Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
   Cytokines
   Cytokine receptors
     Interleukin receptors
     Interferon receptors
     CSF and other factor receptors
     Chemokine receptors
     Tumor necrosis factor receptors
       TNFRSF1 (CD120) [HSA:7132 7133] [KO:K03158 K05141]
       TNFRSF4 (CD134, OX40) [HSA:7293] [KO:K05142]
       TNFRSF5 (CD40) [HSA:958] [KO:K03160]
       TNFRSF7 (CD27) [HSA:939] [KO:K05144]
       TNFRSF8 (CD30) [HSA:943] [KO:K05145]
         D09587  Brentuximab vedotin (USAN/INN) <JP/US>
         D04612  Iratumumab (USAN)
       TNFRSF9 (CD137) [HSA:3604] [KO:K05146]
       TNFRSF10A (TRAILR1, CD261) [HSA:8797] [KO:K04722]
       TNFRSF10B (TRAILR2, CD262) [HSA:8795] [KO:K04722]
       TNFRSF12A (TWEAKR, CD266) [HSA:51330] [KO:K05149]
       TNFRSF13B (CD267, TACI) [HSA:23495] [KO:K05150]
       TNFRSF13C (BAFF-R, CD268) [HSA:115650] [KO:K05151]
       TNFRSF18 [HSA:8784] [KO:K05154]
       NGFR (TNFRSF16, CD271) [HSA:4804] [KO:K02583]
       TNFRSF17 (BCMA, CD269) [HSA:608] [KO:K05153]
   Pattern recognition receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified
   Signaling molecules
   Cellular process
     Cell cycle
     Apoptosis
     Membrane trafficking
     Cytoskeleton
       MYL2 [HSA:4633] [KO:K10351]
       MYL3 [HSA:4634] [KO:K12749]
       MYL4 [HSA:4635] [KO:K12750]
       MYH6_7 [HSA:4624 4625] [KO:K17751]
       MYH7 [HSA:4625] [KO:K17751]
       TNNC1 [HSA:7134] [KO:K05865]
       TNNC2 [HSA:7125] [KO:K12042]
       TNNI2 [HSA:7136] [KO:K12043]
       TNNI3 [HSA:7137] [KO:K12044]
       TNNT2 [HSA:7139] [KO:K12045]
       TNNT3 [HSA:7140] [KO:K12046]
       DMD [HSA:1756] [KO:K10366]
       DMD* [HSA_VAR:1756v1] [HSA:1756] [KO:K10366]
       TUBB [HSA:10381 10382 10383 203068 347688 347733 7280 81027 84617] [KO:K07375]
         D11691  Tirbanibulin (USAN/INN) <US>
         D11692  Tirbanibulin mesylate (USAN)
         D08675  Vinblastine (INN)
         D01068  Vinblastine sulfate (JP18/USP) <JP/US>
         D08679  Vincristine (INN)
         D02197  Vincristine sulfate (JP18/USP) <JP/US>
         D06304  Vindesine (USAN/INN)
         D01769  Vindesine sulfate (JAN/USAN) <JP>
         D08680  Vinorelbine (INN)
         D01935  Vinorelbine tartrate (USP) <JP/US>
         D09032  Vinflunine ditartrate (USAN)
         D00491  Paclitaxel (JAN/USP/INN) <JP/US>
         D07866  Docetaxel (JAN/INN) <JP/US>
         D02165  Docetaxel (USP) <JP/US>
         D05333  Paclitaxel poliglumex (USAN/INN)
         D09755  Cabazitaxel (USAN/INN)
         D10452  Cabazitaxel acetonate (JAN) <JP/US>
         D04645  Ixabepilone (JAN/USAN/INN) <US>
         D09980  Trastuzumab emtansine (USAN/INN) <JP/US>
         D09587  Brentuximab vedotin (USAN/INN) <JP/US>
         D11525  Enfortumab vedotin (USAN) <JP/US>
         D11595  Belantamab mafodotin (USAN) <US>
         D11814  Tisotumab vedotin (USAN/INN) <US>
         D10954  Mirvetuximab soravtansine (USAN/INN) <US>
         D04066  Estramustine (USAN/INN)
         D02398  Estramustine phosphate sodium (USAN)
         D06397  Estramustine phosphate sodium hydrate (JAN) <JP/US>
         D08914  Eribulin mesylate (USAN) <JP/US>
         D00570  Colchicine (JP18/USP) <JP/US>
         D01919  Soblidotin (JAN/INN)
         D03059  Batabulin sodium (USAN)
         D03364  Cantuzumab mertansine (USAN)
         D04864  Maytansine (USAN)
         D05062  Mivobulin isethionate (USAN)
         D06001  Taltobulin (USAN/INN)
         D06009  Tasidotin hydrochloride (USAN)
         D06305  Vinepidine sulfate (USAN)
         D06306  Vinglycinate sulfate (USAN)
         D06307  Vinleurosine sulfate (USAN)
         D06308  Vinrosidine sulfate (USAN)
         D06309  Vinzolidine sulfate (USAN)
         D06560  Batabulin (USAN/INN)
         D06576  Cevipabulin fumarate (USAN)
         D08889  Cevipabulin succinate (USAN)
         D09691  Vedotin (USAN)
         D09912  Glembatumumab vedotin (USAN)
         D09927  Lorvotuzumab mertansine (USAN/INN)
         D10013  Indibulin (USAN/INN)
         D10029  Verubulin (USAN/INN)
         D10030  Verubulin hydrochloride (USAN)
         D10073  Lexibulin (USAN)
         D10454  Cantuzumab ravtansine (USAN/INN)
         D11228  Soravtansine (USAN)
         D11232  Denintuzumab mafodotin (USAN/INN)
         D11238  Lifastuzumab vedotin (USAN/INN)
         D11494  Lisavanbulin (USAN/INN)
         D11681  Avanbulin (USAN/INN)
         D12183  Farletuzumab ecteribulin (USAN)
         D12210  Ozuriftmab vedotin (USAN)
         D12220  Mecbotamab vedotin
         D12310  Tusamitamab ravtansine (USAN/INN)
         D12519  Sabizabulin (USAN/INN)
         D12520  Sabizabulin hydrochloride (USAN)
         D12582  Opadotin (USAN)
         D12583  Anvatabart opadotin (USAN/INN)
       KIF11 [HSA:3832] [KO:K10398]
       MAPT (TAU) [HSA:4137] [KO:K04380]
       FLNA [HSA:2316] [KO:K04437]
     Ubiquitin system
     Chromatin
     Cilia formation
   Organismal systems
   Unclassified

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Last updated: May 9, 2024

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