Anileridine hydrochloride (USP) |
| Remifentanil |
| Remifentanil (INN) |
| Remifentanil hydrochloride (JAN/USAN) <JP/US> |
| Droperidol and fentanyl citrate |
| Ketamine |
| Ketamine (INN) |
| Ketamine hydrochloride (JP18/USP) <JP/US> |
| Propanidid (USAN/INN) |
| Alfaxalone (INN) |
| Etomidate (USP/INN) <US> |
| Propofol |
| Propofol (JAN/USP/INN) <JP/US> |
| Fospropofol disodium (USAN) |
| Hydroxybutyric acid |
| 4-Hydroxybutanoic acid |
| Sodium oxybate (USAN) <US> |
| Local anesthetic |
| Esterified local anesthetic |
| Metabutethamine |
| Procaine |
| Procaine (INN) |
| Procaine hydrochloride (JP18/USP) <JP> |
| Tetracaine |
| Tetracaine (USP/INN) |
| Tetracaine hydrochloride (JP18/USP) <US> |
| Chloroprocaine |
| Chloroprocaine (INN) |
| Chloroprocaine hydrochloride (USP) <US> |
| Cocaine |
| Cocaine (USP) |
| Cocaine hydrochloride (JP18/USP) <US> |
| Aminobenzoic acid |
| Aminobenzoic acid (USP) |
| Benzocaine (USP/INN); Ethyl aminobenzoate (JP18) <JP> |
| Aminobenzoate potassium (USP) |
| Aminobenzoate sodium (USP) |
| Amide type local anesthetic |
| Bupivacaine |
| Bupivacaine (USAN/INN) <US> |
| Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18) <JP/US> |
| Lidocaine |
| Lidocaine (JP18/USP/INN) <JP/US> |
| Lidocaine hydrochloride (JAN/USP) <JP/US> |
| Lidocaine hydrochloride monohydrate <JP/US> |
| Mepivacaine |
| Mepivacaine (INN) |
| Mepivacaine hydrochloride (JP18/USP) <JP/US> |
| Prilocaine |
| Prilocaine (USP/INN); Propitocaine (JAN) |
| Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN) <US> |
| Butanilicaine (INN) |
| Dibucaine |
| Dibucaine (USP); Cinchocaine (INN) |
| Dibucaine hydrochloride (JP18/USP) |
| Etidocaine |
| Etidocaine (USAN/INN) |
| Etidocaine hydrochloride |
| Articaine |
| Articaine (INN) |
| Articaine hydrochloride (JAN/USP) |
| Ropivacaine |
| Ropivacaine (INN) |
| Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN) <JP/US> |
| Levobupivacaine |
| Levobupivacaine (INN) |
| Levobupivacaine hydrochloride (JAN/USAN) <JP> |
| Oxetacaine |
| Oxethazaine (JP18/USAN); Oxetacaine (INN) <JP> |
| Oxetacaine hydrochloride |
| Trimecaine |
| Trimecaine (INN) |
| Trimecaine hydrochloride |
| Tolycaine hydrochloride (JAN) |
| Dexivacaine (USAN/INN) |
| Pyrrocaine (USAN/INN) |
| Rodocaine (USAN) |
| Ethyl chloride (USP) |
| Dyclonine |
| Dyclonine (INN) |
| Dyclonine hydrochloride (USP) <US> |
| Phenol |
| Phenol (JP18/USP); Liquefied phenol (JP18); Phenol for disinfection (JP18) <JP> |
| Phenolated water (JP18); Phenolated water for disinfection (JP18) <JP> |
| Capsaicin (JAN/USP) <US> |
| Oxybuprocaine |
| Oxybuprocaine (INN) |
| Benoxinate hydrochloride (USP); Oxybuprocaine hydrochloride (JP18) <JP> |
| Proxymetacaine |
| Proxymetacaine (INN) |
| Proparacaine hydrochloride (USP) <US> |
| p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN); Diethylaminoethyl p-butylaminobenzoate hydrochloride (JAN) |